BChE

BChE产品

所有产品(7)
BChE抑制剂 (7)
新BChE产品

目录号	产品名	产品描述
S0924	Pteryxin	Pteryxin ((+)-Pteryxin) 是一种在 Apiaceae 伞形科中发现的二氢吡喃香豆素衍生物，也是一种有效的 butyrylcholinesterase (BChE) 的抑制剂，IC50值为12.96 μg/ml。Pteryxin 可抑制LPS诱导的小鼠腹膜巨噬细胞中 nitric oxide 的产生，其IC50值为20 μM。Pteryxin 具有治疗阿尔茨海默氏病 (AD) 的潜力。
S3245	Nodakenetin	Nodakenetin (NANI) 是从Angelica decursiva中分离出的植物性香豆素，可抑制 α-glucosidase、PTP1B、rat lens aldose reductase (RLAR)、AChE、BChE 和 β-site amyloid precursor protein cleaving enzyme 1 (BACE1)。Nodakenetin 可改变 Bax 和 Bcl-2 的蛋白质表达，并促进线粒体凋亡。Nodakenetin 具有抗肿瘤活性。
S5665	Drofenine Hydrochloride	Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
S3835	Loganin	Loganin (Loganoside) is an iridoid glycoside first isolated from the seeds of Strychnos nux-vomica, a member of the Loganiaceae family. It is a non-competitive inhibitor of BACE1 with IC50 of 47.97 μM an also inhibits AChE and BChE with IC50 values of 3.95 μM and 33.02 μM, respectively.
E2237	Vasicine (hydrochloride)	Vasicine hydrochloride(Peganine hydrochloride)是一种从Adhatoda vasica中分离出来的生物碱vasicine (VAS)的盐，是一种潜在的天然胆碱酯酶抑制剂。VAS抑制乙酰胆碱酯酶(AChE)和丁酰胆碱酯酶(BChE)。
S5511	Ethyl (triphenylphosphoranylidene) acetate	Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
E0784	MAO-B-IN-2	MAO-B-in-2是MAO-B和BChE的选择性，竞争性抑制剂，其IC50分别为0.51和7.00 μM。
S0924	Pteryxin	Pteryxin ((+)-Pteryxin) 是一种在 Apiaceae 伞形科中发现的二氢吡喃香豆素衍生物，也是一种有效的 butyrylcholinesterase (BChE) 的抑制剂，IC50值为12.96 μg/ml。Pteryxin 可抑制LPS诱导的小鼠腹膜巨噬细胞中 nitric oxide 的产生，其IC50值为20 μM。Pteryxin 具有治疗阿尔茨海默氏病 (AD) 的潜力。
S3245	Nodakenetin	Nodakenetin (NANI) 是从Angelica decursiva中分离出的植物性香豆素，可抑制 α-glucosidase、PTP1B、rat lens aldose reductase (RLAR)、AChE、BChE 和 β-site amyloid precursor protein cleaving enzyme 1 (BACE1)。Nodakenetin 可改变 Bax 和 Bcl-2 的蛋白质表达，并促进线粒体凋亡。Nodakenetin 具有抗肿瘤活性。
S5665	Drofenine Hydrochloride	Drofenine hydrochloride is a potent competitive inhibitor of BChE. It is an anticholinergic that acts both at the level of the nerves and the muscle fibers.
S3835	Loganin	Loganin (Loganoside) is an iridoid glycoside first isolated from the seeds of Strychnos nux-vomica, a member of the Loganiaceae family. It is a non-competitive inhibitor of BACE1 with IC50 of 47.97 μM an also inhibits AChE and BChE with IC50 values of 3.95 μM and 33.02 μM, respectively.
E2237	Vasicine (hydrochloride)	Vasicine hydrochloride(Peganine hydrochloride)是一种从Adhatoda vasica中分离出来的生物碱vasicine (VAS)的盐，是一种潜在的天然胆碱酯酶抑制剂。VAS抑制乙酰胆碱酯酶(AChE)和丁酰胆碱酯酶(BChE)。
S5511	Ethyl (triphenylphosphoranylidene) acetate	Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
E0784	MAO-B-IN-2	MAO-B-in-2是MAO-B和BChE的选择性，竞争性抑制剂，其IC50分别为0.51和7.00 μM。

BChE抑制剂选择性比较