Paclitaxel

别名: NSC 125973，PTX 中文名称：紫杉醇

目录号：S1150 Purity: 99.99%

Paclitaxel是一种microtubule聚合物稳定剂，在人内皮细胞中IC50为0.1 pM。Paclitaxel可引起有丝分裂停滞和细胞凋亡。 Paclitaxel还会诱导自噬。

Paclitaxel Chemical Structure

CAS: 33069-62-4

规格	价格	库存
10mM (1mL in DMSO)	749.07	现货
10mg	571.49	现货
50mg	1711.71	现货
100mg	2694.51	现货
1g	7944.3	现货
更大包装有超大折扣
400-668-6834 info@selleck.cn

产品质控

批次：纯度： 99.99%

99.99

Paclitaxel相关产品

相关产品	Puromycin 2HCl Staurosporine (STS) Oligomycin A Geldanamycin Honokiol Geneticin (G418 Sulfate) Nigericin sodium salt STZ (Streptozotocin) Cephalomannine Sodium Monensin (NSC 343257) 10-Deacetylbaccatin-III Pirarubicin Hygromycin B Roxithromycin	点击展开
相关化合物库	激酶抑制剂库血管生成相关化合物库 TGF-beta/Smad信号通路库细胞骨架信号通路化合物库抗心血管疾病化合物库	点击展开

细胞实验数据示例

细胞系	实验类型	孵育时间	活性描述	文献信息
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.002 μM	11325226
SW626	Cytotoxicity assay	72 h	IC50 = 0.00001 μM	12088425
Lu1	Cytotoxicity assay	72 h	IC50 = 0.01 μM	12088425
MCF7	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
P388	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
LNCAP	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
KB	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
Col2	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
BC1	Cytotoxicity assay	72 h	IC50 = 0.02 μM	12088425
SK-MEL-2	Cytotoxicity assay	72 h	IC50 = 0.07 μM	12088425
NCI-H460	Cytotoxicity assay	48 h	IC50 = 0.0095 μM	14695798
MCF7	Cytotoxicity assay	48 h	IC50 = 0.0112 μM	14695798
SF268	Cytotoxicity assay	48 h	IC50 = 0.0217 μM	14695798
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 0.0045 μM	14987051
MCF7	Cytotoxicity assay	48 h	IC50 = 0.0049 μM	14987051
A2780	Cytotoxicity assay	48 h	IC50 = 0.025 μM	14987051
PC3	Cytotoxicity assay	48 h	IC50 = 0.077 μM	14987051
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0014 μM	14987056
multidrug-resistant MCF7	Cytotoxicity assay	72 h	IC50 = 0.354 μM	14987056
PC3	Cytotoxicity assay	48 h	IC50 = 0.016 μM	15043402
Hep3B	Cytotoxicity assay	48 h	IC50 = 0.031 μM	15043402
NCI-H460	Cytotoxicity assay	48 h	IC50 = 0.0095 μM	15043404
MCF7	Cytotoxicity assay	48 h	IC50 = 0.0112 μM	15043404
SF268	Cytotoxicity assay	48 h	IC50 = 0.0217 μM	15043404
T47D	Apoptosis assay	24 h	EC50 = 0.03 μM	15566300
DLD1	Apoptosis assay	24 h	EC50 = 0.075 μM	15566300
H1299	Apoptosis assay	24 h	EC50 = 0.163 μM	15566300
VA13	Cytotoxicity assay	48 h	IC50 = 0.005 μM	15730243
WI 38	Cytotoxicity assay	48 h	IC50 = 0.04 μM	15730243
Hep G2	Cytotoxicity assay	48 h	IC50 = 8.1 μM	15730243
A549	Cytotoxicity assay	48 h	IC50 = 1.25 μM	15787460
SKOV3	Cytotoxicity assay	48 h	IC50 = 1.35 μM	15787460
KB	Cytotoxicity assay	3 days	IC50 = 0.001 μM	16038545
1A9	Cytotoxicity assay	3 days	IC50 = 0.002 μM	16038545
HCT8	Cytotoxicity assay	3 days	IC50 = 0.013 μM	16038545
VA13	Growth inhibition assay	48 h	IC50 = 0.0043 μM	16499322
WI38	Growth inhibition assay	48 h	IC50 = 0.034 μM	16499322
HepG2	Growth inhibition assay	48 h	IC50 = 6.9 μM	16499322
U937 GTB	Cytotoxicity assay	72 h	IC50 = 0.0059 μM	16562840
RPMI 8226/s	Cytotoxicity assay	72 h	IC50 = 0.007 μM	16562840
CEM/s	Cytotoxicity assay	72 h	IC50 = 0.007 μM	16562840
LT12	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	17181164
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	17181164
NCI-H460	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	17181164
SF268	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	17181164
RKO	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	17181164
KB/HeLa	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	17181164
P388	Antiproliferative activity assay	48 h	IC50 = 0.04 μM	17181164
L1210	Antiproliferative activity assay	48 h	IC50 = 0.06 μM	17181164
LT12 MDR	Antiproliferative activity assay	48 h	IC50 = 0.4 μM	17181164
NCI-H1299	Cytotoxicity assay	96 h	IC50 = 0.015 μM	17419065
HT29	Growth inhibition assay	48 h	GI50 = 0.015 μM	17498960
M21	Growth inhibition assay	48 h	GI50 = 0.037 μM	17498960
MCF7	Growth inhibition assay	48 h	GI50 = 0.054 μM	17498960
1A9	Growth inhibition assay	72 h	GI50 = 0.00071 μM	17542572
1A9/Ptx22	Growth inhibition assay	72 h	GI50 = 0.051 μM	17542572
1A9/Ptx10	Growth inhibition assay	72 h	GI50 = 0.064 μM	17542572
HL60	Cytotoxicity assay	72 h	IC50 = 0.93 μM	17896816
P388	Cytotoxicity assay	72 h	IC50 = 0.93 μM	17896816
BEL-7402	Cytotoxicity assay	24 h	IC50 = 0.93 μM	17896816
A459	Cytotoxicity assay	24 h	IC50 = 0.93 μM	17896816
Aro	Cytotoxicity assay	72 h	IC50 = 0.0002 μM	17915851
PT45	Cytotoxicity assay	72 h	IC50 = 0.005 μM	17915851
A549	Cytotoxicity assay	72 h	IC50 = 0.006 μM	17915851
MCF7	Cytotoxicity assay	72 h	IC50 = 0.007 μM	17915851
HeLa	Cytotoxicity assay	72 h	IC50 = 0.008 μM	17915851
Ovcar3	Cytotoxicity assay	72 h	IC50 = 0.01 μM	17915851
HT29	Cytotoxicity assay	72 h	IC50 = 0.05 μM	17915851
A549T12	Cytotoxicity assay	72 h	IC50 = 0.06 μM	17915851
H295R	Cytotoxicity assay	72 h	IC50 = 0.08 μM	17915851
A549T24	Cytotoxicity assay	72 h	IC50 = 0.102 μM	17915851
OE33	Cytotoxicity assay	72 h	IC50 = 0.2 μM	17915851
HepG2	Cytotoxicity assay	72 h	IC50 = 0.3 μM	17915851
OE19	Cytotoxicity assay	72 h	IC50 = 0.4 μM	17915851
L12	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	17973361
NCI-H460	Cytotoxicity assay	48 h	IC50 = 0.01 μM	17973361
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.01 μM	17973361
SF268	Cytotoxicity assay	48 h	IC50 = 0.01 μM	17973361
RKO	Cytotoxicity assay	48 h	IC50 = 0.01 μM	17973361
KB/HeLa	Cytotoxicity assay	48 h	IC50 = 0.01 μM	17973361
P388	Antiproliferative activity assay	48 h	IC50 = 0.04 μM	17973361
L1210	Antiproliferative activity assay	48 h	IC50 = 0.06 μM	17973361
PANC1	Cytotoxicity assay	72 h	IC50 = 0.007 μM	18081257
DLD1	Cytotoxicity assay	72 h	IC50 = 0.011 μM	18081257
AsPC1	Cytotoxicity assay	72 h	IC50 = 0.02 μM	18081257
NCI/ADR	Cytotoxicity assay	72 h	IC50 = 1 μM	18081257
SK-BR3	Antiproliferative activity assay	96 h	GI50 = 6.1 μM	18164205
A2780	Antiproliferative activity assay	96 h	IC50 = 0.0234 μM	18177014
SNU398	Apoptosis assay	24 h	EC50 = 0.011 μM	18197614
HCT116	Apoptosis assay	24 h	EC50 = 0.024 μM	18197614
T47D	Apoptosis assay	24 h	EC50 = 0.036 μM	18197614
SJSA1	Cytotoxicity assay	6 h	IC50 = 0.0032 μM	18243696
P388	Cytotoxicity assay	72 h	IC50 = 0.93 μM	18281952
HL60	Cytotoxicity assay	72 h	IC50 = 0.93 μM	18281952
Bel7402	Cytotoxicity assay	24 h	IC50 = 0.93 μM	18281952
A549	Cytotoxicity assay	24 h	IC50 = 0.93 μM	18281952
KB	Cytotoxicity assay	48 h	IC50 = 0.0042 μM	18295490
KBV20C	Cytotoxicity assay	48 h	IC50 = 1.44 μM	18295490
DU145	Cytotoxicity assay	72 h	IC50 = 0.005 μM	18308566
HL60	Cytotoxicity assay	72 h	IC50 = 0.005 μM	18308566
MDA435	Cytotoxicity assay	72 h	IC50 = 0.005 μM	18308566
MESSA	Cytotoxicity assay	72 h	IC50 = 0.005 μM	18308566
P388	Cytotoxicity assay	72 h	IC50 = 0.01 μM	18308566
HL60/TX1000	Cytotoxicity assay	72 h	IC50 = 5 μM	18308566
MESSA/DX5	Cytotoxicity assay	72 h	IC50 = 5 μM	18308566
K562	Growth inhibition assay	72 h	IC50 = 0.0006 μM	18313307
KB3-1	Growth inhibition assay	72 h	IC50 = 0.002 μM	18313307
HepG2	Growth inhibition assay	72 h	IC50 = 0.007 μM	18313307
KB V1	Growth inhibition assay	72 h	IC50 = 8 μM	18313307
A549	Cytotoxicity assay	3 days	IC50 = 0.007 μM	18419154
MCF7	Cytotoxicity assay	3 days	IC50 = 0.0117 μM	18419154
HepG2	Cytotoxicity assay	3 days	IC50 = 0.0468 μM	18419154
MDA-MB-231	Cytotoxicity assay	3 days	IC50 = 0.0703 μM	18419154
Hep3B	Cytotoxicity assay	3 days	IC50 = 0.13 μM	18419154
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.001274 μM	18450456
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0013 μM	18450456
MX1	Cytotoxicity assay	72 h	IC50 = 0.035 μM	18450456
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0015 μM	18461997
