- PARP1
- PARP2
- PARP3
- Tankyrase-1
Tankyrase-1 抑制剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S1060 | Olaparib (AZD2281, Ku-0059436) | Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1/2 with IC50 of 5 nM/1 nM, 300-times less effective against tankyrase-1. Phase 3. | Pan | Tankyrase-1, IC50: 1.5 μM |
