WDR5

WDR5产品

  • 所有产品(2)
  • WDR5抑制剂 (1)
  • WDR5拮抗剂 (1)
目录号 产品名 产品描述 文献引用 实验数据
S7833 OICR-9429 OICR-9429是一种有效的WDR5-MLLWDR5-Histone3相互作用的拮抗剂,能在体外实验中降低急性髓性白血病细胞的活性。它与WDR5高亲和结合,Kd值为93 ± 28 nM。
Journal of Experimental & Clinical Cancer Research, June 21, 2021, 203
iScience, December 25, 2021, 103679
FASEB Journal, April 30, 2025, e70543
S2184 WDR5-0103 WDR5-0103 (WD-Repeat Protein 5-0103)是一种WDR5 (WD40 repeat protein 5)的小分子拮抗剂,Kd值为450 nM。
Cell Reports, September 26, 2023, 113145
Journal of Clinical Investigation, July 3, 2023, e169993
Frontiers in Immunology, August 9, 2022, 938944
S7833 OICR-9429 OICR-9429是一种有效的WDR5-MLLWDR5-Histone3相互作用的拮抗剂,能在体外实验中降低急性髓性白血病细胞的活性。它与WDR5高亲和结合,Kd值为93 ± 28 nM。
Journal of Experimental & Clinical Cancer Research, June 21, 2021, 203
iScience, December 25, 2021, 103679
FASEB Journal, April 30, 2025, e70543
S2184 WDR5-0103 WDR5-0103 (WD-Repeat Protein 5-0103)是一种WDR5 (WD40 repeat protein 5)的小分子拮抗剂,Kd值为450 nM。
Cell Reports, September 26, 2023, 113145
Journal of Clinical Investigation, July 3, 2023, e169993
Frontiers in Immunology, August 9, 2022, 938944
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