HT29	Antiproliferative activity assay	48 h	IC50 = 0.0019 μM	18461997
U2OS	Antiproliferative activity assay	48 h	IC50 = 0.024 μM	18461997
A2780	Cytotoxicity assay	72 h	IC50 = 0.00138 μM	18465846
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0017 μM	18465846
LCC6	Cytotoxicity assay	72 h	IC50 = 0.0031 μM	18465846
1A9PTX22	Cytotoxicity assay	72 h	IC50 = 0.1607 μM	18465846
NCI/ADR	Cytotoxicity assay	72 h	IC50 = 0.3 μM	18465846
1A9PTX10	Cytotoxicity assay	72 h	IC50 = 0.53295 μM	18465846
HepG2	Growth inhibition assay	72 h	IC50 = 0.0059 μM	18512984
HepG2/Dox	Growth inhibition assay	72 h	IC50 = 1.4 μM	18512984
HT29	Growth inhibition assay	48 h	GI50 = 0.015 μM	18579387
M21	Growth inhibition assay	48 h	GI50 = 0.037 μM	18579387
MCF7	Growth inhibition assay	48 h	GI50 = 0.054 μM	18579387
KB403	Cytotoxicity assay	24 h	IC50 = 0.001 μM	18586491
WRL68	Cytotoxicity assay	24 h	IC50 = 0.004 μM	18586491
MCF7	Cytotoxicity assay	24 h	IC50 = 0.006 μM	18586491
CaCO2	Cytotoxicity assay	24 h	IC50 = 0.008 μM	18586491
HEPG2	Cytotoxicity assay	24 h	IC50 = 0.009 μM	18586491
MDA-MB-435	Antiproliferative activity assay	72 h	GI50 = 0.004 μM	18610995
HT29	Antiproliferative activity assay	48 h	GI50 = 0.015 μM	18617414
M21	Antiproliferative activity assay	48 h	GI50 = 0.037 μM	18617414
MCF7	Antiproliferative activity assay	48 h	GI50 = 0.054 μM	18617414
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.62 μM	18701301
PC3	Antiproliferative activity assay	48 h	IC50 = 2.73 μM	18701301
HCT116	Antiproliferative activity assay	48 h	IC50 = 6.18 μM	18701301
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	18752869
SKOV3	Anticancer assay	72 h	IC50 = 0.00134 μM	18762358
PANC1	Cytotoxicity assay	72 h	IC50 = 0.0099 μM	18951787
DLD1	Cytotoxicity assay	72 h	IC50 = 0.022 μM	18951787
AsPC1	Cytotoxicity assay	72 h	IC50 = 0.089 μM	18951787
NCI/ADR-RES	Cytotoxicity assay	72 h	IC50 = 1.3 μM	18951787
A431	Cytotoxicity assay	72 h	IC50 = 0.0251 μM	18990574
MCF7	Cytotoxicity assay	72 h	IC50 = 0.039 μM	18990574
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0471 μM	18990574
SKOV3	Cytotoxicity assay	72 h	IC50 = 0.0658 μM	18990574
PANC1	Growth inhibition assay	72 h	IC50 = 0.0099 μM	19022679
DLD1	Growth inhibition assay	72 h	IC50 = 0.022 μM	19022679
AsPC1	Growth inhibition assay	72 h	IC50 = 0.089 μM	19022679
NCI/ADR	Growth inhibition assay	72 h	IC50 = 1.3 μM	19022679
A2780	Antiproliferative activity assay	2 days	IC50 = 0.0234 μM	19028102
KB	Antiproliferative activity assay	3 days	IC50 = 0.0025 μM	19041247
COLO205	Antiproliferative activity assay	24 h	IC50 = 0.0033 μM	19041247
KB 8.5	Antiproliferative activity assay	3 days	IC50 = 0.026 μM	19041247
KBV1	Antiproliferative activity assay	3 days	IC50 = 2.013 μM	19041247
KB	Growth inhibition assay	72 h	IC50 = 0.0033 μM	19053773
KB-7D	Growth inhibition assay	72 h	IC50 = 0.0079 μM	19053773
Pgp170 overexpressing multidrug resistant-KB-TAX50	Growth inhibition assay	72 h	IC50 = 0.273 μM	19053773
NPC-TW01	Cytotoxicity assay	72 h	IC50 = 0.006 μM	19053781
MES-SA	Cytotoxicity assay	72 h	IC50 = 0.008 μM	19053781
NCI-H838	Cytotoxicity assay	72 h	IC50 = 0.026 μM	19053781
HCT116	Cytotoxicity assay	72 h	IC50 = 0.061 μM	19053781
Hep3B	Cytotoxicity assay	72 h	IC50 = 7.26 μM	19053781
A498	Cytotoxicity assay	72 h	IC50 = 8.81 μM	19053781
NB4	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19072209
A549	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19072209
MCF7	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19072209
SH-SY5Y	Cytotoxicity assay	48 h	IC50 = 0.2 μM	19072209
PC3	Cytotoxicity assay	48 h	IC50 = 0.2 μM	19072209
DLD1	Cytotoxicity assay	72 h	GI50 = 0.01 μM	19081249
B16	Cytotoxicity assay	72 h	GI50 = 0.01 μM	19081249
A172	Cytotoxicity assay	72 h	GI50 = 0.01 μM	19081249
HeLa	Cytotoxicity assay	72 h	GI50 = 0.02 μM	19081249
U87	Cytotoxicity assay	72 h	GI50 = 0.02 μM	19081249
SiHa	Cytotoxicity assay	72 h	GI50 = 0.03 μM	19081249
HeLa	Antiproliferative activity assay	96 h	IC50 = 0.001 μM	19091579
SKOV3	Antiproliferative activity assay	96 h	IC50 = 0.016 μM	19091579
BGC823	Antiproliferative activity assay	96 h	IC50 = 0.0189 μM	19091579
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	19124250
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.0031 μM	19124250
MX1	Cytotoxicity assay	72 h	IC50 = 0.046 μM	19124250
HCT116	Cytotoxicity assay	4 days	IC50 = 0.0011 μM	19128156
HT-29	Cytotoxicity assay	4 days	IC50 = 0.0036 μM	19128156
A2780	Cytotoxicity assay	48 h	IC50 = 0.0013 μM	19128972
P388	Antiproliferative activity assay	48 h	IC50 = 0.05 μM	19220018
cells ectopic expression of human	Antiproliferative activity assay	48 h	IC50 = 0.05 μM	19220018
L1210	Antiproliferative activity assay	48 h	IC50 = 0.06 μM	19220018
	Antiproliferative activity assay	48 h	IC50 = 0.3 μM	19220018
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0012 μM	19239240
A2780	Cytotoxicity assay	72 h	IC50 = 0.00138 μM	19239240
wild type A2780	Cytotoxicity assay	72 h	IC50 = 0.0017 μM	19239240
cisplatin-resistant A2780	Cytotoxicity assay	72 h	IC50 = 0.0022 μM	19239240
LCC-6	Cytotoxicity assay	72 h	IC50 = 0.00245 μM	19239240
HT-29	Cytotoxicity assay	72 h	IC50 = 0.0036 μM	19239240
H460	Cytotoxicity assay	72 h	IC50 = 0.0049 μM	19239240
topotecan-resistant A2780	Cytotoxicity assay	72 h	IC50 = 0.0072 μM	19239240
PANC1	Cytotoxicity assay	72 h	IC50 = 0.0257 μM	19239240
1A9PTX22	Cytotoxicity assay	72 h	IC50 = 0.1607 μM	19239240
NCI/ADR	Cytotoxicity assay	72 h	IC50 = 0.3 μM	19239240
1A9PTX10	Cytotoxicity assay	72 h	IC50 = 0.53295 μM	19239240
A2780/ADR	Cytotoxicity assay	72 h	IC50 = 1.239 μM	19239240
A549	Cytotoxicity assay	24 h	IC50 = 0.0052 μM	19245261
PC3M	Cytotoxicity assay	24 h	IC50 = 0.027 μM	19245261
HCT8	Cytotoxicity assay	24 h	IC50 = 0.037 μM	19245261
Bel7402	Cytotoxicity assay	24 h	IC50 = 0.095 μM	19245261
SNU398	Apoptosis assay	48 h	GI50 = 0.01 μM	19282188
HCT116	Apoptosis assay	48 h	EC50 = 0.023 μM	19282188
T47D	Apoptosis assay	48 h	EC50 = 0.035 μM	19282188
PC3	Cytotoxicity assay	4 days	IC50 = 0.0014 μM	19359169
A2780	Cytotoxicity assay	4 days	IC50 = 0.0149 μM	19359169
K562	Cytotoxicity assay	48 h	IC50 = 1.16 μM	19359185
MCF7	Cytotoxicity assay	48 h	IC50 = 2.11 μM	19359185
A549	Cytotoxicity assay	48 h	IC50 = 2.46 μM	19359185
SGC	Cytotoxicity assay	48 h	IC50 = 3.34 μM	19359185
HCT116	Cytotoxicity assay	48 h	IC50 = 4.37 μM	19359185
wild type A2780	Growth inhibition assay	72 h	IC50 = 0.0017 μM	19423340
cisplatin-resistant A2780	Growth inhibition assay	72 h	IC50 = 0.0022 μM	19423340
topotecan-resistant A2780	Growth inhibition assay	72 h	IC50 = 0.0072 μM	19423340
adriamycin and doxorubicin-resistant A2780	Growth inhibition assay	72 h	IC50 = 1.239 μM	19423340
NB4	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19425589
A549	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19425589
MCF7	Cytotoxicity assay	48 h	IC50 = 0.1 μM	19425589
SH-SY5Y	Cytotoxicity assay	48 h	IC50 = 0.2 μM	19425589
PC3	Cytotoxicity assay	48 h	IC50 = 0.2 μM	19425589
SNU398	Apoptosis assay	48 h	EC50 = 0.009 μM	19467598
HCT116	Apoptosis assay	48 h	EC50 = 0.018 μM	19467598
T47D	Growth inhibition assay	48 h	GI50 = 0.026 μM	19467598
MCF7	Cytotoxicity assay	48 h	IC50 = 0.08 μM	19467877
H1299	Growth inhibition assay	48 h	GI50 = 0.023 μM	19500976
T47D	Growth inhibition assay	48 h	GI50 = 0.026 μM	19500976
DLD1	Apoptosis assay	48 h	EC50 = 0.054 μM	19500976
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	19576785
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.0012 μM	19576785
MX1	Cytotoxicity assay	72 h	IC50 = 0.046 μM	19576785
vinblastine-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.4 μM	19576785
