- serine/threonine kinase
- STK
- WNK
- DCLK
- GCN
- GAK
- SRPK
- PASK
- BUB1
DCLK 选择性抑制剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S8976 | DCLK1-IN-1 | DCLK1-IN-1 is a selective, in vivo-compatible chemical probe of the doublecortin like kinase 1 (DCLK1) domain that binds to DCLK1 and DCLK2 with IC50 of 9.5 nM and 31 nM, respectively. DCLK1-IN-1 inhibits DCLK1 and DCLK2 kinases with IC50 of 57.2 nM and 103 nM in kinase assay, respectively. | Selective | DCLK1, IC50: 9.5 nM; DCLK2, IC50: 31 nM; DCLK1, IC50: 57.2 nM; DCLK2, IC50: 103 nM |
