RORα
RORγ

RORalpha 选择性激动剂

目录号	产品名	产品描述	Selective / Pan	IC50 / Ki
S2654	Neoruscogenin	Neoruscogenin, a natural sapogenin isolated from R. rhizoma, is a potent and high-affinity agonist of RAR-related orphan receptor alpha (RORα or nuclear receptor NR1F1).	Selective
S2969	SR3335	SR3335 (ML-176) is a selective and inverse agonist of retinoic acid receptor-related receptor α (RORα) that directly binds to RORα with Ki of 220 nM.	Selective	RORα, Ki: 220 nM
S5775	SR1078	SR1078, a synthetic ligand for RORα and RORγ, functions as a RORα/γ agonist.	Pan
S6724	SR1001	SR1001 is a RORα inverse agonist with Ki values of 172 nM and 111 nM for RORα and RORγ respectively.	Pan	RORα, Ki: 172 nM