taxol-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 1.2 μM	19576785
MCF7	Growth inhibition assay	48 h	IC50 = 0.003 μM	19601594
HCT116	Antiproliferative activity assay	72 h	IC50 = 0.0008 μM	19665384
PC3	Antiproliferative activity assay	72 h	IC50 = 0.0008 μM	19665384
NCI/ADR	Antiproliferative activity assay	72 h	IC50 = 0.004 μM	19665384
HuH7	Antiproliferative activity assay	72 h	IC50 = 0.008 μM	19665384
Caco-2	Antiproliferative activity assay	72 h	IC50 = 0.02 μM	19665384
DG75	Antiproliferative activity assay	24 to 72 h	IC50 = 0.01 μM	19717215
MUTU-I	Antiproliferative activity assay	24 h	IC50 = 0.01 μM	19717215
HCT116	Antiproliferative activity assay	72 h	IC50 = 0.001 μM	19743863
SW48	Antiproliferative activity assay	72 h	IC50 = 0.001 μM	19743863
MES-SA	Antiproliferative activity assay	72 h	IC50 = 0.001 μM	19743863
CEM	Antiproliferative activity assay	72 h	IC50 = 0.002 μM	19743863
SW480	Antiproliferative activity assay	72 h	IC50 = 0.002 μM	19743863
MCF7	Cytotoxicity assay	72 h	IC50 = 0.003 μM	19743863
RL	Antiproliferative activity assay	72 h	IC50 = 0.003 μM	19743863
T47D	Antiproliferative activity assay	72 h	IC50 = 0.004 μM	19743863
UACC-812	Antiproliferative activity assay	72 h	IC50 = 0.7 μM	19743863
DU145	Cytotoxicity assay	72 h	IC50 = 4.84 μM	19754130
LNCAP	Cytotoxicity assay	72 h	IC50 = 6.32 μM	19754130
HT-29	Cytotoxicity assay	1 h	IC50 = 0.0034 μM	19778067
HCT116	Cytotoxicity assay	1 h	IC50 = 0.0035 μM	19778067
K562	Antiproliferative activity assay	48 h	IC50 = 1.16 μM	19815316
A549	Antiproliferative activity assay	48 h	IC50 = 2.28 μM	19815316
SGC7901	Antiproliferative activity assay	48 h	IC50 = 3.34 μM	19815316
HCT116	Antiproliferative activity assay	48 h	IC50 = 4.37 μM	19815316
IGROV1	Antiproliferative activity assay	72 h	IC50 = 0.06 μM	19833515
MCF7	Cytotoxicity assay	72 h	IC50 = 0.002 μM	19860383
KB	Cytotoxicity assay	48 h	IC50 = 0.02 μM	19879765
BT549	Cytotoxicity assay	48 h	IC50 = 0.02 μM	19879765
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.53 μM	19879765
african green monkey Vero	Toxicity assay	48 h	TC50 = 0.53 μM	19879765
SK-MEL	Cytotoxicity assay	48 h	IC50 = 4.1 μM	19879765
pig LLC-PK11	Toxicity assay	48 h	TC50 = 4.39 μM	19879765
OVCAR-3	Growth inhibition assay	48 h	IC50 = 2.7 μM	19939522
A549	Growth inhibition assay	48 h	IC50 = 2.7 μM	19939522
SNU398	Apoptosis assay	48 h	EC50 = 0.009 μM	20034792
HCT116	Apoptosis assay	48 h	EC50 = 0.018 μM	20034792
T47D	Growth inhibition assay	48 h	GI50 = 0.026 μM	20034792
HCT116	Cytotoxicity assay	72 h	IC50 = 0.002399 μM	20116905
MCF7	Antiproliferative activity assay	20 h	IC50 = 0.021 μM	20149494
HeLa	Cytotoxicity assay	48 h	IC50 = 0.03 μM	20180542
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0013 μM	20181487
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.0031 μM	20181487
MX1	Cytotoxicity assay	72 h	IC50 = 0.035 μM	20181487
KB3-1	Cytotoxicity assay	72 h	IC50 = 0.0012 μM	20302303
HT-29	Cytotoxicity assay	3 days	ED50 = 0.0001 μM	20384315
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	20521771
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	20521771
PANC1	Growth inhibition assay	48 h	IC50 = 0.008 μM	20521771
SK-BR-3	Cytotoxicity assay	48 h	IC50 = 0.11 μM	20521771
A549	Cytotoxicity assay	48 h	IC50 = 1.4 μM	20521771
LT12	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	20537765
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	20537765
SF268	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	20537765
NCI-H460	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	20537765
RKO	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	20537765
KB/HeLa	Antiproliferative activity assay	48 h	IC50 = 0.01 μM	20537765
P388	Antiproliferative activity assay	48 h	IC50 = 0.04 μM	20537765
L1210	Antiproliferative activity assay	48 h	IC50 = 0.06 μM	20537765
DLD1	Cytotoxicity assay	72 h	GI50 = 0.01 μM	20538462
B16	Cytotoxicity assay	72 h	GI50 = 0.01 μM	20538462
A172	Cytotoxicity assay	72 h	GI50 = 0.01 μM	20538462
HeLa	Cytotoxicity assay	72 h	GI50 = 0.02 μM	20538462
U87	Cytotoxicity assay	72 h	GI50 = 0.02 μM	20538462
SiHa	Cytotoxicity assay	72 h	GI50 = 0.03 μM	20538462
A549	Cytotoxicity assay	96 h	IC50 = 0.001 μM	20560647
BGC823	Cytotoxicity assay	96 h	IC50 = 0.04 μM	20560647
A2780	Cytotoxicity assay	96 h	IC50 = 0.9 μM	20560647
HCT8	Cytotoxicity assay	96 h	IC50 = 3.6 μM	20560647
Bel7402	Cytotoxicity assay	96 h	IC50 = 6.3 μM	20560647
A2780	Cytotoxicity assay	3 days	IC50 = 0.65 μM	20593839
HCT8	Cytotoxicity assay	3 days	IC50 = 0.67 μM	20593839
Bel7402	Cytotoxicity assay	3 days	IC50 = 1.8 μM	20593839
BGC823	Cytotoxicity assay	72 h	IC50 = 0.001 μM	20719510
A2780	Cytotoxicity assay	72 h	IC50 = 0.001 μM	20719510
A549	Cytotoxicity assay	72 h	IC50 = 0.016 μM	20719510
HCT8	Cytotoxicity assay	72 h	IC50 = 0.051 μM	20719510
Bel7402	Cytotoxicity assay	72 h	IC50 = 0.06 μM	20719510
A549	Cytotoxicity assay	72 h	IC50 = 0.0038 μM	20732809
HEK	Cytotoxicity assay	72 h	IC50 = 0.0039 μM	20732809
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0044 μM	20732809
HeLa	Cytotoxicity assay	72 h	IC50 = 0.0089 μM	20732809
Hep3B	Anticancer assay	3 days	GI50 = 0.0004 μM	20735140
MCF7	Cytotoxicity assay	72 h	IC50 = 0.002 μM	20800500
wild type LCC-6	Cytotoxicity assay	72 h	IC50 = 0.003 μM	20800500
A2780	Cytotoxicity assay	72 h	IC50 = 0.02 μM	20800500
CFPAC-1	Cytotoxicity assay	72 h	IC50 = 0.047 μM	20800500
multidrug-resistant LCC-6	Cytotoxicity assay	72 h	IC50 = 0.379 μM	20800500
NCI/ADR	Cytotoxicity assay	72 h	IC50 = 0.41 μM	20800500
multidrug-resistant MDA-MB-435/LCCMDR1	Cytotoxicity assay	48 h	IC50 = 0.004 μM	20919720
MDA-MB-435	Cytotoxicity assay	48 h	IC50 = 0.277 μM	20919720
HT-29	Cytotoxicity assay	3 days	ED50 = 0.0006 μM	20939540
HCT116	Growth inhibition assay	96 h	IC50 = 0.002 μM	20943401
HCT15	Growth inhibition assay	96 h	IC50 = 0.14 μM	20943401
A549	Antiproliferative activity assay	96 h	IC50 = 0.0049 μM	20974505
MCF7	Antiproliferative activity assay	96 h	IC50 = 0.021 μM	20974505
K562	Cytotoxicity assay	48 h	IC50 = 1.16 μM	21067933
MCF7	Cytotoxicity assay	48 h	IC50 = 2.11 μM	21067933
A549	Cytotoxicity assay	48 h	IC50 = 2.46 μM	21067933
SGC	Cytotoxicity assay	48 h	IC50 = 3.34 μM	21067933
HCT116	Cytotoxicity assay	48 h	IC50 = 4.37 μM	21067933
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.003 μM	21106377
MCF7	Cytotoxicity assay	72 h	GI50 = 0.003 μM	21115210
HT-29	Cytotoxicity assay	72 h	GI50 = 0.003 μM	21115210
K562	Cytotoxicity assay	72 h	GI50 = 0.004 μM	21115210
PC3	Cytotoxicity assay	72 h	GI50 = 0.004 μM	21115210
MCF7	Cytotoxicity assay	24 h	IC50 = 0.63 μM	21115212
SMMC7721	Cytotoxicity assay	24 h	IC50 = 1.42 μM	21115212
A2780	Cytotoxicity assay	48 to 72 h	IC50 = 0.01 μM	21126027
Jurkat	Cell cycle arrest assay	24 h	IC50 = 0.01 μM	21126027
HeLa	Cytotoxicity assay	48 to 72 h	IC50 = 0.02 μM	21126027
SW620	Cytotoxicity assay	48 to 72 h	IC50 = 0.03 μM	21126027
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0013 μM	21144756
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.003 μM	21144756
MX1	Cytotoxicity assay	72 h	IC50 = 0.035 μM	21144756
chemoresistant DG75	Cytotoxicity assay	72 h	IC50 = 0.01 μM	21227702
chemosensitive MUTU-I	Cytotoxicity assay	24 h	IC50 = 0.01 μM	21227702
HT1080	Antiproliferative activity assay	96 h	IC50 = 0.0012 μM	21296467
A549	Antiproliferative activity assay	96 h	IC50 = 0.0044 μM	21296467
A375	Antiproliferative activity assay	96 h	IC50 = 0.0046 μM	21296467
NCI-N87	Antiproliferative activity assay	96 h	IC50 = 0.0059 μM	21296467
MCF7	Antiproliferative activity assay	96 h	IC50 = 0.0205 μM	21296467
HeLa	Antiproliferative activity assay	96 h	IC50 = 0.1 μM	21296467
PANC1	Antiproliferative activity assay	96 h	IC50 = 0.3841 μM	21296467
Bel7402	Antiproliferative activity assay	96 h	IC50 = 0.5782 μM	21296467
1A9	Antiproliferative activity assay	3 days	ED50 = 0.00209 μM	21296579
A549	Antiproliferative activity assay	3 days	ED50 = 0.00256 μM	21296579
KB	Antiproliferative activity assay	3 days	ED50 = 0.00287 μM	21296579
PC3	Antiproliferative activity assay	3 days	ED50 = 0.00887 μM	21296579
KB	Cytotoxicity assay	72 h	GI50 = 0.00487 μM	21316977
DU145	Cytotoxicity assay	72 h	GI50 = 0.00555 μM	21316977
A549	Cytotoxicity assay	72 h	GI50 = 0.00558 μM	21316977
MCF7	Cytotoxicity assay	48 h	IC50 = 0.006 μM	21341718
HT-29	Cytotoxicity assay	48 h	IC50 = 0.007 μM	21341718
K562	Cytotoxicity assay	48 h	IC50 = 1.16 μM	21342735
MCF7	Cytotoxicity assay	48 h	IC50 = 2.11 μM	21342735
A549	Cytotoxicity assay	48 h	IC50 = 2.46 μM	21342735
SGC	Cytotoxicity assay	48 h	IC50 = 3.34 μM	21342735
HCT116	Cytotoxicity assay	48 h	IC50 = 4.37 μM	21342735
multidrug-resistant K562	Cytotoxicity assay	48 h	IC50 = 5.63 μM	21342735
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.003 μM	21356592
taxol-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.43 μM	21356592
vinblastine-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 1.27 μM	21356592
KB	Cytotoxicity assay	3 days	GI50 = 0.00516 μM	21377368
DU145	Cytotoxicity assay	3 days	GI50 = 0.00523 μM	21377368
A549	Cytotoxicity assay	3 days	GI50 = 0.0076 μM	21377368
A2780	Cytotoxicity assay	24 h	IC50 = 0.00082 μM	21396747
A2780AD	Cytotoxicity assay	24 h	IC50 = 0.949 μM	21396747
HT-29	Cytotoxicity assay	3 days	ED50 = 0.0001 μM	21428375
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.002 μM	21440449
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0026 μM	21446699
HT-29	Cytotoxicity assay	48 h	IC50 = 0.003 μM	21446699
A549	Antiproliferative activity assay	72 h	IC50 = 0.0023 μM	21480626
HT-29	Antiproliferative activity assay	72 h	IC50 = 0.0061 μM	21480626
A431	Antiproliferative activity assay	72 h	IC50 = 0.0092 μM	21480626
SKOV3	Antiproliferative activity assay	72 h	IC50 = 0.0145 μM	21480626
NCI-H460	Antiproliferative activity assay	72 h	IC50 = 0.0146 μM	21480626
MCF7	Cytotoxicity assay	48 h	GI50 = 0.012 μM	21513294
HT-29	Cytotoxicity assay	48 h	GI50 = 0.012 μM	21513294
SF268	Cytotoxicity assay	48 h	GI50 = 0.012 μM	21513294
H460	Cytotoxicity assay	48 h	GI50 = 0.024 μM	21513294
CHOK1	Cytotoxicity assay	48 h	GI50 = 5.9 μM	21513294
HeLa	Cytotoxicity assay	24 h	IC50 = 6.62 μM	21514015
HELF	Cytotoxicity assay	24 h	IC50 = 7.17 μM	21514015
SH-SY5Y	Cytotoxicity assay	24 h	IC50 = 8.56 μM	21514015
BGC823	Cytotoxicity assay	24 h	IC50 = 9.24 μM	21514015
A2780	Cytotoxicity assay	72 h	IC50 = 0.001 μM	21530251
BGC823	Cytotoxicity assay	72 h	IC50 = 0.001 μM	21530251
Bel7402	Cytotoxicity assay	72 h	IC50 = 0.006 μM	21530251
A549	Cytotoxicity assay	72 h	IC50 = 0.016 μM	21530251
HCT8	Cytotoxicity assay	72 h	IC50 = 0.051 μM	21530251
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	21534539
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	21534539
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	21534539
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	21534539
HL60	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21534539
OVCAR8	Anticancer assay	96 h	IC50 = 0.0047 μM	21557538
NCI/ADR-RES	Anticancer assay	96 h	IC50 = 6.263 μM	21557538
NCI-H460	Antiproliferative activity assay	48 h	IC50 = 0.004 μM	21563750
COLO205	Antiproliferative activity assay	48 h	IC50 = 0.005 μM	21563750
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	21563750
BT549	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	21563750
451LU	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	21563750
SW480	Antiproliferative activity assay	48 h	IC50 = 0.011 μM	21563750
DLD1	Antiproliferative activity assay	48 h	IC50 = 0.05 μM	21563750
HT1080	Antiproliferative activity assay	48 h	IC50 = 0.00015 μM	21604746
CEM	Antiproliferative activity assay	48 h	IC50 = 0.00027 μM	21604746
L1210	Antiproliferative activity assay	48 h	IC50 = 0.0004 μM	21604746
K562	Antiproliferative activity assay	48 h	IC50 = 0.00071 μM	21604746
DU145	Antiproliferative activity assay	48 h	IC50 = 0.0013 μM	21604746
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.0026 μM	21604746
MDA-MB-231	Antiproliferative activity assay	48 h	IC50 = 0.0091 μM	21604746
B16F0	Antiproliferative activity assay	48 h	IC50 = 0.028 μM	21604746
P388D1	Antiproliferative activity assay	48 h	IC50 = 0.035 μM	21604746
CHO-VV 3-2	Antiproliferative activity assay	48 h	IC50 = 0.14 μM	21604746
CHO	Antiproliferative activity assay	48 h	IC50 = 0.17 μM	21604746
CHO-TAX 5-6	Antiproliferative activity assay	48 h	IC50 = 0.52 μM	21604746
CEM/VLB	Antiproliferative activity assay	48 h	IC50 = 3.34 μM	21604746
A549	Antiproliferative activity assay	72 h	IC50 = 0.0072 μM	21663319
taxol-resistant A549-T12	Antiproliferative activity assay	72 h	IC50 = 0.0752 μM	21663319
MCF7	Cytotoxicity assay	48 h	IC50 = 0.0025 μM	21680190
MCF7/VP	Cytotoxicity assay	48 h	IC50 = 0.0028 μM	21680190
NCI/ADR	Cytotoxicity assay	48 h	IC50 = 2.7 μM	21680190
LT12	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	21705223
NCI-H460	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21705223
SF268	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21705223
KB/HeLa	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21705223
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21705223
RKOp27	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21705223
P388	Antiproliferative activity assay	48 h	IC50 = 0.04 μM	21705223
L1210	Antiproliferative activity assay	48 h	IC50 = 0.06 μM	21705223
NCI-H460	Anticancer assay	72 h	IC30 = 3.6 μM	21707046
A2780	Cytotoxicity assay	48 h	IC50 = 0.00062 μM	21764308
A2780AD	Cytotoxicity assay	48 h	IC50 = 1.9 μM	21764308
MCF7	Cytotoxicity assay	48 h	IC50 = 0.00162 μM	21779519
COLO205	Cytotoxicity assay	48 h	IC50 = 0.00331 μM	21779519
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0012 μM	21800839
A2780	Cytotoxicity assay	2 days	IC50 = 0.014 μM	21802957
Hep3B2	Cytotoxicity assay	72 h	IC50 = 0.000016 μM	21812410
PANC1	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	21812410
CNE1-LMP1	Cytotoxicity assay	72 h	IC50 = 0.0042 μM	21812410
MGC	Cytotoxicity assay	72 h	IC50 = 0.0064 μM	21812410
A375	Cytotoxicity assay	72 h	IC50 = 0.0089 μM	21812410
MCF7	Cytotoxicity assay	72 h	IC50 = 0.014 μM	21812410
HaCaT	Cytotoxicity assay	72 h	IC50 = 0.024 μM	21812410
A549	Cytotoxicity assay	72 h	IC50 = 0.03 μM	21812410
EC109	Cytotoxicity assay	72 h	IC50 = 0.14 μM	21812410
MES-SA	Cytotoxicity assay	96 h	IC50 = 0.004 μM	21812421
MES-SA/Dx5	Cytotoxicity assay	96 h	IC50 = 0.75 μM	21812421
HL60	Cytotoxicity assay	72 h	IC50 = 0.0034 μM	21848268
MCF7	Antiproliferative activity assay	96 h	IC50 = 0.00091 μM	21870795
A549	Antiproliferative activity assay	72 h	IC50 = 0.00314 μM	21870795
A549	Cytotoxicity assay	24 h	EC50 = 0.0046 μM	21873068
MCF7	Cytotoxicity assay	3 days	GI50 = 1.07 μM	21889341
PC3	Cytotoxicity assay	3 days	GI50 = 1.46 μM	21889341
SK-N-SH	Cytotoxicity assay	3 days	GI50 = 2.19 μM	21889341
HeLa	Cytotoxicity assay	3 days	GI50 = 2.82 μM	21889341
CHO-VV 3-2	Antiproliferative activity assay	48 h	IC50 = 0.14 μM	21920638
CHO-TAX 5-6	Antiproliferative activity assay	48 h	IC50 = 0.52 μM	21920638
multidrug-resistant CEM/VLB	Antiproliferative activity assay	48 h	IC50 = 3.34 μM	21920638
A549	Cytotoxicity assay	48 h	IC50 = 0.01 μM	21973054
HeLa	Cytotoxicity assay	48 h	IC50 = 0.6 μM	21973054
HT-29	Cytotoxicity assay	3 days	ED50 = 0.006 μM	21973101
A549	Antiproliferative activity assay	72 h	IC50 = 0.0072 μM	22027100
taxol-resistant A549-T12	Antiproliferative activity assay	72 h	IC50 = 0.075 μM	22027100
OVCAR8	Growth inhibition assay	96 h	IC50 = 0.002 μM	22044164
NCI-ADR-RES	Growth inhibition assay	96 h	IC50 = 1.5 μM	22044164
KB	Growth inhibition assay	72 h	IC50 = 0.0033 μM	22060033
KB-7d	Growth inhibition assay	72 h	IC50 = 0.0079 μM	22060033
KB-S15	Growth inhibition assay	72 h	IC50 = 0.273 μM	22060033
A2780	Antiproliferative activity assay	2 days	IC50 = 0.015 μM	22071526
KB	Cytotoxicity assay	48 h	IC50 = 0.0045 μM	22074257
L1210	Cytotoxicity assay	48 h	IC50 = 0.12 μM	22074257
A2780	Antiproliferative activity assay	2 days	IC50 = 0.02 μM	22136523
QGY7701	Cytotoxicity assay	72 h	IC50 = 0.04 μM	22153338
HepG2	Cytotoxicity assay	72 h	IC50 = 0.05 μM	22153338
Bel7404	Cytotoxicity assay	72 h	IC50 = 0.82 μM	22153338
SMMC7721	Cytotoxicity assay	72 h	IC50 = 0.88 μM	22153338
Bel7402	Cytotoxicity assay	72 h	IC50 = 1.25 μM	22153338
MCF7	Cytotoxicity assay	24 to 48 h	IC50 = 0.003 μM	22222040
SH-SY5Y	Cytotoxicity assay	24 to 48 h	IC50 = 0.004 μM	22222040
HepG2	Cytotoxicity assay	24 to 48 h	IC50 = 0.007 μM	22222040
H460	Cytotoxicity assay	24 to 48 h	IC50 = 0.008 μM	22222040
HT-29	Cytotoxicity assay	3 days	IC50 = 0.006 μM	22239601
DU145	Antiproliferative activity assay	72 h	GI50 = 0.00386 μM	22265685
KB	Antiproliferative activity assay	72 h	GI50 = 0.00412 μM	22265685
A549	Antiproliferative activity assay	72 h	GI50 = 0.00546 μM	22265685
MCF7	Cytotoxicity assay	96 h	IC50 = 0.1 μM	22360613
A549	Cytotoxicity assay	72 h	IC50 = 0.19 μM	22472043
MCF7	Cytotoxicity assay	48 h	IC50 = 0.006 μM	22472045
K562	Cytotoxicity assay	72 h	IC50 = 0.41 μM	22483090
CaEs17	Cytotoxicity assay	72 h	IC50 = 0.43 μM	22483090
MGC803	Cytotoxicity assay	72 h	IC50 = 0.85 μM	22483090
HeLa	Cytotoxicity assay	72 h	IC50 = 0.89 μM	22483090
Bel7402	Cytotoxicity assay	72 h	IC50 = 1.89 μM	22483090
A549	Cytotoxicity assay	72 h	IC50 = 3.46 μM	22483090
MCF7	Cytotoxicity assay	72 h	IC50 = 4.77 μM	22483090
CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.0012 μM	22507893
taxol-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 0.43 μM	22507893
vinblastine-resistant CCRF-CEM	Cytotoxicity assay	72 h	IC50 = 1.27 μM	22507893
BGC823	Cytotoxicity assay	72 h	IC50 = 0.001 μM	22583079
A2780	Cytotoxicity assay	72 h	IC50 = 0.001 μM	22583079
Bel7402	Cytotoxicity assay	72 h	IC50 = 0.006 μM	22583079
A549	Cytotoxicity assay	72 h	IC50 = 0.016 μM	22583079
HCT8	Cytotoxicity assay	72 h	IC50 = 0.051 μM	22583079
MES-SA	Cytotoxicity assay	96 h	IC50 = 0.004 μM	22587519
MESSA/DX5	Cytotoxicity assay	96 h	IC50 = 0.75 μM	22587519
PC3	Antiproliferative activity assay	48 h	IC50 = 0.0004 μM	22783954
paclitaxel-resistant PC3-TxR	Antiproliferative activity assay	48 h	IC50 = 0.188 μM	22783954
MCF7	Cytotoxicity assay	24 h	IC50 = 0.015 μM	22818081
SKBR3	Growth inhibition assay	48 h	IC50 = 0.0019 μM	22850214
HepG2	Cytotoxicity assay	72 h	IC50 = 0.00044 μM	22871217
MCF7	Cytotoxicity assay	72 h	IC50 = 0.003 μM	22871217
A375	Cytotoxicity assay	72 h	IC50 = 0.0092 μM	22871217
BxPC3	Cytotoxicity assay	72 h	IC50 = 0.09 μM	22871217
SMMC7721	Cytotoxicity assay	72 h	IC50 = 0.15 μM	22871217
PANC1	Cytotoxicity assay	72 h	IC50 = 0.26 μM	22871217
A549	Cytotoxicity assay	72 h	IC50 = 0.72 μM	22871217
AGS	Cytotoxicity assay	72 h	IC50 = 1.6 μM	22871217
NCI-H2126	Cytotoxicity assay	72 h	IC50 = 2.5 μM	22871217
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 5 μM	22871217
U87	Cytotoxicity assay	72 h	IC50 = 8.1 μM	22871217
HELF	Cytotoxicity assay	24 h	IC50 = 7.14 μM	22901410
BGC	Cytotoxicity assay	24 h	IC50 = 9.26 μM	22901410
HELF	Cytotoxicity assay	24 h	IC50 = 7.14 μM	22921966
BGC	Cytotoxicity assay	24 h	IC50 = 9.26 μM	22921966
DU145	Cytotoxicity assay	72 h	GI50 = 0.00255 μM	22932313
KB	Cytotoxicity assay	72 h	GI50 = 0.00265 μM	22932313
A549	Cytotoxicity assay	72 h	GI50 = 0.00489 μM	22932313
KBVIN	Cytotoxicity assay	72 h	GI50 = 0.948 μM	22932313
HL60	Cytotoxicity assay	72 h	IC50 = 0.00282 μM	22959518
HeLa	Cytotoxicity assay	72 h	IC50 = 0.00293 μM	22959518
U937	Cytotoxicity assay	72 h	IC50 = 0.00337 μM	22959518
A549	Antiproliferative activity assay	72 h	IC50 = 0.0072 μM	23117171
taxol-resistant A549-T12	Antiproliferative activity assay	72 h	IC50 = 0.0752 μM	23117171
IGROV1/Pt1	Cytotoxicity assay	72 h	IC50 = 0.0022 μM	23140358
SKOV3	Cytotoxicity assay	72 h	IC50 = 0.0027 μM	23140358
U2OS	Cytotoxicity assay	72 h	IC50 = 0.0034 μM	23140358
PANC1	Cytotoxicity assay	72 h	IC50 = 0.0052 μM	23140358
MIAPaCa2	Cytotoxicity assay	72 h	IC50 = 0.0072 μM	23140358
IGROV1	Cytotoxicity assay	72 h	IC50 = 0.023 μM	23140358
A2780	Antiproliferative activity assay	2 days	IC50 = 0.028 μM	23149304
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.052 μM	23153397
HepG2	Cytotoxicity assay	72 h	IC50 = 0.054 μM	23153397
A549	Cytotoxicity assay	72 h	IC50 = 0.056 μM	23153397
HeLa	Cytotoxicity assay	96 h	IC50 = 0.001 μM	23176628
SW780	Cytotoxicity assay	96 h	IC50 = 0.0011 μM	23176628
MESSA	Cytotoxicity assay	72 h	IC50 = 0.004 μM	23214452
HeLa	Cytotoxicity assay	48 h	IC50 = 0.005 μM	23214452
A549	Cytotoxicity assay	48 h	IC50 = 0.007 μM	23214452
HT-29	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23214452
HCT15	Cytotoxicity assay	72 h	IC50 = 0.09 μM	23214452
MESSA/DX5	Cytotoxicity assay	72 h	IC50 = 1.764 μM	23214452
U937	Cytotoxicity assay	72 h	IC50 = 0.0023 μM	23301703
MOLT4	Cytotoxicity assay	72 h	IC50 = 0.0027 μM	23301703
K562	Cytotoxicity assay	72 h	IC50 = 0.0051 μM	23301703
KU812	Cytotoxicity assay	72 h	IC50 = 0.0053 μM	23301703
HL60	Cytotoxicity assay	72 h	IC50 = 0.0058 μM	23301703
SUP-B15	Cytotoxicity assay	72 h	IC50 = 0.008 μM	23301703
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23327668
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23327668
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23327668
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23327668
SW480	Cytotoxicity assay	48 h	IC50 = 0.15 μM	23327668
HT-29	Cytotoxicity assay	3 days	IC50 = 0.001 μM	23327794
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0016 μM	23332369
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.0044 μM	23332369
JC	Cytotoxicity assay	48 h	IC50 = 0.15 μM	23352482
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0063 μM	23356786
A549	Cytotoxicity assay	48 h	IC50 = 0.0082 μM	23356786
QGY	Cytotoxicity assay	48 h	IC50 = 0.0113 μM	23356786
SW480	Cytotoxicity assay	48 h	IC50 = 0.0121 μM	23356786
K562	Cytotoxicity assay	48 h	IC50 = 0.0157 μM	23356786
A549	Cytotoxicity assay	72 h	IC50 = 0.0035 μM	23445496
A549-T12	Cytotoxicity assay	72 h	IC50 = 0.0923 μM	23445496
MDA-MB-435	Cytotoxicity assay	48 h	IC50 = 0.004 μM	23547728
MDA-MB-435/LCC6MDR1	Cytotoxicity assay	48 h	IC50 = 0.277 μM	23547728
KB403	Cytotoxicity assay	6 h	IC50 = 0.001 μM	23584542
WRL68	Cytotoxicity assay	6 h	IC50 = 0.004 μM	23584542
MCF7	Cytotoxicity assay	6 h	IC50 = 0.005 μM	23584542
Caco2	Cytotoxicity assay	6 h	IC50 = 0.008 μM	23584542
PA1	Cytotoxicity assay	6 h	IC50 = 0.008 μM	23584542
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23586920
A2058	Cytotoxicity assay	96 h	IC50 = 0.0047 μM	23623678
H522-T1	Cytotoxicity assay	96 h	IC50 = 0.0081 μM	23623678
A2780	Cytotoxicity assay	2 days	IC50 = 0.012 μM	23623678
K562	Cytotoxicity assay	72 h	IC50 = 0.41 μM	23644204
CaEs17	Cytotoxicity assay	72 h	IC50 = 0.43 μM	23644204
MGC803	Cytotoxicity assay	72 h	IC50 = 0.85 μM	23644204
Bel7402	Cytotoxicity assay	72 h	IC50 = 1.89 μM	23644204
HT1080	Cytotoxicity assay	24 h	IC50 = 6 μM	23647462
SNU387	Cytotoxicity assay	48 h	IC50 = 0.27 μM	23701597
HepG2	Cytotoxicity assay	72 h	IC50 = 0.006 μM	23708235
SKOV3	Cytotoxicity assay	72 h	IC50 = 0.012 μM	23708235
A549	Cytotoxicity assay	3 days	IC50 = 0.02 μM	23738539
NB4	Cytotoxicity assay	3 days	IC50 = 0.03 μM	23738539
MCF7	Cytotoxicity assay	3 days	IC50 = 0.1 μM	23738539
PC3	Cytotoxicity assay	3 days	IC50 = 0.2 μM	23738539
SH-SY5Y	Cytotoxicity assay	3 days	IC50 = 0.2 μM	23738539
HT-29	Cytotoxicity assay	96 h	IC50 = 0.00198 μM	23746477
HCT116	Cytotoxicity assay	96 h	IC50 = 0.00613 μM	23746477
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23819871
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23819871
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	23819871
SW480	Cytotoxicity assay	48 h	IC50 = 0.04 μM	23819871
A549	Cytotoxicity assay	48 h	IC50 = 1.4 μM	23819871
MCF7	Cytotoxicity assay	72 h	GI50 = 0.003 μM	23831811
HT-29	Cytotoxicity assay	72 h	GI50 = 0.003 μM	23831811
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 1 μM	23848163
PANC1	Cytotoxicity assay	72 h	IC50 = 1 μM	23848163
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0017 μM	23855338
rat lymphatic endothelial	Antiproliferative activity assay	48 h	IC50 = 0.018 μM	23855338
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0012 μM	23855953
A549	Cytotoxicity assay	72 h	IC50 = 0.014 μM	23886686
HT-29	Cytotoxicity assay	72 h	IC50 = 0.0006 μM	23895019
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0016 μM	23895532
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	23895532
SKOV3/M6-6 isogenic	Function assay	48 h	IC50 = 2.6 μM	23895532
MES-SA	Growth inhibition assay	48 h	GI50 = 0.007 μM	23927793
MES-SA/Dx5	Growth inhibition assay	48 h	GI50 = 9.8 μM	23927793
HL60	Antimicrobial assay	48 h	IC50 = 0.008 μM	23957453
SMMC7721	Antimicrobial assay	48 h	IC50 = 0.008 μM	23957453
MCF7	Antimicrobial assay	48 h	IC50 = 0.008 μM	23957453
SW480	Antimicrobial assay	48 h	IC50 = 0.04 μM	23957453
A549	Antimicrobial assay	48 h	IC50 = 0.1 μM	23957453
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.003 μM	24012378
PC3	Cytotoxicity assay	72 h	IC50 = 0.02 μM	24033131
DU145	Cytotoxicity assay	72 h	IC50 = 0.04 μM	24033131
WI38	Cytotoxicity assay	72 h	IC50 = 0.05 μM	24033131
MCF7	Cytotoxicity assay	48 h	IC50 = 0.5 μM	24056146
PC3	Cytotoxicity assay	48 h	IC50 = 1.5 μM	24056146
A549	Cytotoxicity assay	72 h	IC50 = 0.02 μM	24063567
NB4	Cytotoxicity assay	72 h	IC50 = 0.03 μM	24063567
MCF7	Cytotoxicity assay	72 h	IC50 = 0.1 μM	24063567
SH-SY5Y	Cytotoxicity assay	72 h	IC50 = 0.2 μM	24063567
PC3	Cytotoxicity assay	72 h	IC50 = 0.2 μM	24063567
A549	Cytotoxicity assay	48 h	IC50 = 0.02 μM	24063582
NB4	Cytotoxicity assay	48 h	IC50 = 0.03 μM	24063582
MCF7	Cytotoxicity assay	48 h	IC50 = 0.1 μM	24063582
PC3	Cytotoxicity assay	48 h	IC50 = 0.2 μM	24063582
SH-SY5Y	Cytotoxicity assay	48 h	IC50 = 0.2 μM	24063582
HeLa	Cytotoxicity assay	72 h	IC50 = 0.0014 μM	24087857
SKOV3	Cytotoxicity assay	72 h	IC50 = 0.003 μM	24087857
KB	Cytotoxicity assay	72 h	IC50 = 0.0041 μM	24106982
KB-7d	Cytotoxicity assay	72 h	IC50 = 0.0079 μM	24106982
KB-S15	Cytotoxicity assay	72 h	IC50 = 0.273 μM	24106982
A549	Antiproliferative activity assay	96 h	IC50 = 0.0044 μM	24211639
MCF7	Antiproliferative activity assay	96 h	IC50 = 0.0205 μM	24211639
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24219809
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24219809
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24219809
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24219809
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24219809
A2780	Antiproliferative activity assay	2 days	IC50 = 0.024 μM	24239390
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24256484
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24256484
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24256484
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24256484
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24256484
BEAS2B	Cytotoxicity assay	48 h	IC50 = 0.58 μM	24256484
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.035 μM	24269481
A549	Cytotoxicity assay	48 h	IC50 = 0.93 μM	24269481
MCF7	Cytotoxicity assay	72 h	IC50 = 0.00705 μM	24332858
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24417634
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24417634
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24417634
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24417634
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24417634
Bel7402	Cytotoxicity assay	96 h	IC50 = 0.011 μM	24467317
HCT8	Cytotoxicity assay	96 h	IC50 = 0.02 μM	24467317
BGC823	Cytotoxicity assay	96 h	IC50 = 0.026 μM	24467317
A549	Cytotoxicity assay	96 h	IC50 = 0.032 μM	24467317
A2780	Cytotoxicity assay	96 h	IC50 = 0.59 μM	24467317
ViBo	Antiproliferative activity assay	24 h	IC50 = 1.6 μM	24487193
CaSki	Antiproliferative activity assay	24 h	IC50 = 2.9 μM	24487193
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0056 μM	24564494
KB	Cytotoxicity assay	72 h	IC50 = 0.0051 μM	24657567
KB-7d	Cytotoxicity assay	72 h	IC50 = 0.0084 μM	24657567
KB-S15	Cytotoxicity assay	72 h	IC50 = 0.135 μM	24657567
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24697496
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24697496
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24697496
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24697496
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	24697496
HT-29	Growth inhibition assay	48 h	GI50 = 0.001 μM	24727464
U251	Growth inhibition assay	48 h	GI50 = 0.003 μM	24727464
MCF7	Growth inhibition assay	48 h	GI50 = 0.005 μM	24727464
UACC62	Growth inhibition assay	48 h	GI50 = 0.01 μM	24727464
786-0	Growth inhibition assay	48 h	GI50 = 0.02 μM	24727464
African green monkey Vero	Growth inhibition assay	48 h	GI50 = 0.03 μM	24727464
NCI-ADR-RES	Growth inhibition assay	48 h	GI50 = 0.04 μM	24727464
NCI-H460	Growth inhibition assay	48 h	GI50 = 0.1 μM	24727464
PC3	Growth inhibition assay	48 h	GI50 = 0.1 μM	24727464
K562	Growth inhibition assay	48 h	GI50 = 0.1 μM	24727464
OVCAR3	Growth inhibition assay	48 h	GI50 = 0.2 μM	24727464
HepG2	Cytotoxicity assay	3 days	IC50 = 0.00019 μM	24745968
KB	Cytotoxicity assay	3 days	IC50 = 0.0039 μM	24745968
NALM6	Antiproliferative activity assay	48 to 72 h	IC50 = 0.0041 μM	24852281
Jurkat	Antiproliferative activity assay	48 to 72 h	IC50 = 0.0045 μM	24852281
K562	Antiproliferative activity assay	48 to 72 h	IC50 = 0.0055 μM	24852281
PC3	Cytotoxicity assay	96 h	IC50 = 0.0025 μM	24900437
HeLa	Growth inhibition assay	96 h	IC50 = 0.0053 μM	24900865
OVCAR8	Growth inhibition assay	96 h	IC50 = 0.01 μM	24900865
NCI/ADR-RES	Growth inhibition assay	96 h	IC50 = 5 μM	24900865
MCF7	Cytotoxicity assay	72 h	IC50 = 0.045 μM	24929344
HCT116	Cytotoxicity assay	72 h	IC50 = 0.069 μM	24929344
HepG2	Cytotoxicity assay	72 h	IC50 = 0.084 μM	24929344
HeLa	Cytotoxicity assay	72 h	IC50 = 0.096 μM	24929344
U251	Cytotoxicity assay	72 h	IC50 = 0.128 μM	24929344
HT-29	Antiproliferative activity assay	24 and 72 h	IC50 = 0.29 μM	24941130
HeLa	Antiproliferative activity assay	24 and 72 h	IC50 = 0.29 μM	24941130
Caco2	Antiproliferative activity assay	24 and 72 h	IC50 = 0.31 μM	24941130
HL60	Antiproliferative activity assay	24 and 72 h	IC50 = 0.32 μM	24941130
MCF7	Antiproliferative activity assay	24 and 72 h	IC50 = 0.33 μM	24941130
Saos2	Antiproliferative activity assay	24 and 72 h	IC50 = 0.35 μM	24941130
SKOV3-MDR1-M6/6	Anticancer assay	48 h	IC50 = 0.97 μM	24946145
SKOV3	Anticancer assay	48 h	IC50 = 1 μM	24946145
MDA435/LCC6	Cytotoxicity assay	5 days	IC50 = 0.0026 μM	24952376
MDA435/LCC6MDR	Cytotoxicity assay	5 days	IC50 = 0.1493 μM	24952376
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.02581 μM	24996136
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.06727 μM	24996136
A549	Antiproliferative activity assay	48 h	IC50 = 1.525 μM	24996136
KB	Cytotoxicity assay	72 h	IC50 = 0.0039 μM	25008456
A549	Cytotoxicity assay	72 h	IC50 = 0.0057 μM	25008456
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0066 μM	25008456
KBVIN	Cytotoxicity assay	72 h	IC50 = 1.44 μM	25008456
MESSA	Cytotoxicity assay	72 h	IC50 = 0.004 μM	25025991
OVCAR8	Cytotoxicity assay	96 h	IC50 = 0.005 μM	25025991
MESSA/DX5	Cytotoxicity assay	72 h	IC50 = 1.764 μM	25025991
HepG2	Cytotoxicity assay	48 h	IC50 = 2.037 μM	25025991
NCI/ADR-RES	Cytotoxicity assay	96 h	IC50 = 3.3 μM	25025991
PC3	Cytotoxicity assay	48 h	IC50 = 3.99 μM	25025991
TCT1	Cytotoxicity assay	48 h	IC50 = 2.5 μM	25046128
CNE2	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	25061803
A549	Antiproliferative activity assay	48 h	IC50 = 0.005 μM	25061803
SW480	Antiproliferative activity assay	48 h	IC50 = 0.007 μM	25061803
A2780	Antiproliferative activity assay	48 h	IC50 = 0.015 μM	25061803
HCT8	Antiproliferative activity assay	48 h	IC50 = 0.021 μM	25061803
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.023 μM	25061803
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.028 μM	25061803
MCF7	Cytotoxicity assay	48 h	IC50 = 0.004 μM	25084144
A549	Cytotoxicity assay	48 h	IC50 = 0.082 μM	25084144
K562	Cytotoxicity assay	72 h	IC50 = 0.004 μM	25091926
A431	Cytotoxicity assay	72 h	IC50 = 0.007 μM	25091926
MDA-MB-435S	Cytotoxicity assay	72 h	IC50 = 0.009 μM	25091926
HeLa	Cytotoxicity assay	72 h	IC50 = 0.41 μM	25091926
HepG2	Cytotoxicity assay	72 h	IC50 = 0.99 μM	25091926
MDA-MB-DYT2	Cytotoxicity assay	4 days	IC50 = 0.00608 μM	25098528
MDA-MB-468	Cytotoxicity assay	4 days	IC50 = 0.00717 μM	25098528
NCI-N87	Cytotoxicity assay	4 days	IC50 = 0.00753 μM	25098528
NCI-H1975	Cytotoxicity assay	4 days	IC50 = 0.00794 μM	25098528
BT474	Cytotoxicity assay	4 days	IC50 = 0.00836 μM	25098528
MCF7	Cytotoxicity assay	48 h	IC50 = 0.2 μM	25176329
NCI-H358	Antiproliferative activity assay	48 h	IC50 = 0.002 μM	25208345
A2780S	Antiproliferative activity assay	48 h	IC50 = 0.004 μM	25208345
HCT8	Antiproliferative activity assay	48 h	IC50 = 0.005 μM	25208345
AGS	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	25208345
DLD1	Antiproliferative activity assay	48 h	IC50 = 0.016 μM	25208345
HCT116	Antiproliferative activity assay	48 h	IC50 = 0.018 μM	25208345
ES2	Antiproliferative activity assay	48 h	IC50 = 0.02 μM	25208345
U251	Antiproliferative activity assay	48 h	IC50 = 0.023 μM	25208345
HCT15	Antiproliferative activity assay	48 h	IC50 = 0.024 μM	25208345
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.038 μM	25208345
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.132 μM	25208345
C26	Antiproliferative activity assay	48 h	IC50 = 0.21 μM	25208345
HL60	Cytotoxicity assay	48 h	IC50 = 1.5 μM	25211032
K562	Cytotoxicity assay	48 h	IC50 = 2.4 μM	25211032
HepG2	Cytotoxicity assay	48 h	IC50 = 2.7 μM	25211032
MCF7	Cytotoxicity assay	48 h	IC50 = 3.2 μM	25211032
HT-29	Cytotoxicity assay	48 h	IC50 = 3.5 μM	25211032
KB	Cytotoxicity assay	48 h	IC50 = 3.8 μM	25211032
NCI-H1688	Cytotoxicity assay	24 h	IC50 = 0.85 μM	25226363
PC3	Cytotoxicity assay	24 h	IC50 = 0.94 μM	25226363
A549	Cytotoxicity assay	24 h	IC50 = 1.04 μM	25226363
DU145	Cytotoxicity assay	24 h	IC50 = 1.79 μM	25226363
A549	Antiproliferative activity assay	3 days	IC50 = 0.0024 μM	25241925
KB	Antiproliferative activity assay	3 days	IC50 = 0.0037 μM	25241925
DU145	Antiproliferative activity assay	3 days	IC50 = 0.00488 μM	25241925
KBVIN	Antiproliferative activity assay	3 days	IC50 = 1.58 μM	25241925
HeLa	Growth inhibition assay	48 h	GI50 = 0.025 μM	25264072
MiaPaCa	Growth inhibition assay	48 h	GI50 = 0.056 μM	25264072
IMR32	Growth inhibition assay	48 h	GI50 = 0.075 μM	25264072
MDA-MB-231	Growth inhibition assay	48 h	GI50 = 0.091 μM	25264072
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25375202
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25375202
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25375202
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25375202
SW480	Cytotoxicity assay	48 h	IC50 = 0.15 μM	25375202
HepG2	Cytotoxicity assay	3 days	IC50 = 0.00019 μM	25442315
KB	Cytotoxicity assay	3 days	IC50 = 0.0039 μM	25442315
MDA-MB-231	Antiproliferative activity assay	4 h	IC50 = 6.2 μM	25453798
MDA435	Cytotoxicity assay	24 h	IC50 = 0.005 μM	25462222
HL60	Cytotoxicity assay	24 h	IC50 = 0.007 μM	25462222
MES-SA	Cytotoxicity assay	24 h	IC50 = 0.008 μM	25462222
MDA-MB-231	Cytotoxicity assay	24 h	IC50 = 0.457 μM	25462222
MES-SA/Dx5	Cytotoxicity assay	24 h	IC50 = 5.1 μM	25462222
HeLa	Antiproliferative activity assay	48 h	GI50 = 0.025 μM	25462234
MiaPaCa	Antiproliferative activity assay	48 h	GI50 = 0.056 μM	25462234
IMR32	Antiproliferative activity assay	48 h	GI50 = 0.075 μM	25462234
MDA-MB-231	Antiproliferative activity assay	48 h	GI50 = 0.091 μM	25462234
HCT116	Cytotoxicity assay	72 h	IC50 = 0.004 μM	25462279
A549	Cytotoxicity assay	72 h	IC50 = 0.006 μM	25462279
HeLa	Cytotoxicity assay	72 h	IC50 = 0.008 μM	25462279
SKOV3	Cytotoxicity assay	48 h	IC50 = 0.001 μM	25462285
HCT116	Cytotoxicity assay	72 h	IC50 = 0.0027 μM	25499433
MCF7	Cytotoxicity assay	48 h	IC50 = 2.58 μM	25563891
A549	Cytotoxicity assay	48 h	IC50 = 4.9 μM	25563891
A375	Cytotoxicity assay	48 h	IC50 = 8 μM	25563891
LC2/ad	Antiproliferative activity assay	72 h	IC50 = 0.0025 μM	25625617
GSS	Antiproliferative activity assay	72 h	IC50 = 0.0034 μM	25625617
MKN45	Antiproliferative activity assay	72 h	IC50 = 0.004 μM	25625617
PC14	Antiproliferative activity assay	72 h	IC50 = 0.0044 μM	25625617
Lu116	Antiproliferative activity assay	72 h	IC50 = 0.0051 μM	25625617
LU99A	Antiproliferative activity assay	72 h	IC50 = 0.0052 μM	25625617
MIAPaCa2	Antiproliferative activity assay	72 h	IC50 = 0.0061 μM	25625617
HCT116	Antiproliferative activity assay	72 h	IC50 = 0.0061 μM	25625617
HT-29	Antiproliferative activity assay	72 h	IC50 = 0.007 μM	25625617
NCI-H358	Antiproliferative activity assay	72 h	IC50 = 0.0079 μM	25625617
HL60	Antiproliferative activity assay	72 h	IC50 = 0.0079 μM	25625617
NCI-H460	Antiproliferative activity assay	72 h	IC50 = 0.01 μM	25625617
MRC5	Antiproliferative activity assay	72 h	IC50 = 0.08 μM	25625617
HCT15	Antiproliferative activity assay	72 h	IC50 = 0.24 μM	25625617
HeLa	Cytotoxicity assay	48 h	IC50 = 0.01 μM	25647428
PC3	Cytotoxicity assay	48 h	IC50 = 0.012 μM	25647428
A549	Cytotoxicity assay	48 h	IC50 = 0.025 μM	25647428
MES-SA	Antiproliferative activity assay	48 h	GI50 = 0.007 μM	25671501
MES-SA/Dx5	Antiproliferative activity assay	48 h	GI50 = 9.8 μM	25671501
A549	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	25682561
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	25682561
A549/CDDP	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	25682561
A2780	Antiproliferative activity assay	48 h	IC50 = 0.006 μM	25682561
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.009 μM	25682561
SW480	Antiproliferative activity assay	48 h	IC50 = 0.021 μM	25682561
HCT8	Antiproliferative activity assay	48 h	IC50 = 0.066 μM	25682561
NIH/3T3	Antiproliferative activity assay	48 h	IC50 = 0.58 μM	25682561
A2780/TAX	Antiproliferative activity assay	48 h	IC50 = 4.4 μM	25682561
MCF7/DX	Antiproliferative activity assay	48 h	IC50 = 6.2 μM	25682561
MCF7	Cytotoxicity assay	48 h	IC50 = 0.032 μM	25728023
HepG2	Cytotoxicity assay	48 h	IC50 = 0.045 μM	25728023
HL60	Antiproliferative activity assay	72 h	IC50 = 0.0017 μM	25771484
HCT116	Antiproliferative activity assay	72 h	IC50 = 0.0049 μM	25771484
KB	Antiproliferative activity assay	72 h	IC50 = 0.015 μM	25771484
A549	Antiproliferative activity assay	72 h	IC50 = 0.058 μM	25771484
SMMC7721	Antiproliferative activity assay	72 h	IC50 = 0.12 μM	25771484
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25798528
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25798528
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25798528
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25798528
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25798528
HL60	Cytotoxicity assay	72 h	IC50 = 0.0018 μM	25819096
MOLT4	Cytotoxicity assay	72 h	IC50 = 0.0022 μM	25819096
U937	Cytotoxicity assay	72 h	IC50 = 0.0025 μM	25819096
HeLa	Cytotoxicity assay	72 h	IC50 = 0.0032 μM	25819096
DU145	Cytotoxicity assay	72 h	IC50 = 0.0034 μM	25819096
A549	Cytotoxicity assay	72 h	IC50 = 0.0044 μM	25819096
SGC7901	Cytotoxicity assay	72 h	IC50 = 0.0051 μM	25819096
K562	Cytotoxicity assay	72 h	IC50 = 0.0052 μM	25819096
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0062 μM	25819096
NCI-H1975	Cytotoxicity assay	72 h	IC50 = 0.0077 μM	25819096
MX1	Cytotoxicity assay	72 h	IC50 = 0.00559 μM	25819334
ID8	Cytotoxicity assay	72 h	IC50 = 0.0138 μM	25819334
L1210	Cytotoxicity assay	72 h	IC50 = 0.0276 μM	25819334
WI38	Cytotoxicity assay	72 h	IC50 = 0.0557 μM	25819334
MDA-MB-231	Antiproliferative activity assay	48 h	GI50 = 0.01 μM	25827522
A549	Antiproliferative activity assay	48 h	GI50 = 0.01 μM	25827522
PANC1	Antiproliferative activity assay	48 h	GI50 = 0.012 μM	25827522
HeLa	Antiproliferative activity assay	48 h	GI50 = 0.02 μM	25827522
HEK293	Cytotoxicity assay	72 h	IC50 = 0.04 μM	25842364
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25871261
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25871261
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25871261
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25871261
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	25871261
SCC114	Antiproliferative activity assay	72 h	IC50 = 0.0003 μM	25872984
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0019 μM	25882519
MDA-MB-435	Antiproliferative activity assay	48 h	IC50 = 0.0033 μM	25882519
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.0063 μM	25882519
SKOV3-MDR1-M6/6	Antiproliferative activity assay	48 h	IC50 = 1.1872 μM	25882519
A549	Antiproliferative activity assay	48 h	IC50 = 0.0023 μM	25937236
taxol-resistant A549	Antiproliferative activity assay	48 h	IC50 = 0.52 μM	25937236
EL4	Cytotoxicity assay	48 h	IC50 = 1.7 μM	25951057
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.38 μM	25959813
A549	Antiproliferative activity assay	48 h	IC50 = 2.82 μM	25959813
LCC-6	Cytotoxicity assay	3 days	IC50 = 0.0016 μM	25985195
MDA435/LCC6MDR	Cytotoxicity assay	3 days	IC50 = 0.1446 μM	25985195
A2780	Antiproliferative activity assay	2 days	IC50 = 0.028 μM	26042470
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	26068802
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	26068802
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	26068802
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	26068802
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	26068802
BEAS2B	Cytotoxicity assay	48 h	IC50 = 0.58 μM	26068802
NB4	Cytotoxicity assay	48 h	IC50 = 0.0023 μM	26132075
NCI-H1975	Cytotoxicity assay	72 h	IC50 = 0.0025 μM	26132075
OVCAR8	Cytotoxicity assay	48 h	IC50 = 0.0037 μM	26132075
MESSA	Cytotoxicity assay	72 h	IC50 = 0.004 μM	26132075
MDA-MB-468	Cytotoxicity assay	72 h	IC50 = 0.005 μM	26132075
A549	Cytotoxicity assay	72 h	IC50 = 0.007 μM	26132075
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.007 μM	26132075
MDA-MB-436	Cytotoxicity assay	72 h	IC50 = 0.008 μM	26132075
MESSA/DX5	Cytotoxicity assay	72 h	IC50 = 1.764 μM	26132075
HepG2	Cytotoxicity assay	48 h	IC50 = 2.6 μM	26132075
PC3	Cytotoxicity assay	48 h	IC50 = 4.9 μM	26132075
NCI-ADR-RES	Cytotoxicity assay	48 h	IC50 = 6 μM	26132075
KB	Antiproliferative activity assay	72 h	IC50 = 0.0051 μM	26160020
KB-7d	Antiproliferative activity assay	72 h	IC50 = 0.0084 μM	26160020
KB-S15	Antiproliferative activity assay	72 h	IC50 = 0.135 μM	26160020
U937	Cytotoxicity assay	72 h	IC50 = 2.1 μM	26316467
A549	Cytotoxicity assay	72 h	IC50 = 2.1 μM	26316467
MCF7	Cytotoxicity assay	72 h	IC50 = 2.3 μM	26316467
MOLT4	Cytotoxicity assay	72 h	IC50 = 2.7 μM	26316467
NCI-H1975	Cytotoxicity assay	72 h	IC50 = 2.8 μM	26316467
HeLa	Cytotoxicity assay	72 h	IC50 = 2.9 μM	26316467
DU145	Cytotoxicity assay	72 h	IC50 = 3.1 μM	26316467
K562	Cytotoxicity assay	72 h	IC50 = 3.8 μM	26316467
HL60	Cytotoxicity assay	72 h	IC50 = 3.8 μM	26316467
SGC7901	Cytotoxicity assay	72 h	IC50 = 9.8 μM	26316467
MES-SA	Cytotoxicity assay	48 h	GI50 = 0.007 μM	26360047
Rhabdomyosarcoma	Antiproliferative activity assay	96 h	IC50 = 0.0084 μM	26386818
HT-29	Cytotoxicity assay	3 days	IC50 = 0.0008 μM	26422131
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.001 μM	26448037
PC3	Cytotoxicity assay	72 h	IC50 = 0.001 μM	26448037
HCT116	Cytotoxicity assay	48 h	IC50 = 0.0028 μM	26448037
HepG2	Cytotoxicity assay	48 h	IC50 = 1.217 μM	26448037
H460	Cytotoxicity assay	48 h	IC50 = 4.287 μM	26448037
HeLa	Antiproliferative activity assay	72 h	IC50 = 2.29 μM	26602827
184B5	Antiproliferative activity assay	72 h	IC50 = 2.32 μM	26602827
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 2.56 μM	26602827
MDA-MB-468	Antiproliferative activity assay	72 h	IC50 = 3.87 μM	26602827
MCF7	Antiproliferative activity assay	72 h	IC50 = 3.99 μM	26602827
Jurkat	Cytotoxicity assay	48 h	IC50 = 0.0005 μM	26638041
U937	Cytotoxicity assay	48 h	IC50 = 0.006 μM	26638041
HeLa	Cytotoxicity assay	48 h	IC50 = 0.099 μM	26638041
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0039 μM	26690274
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0074 μM	26690274
U937	Cytotoxicity assay	72 h	IC50 = 0.00166 μM	26697718
HL60	Cytotoxicity assay	72 h	IC50 = 0.00199 μM	26697718
A549	Cytotoxicity assay	72 h	IC50 = 0.00212 μM	26697718
DU145	Cytotoxicity assay	72 h	IC50 = 0.0023 μM	26697718
HeLa	Cytotoxicity assay	72 h	IC50 = 0.00301 μM	26697718
HT-29	Cytotoxicity assay	72 h	IC50 = 0.00304 μM	26697718
K562	Cytotoxicity assay	72 h	IC50 = 0.00717 μM	26697718
MCF7	Cytotoxicity assay	72 h	IC50 = 0.00732 μM	26697718
NCI-H292	Cytotoxicity assay	72 h	IC50 = 0.006 μM	26712098
KB	Growth inhibition assay	72 h	GI50 = 0.001 μM	26778612
DU145	Antiproliferative activity assay	48 h	IC50 = 0.0038 μM	26785306
PC3	Antiproliferative activity assay	48 h	IC50 = 0.02 μM	26785306
A549	Antiproliferative activity assay	3 days	IC50 = 0.00003 μM	26865176
KB	Antiproliferative activity assay	3 days	IC50 = 0.00004 μM	26865176
MCF7	Antiproliferative activity assay	3 days	IC50 = 0.0039 μM	26865176
MDA-MB-231	Antiproliferative activity assay	3 days	IC50 = 0.018 μM	26865176
KBVIN	Antiproliferative activity assay	3 days	IC50 = 2.6 μM	26865176
PC3	Cytotoxicity assay	72 h	IC50 = 0.002 μM	26904921
SKOV3	Cytotoxicity assay	72 h	IC50 = 0.0047 μM	26974508
A549	Cytotoxicity assay	48 h	IC50 = 0.0132 μM	26985296
SKMES1	Cytotoxicity assay	48 h	IC50 = 0.0135 μM	26985296
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0189 μM	26985296
WPMY-1	Cytotoxicity assay	48 h	GI50 = 0.01 μM	26994690
A549	Antiproliferative activity assay	48 h	GI50 = 0.01 μM	26994690
MDA-MB-231	Antiproliferative activity assay	48 h	GI50 = 0.01 μM	26994690
HeLa	Antiproliferative activity assay	48 h	GI50 = 0.023 μM	26994690
HepG2	Antiproliferative activity assay	48 h	IC50 = 0.02171 μM	27017265
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.02581 μM	27017265
HCT116	Antiproliferative activity assay	48 h	IC50 = 0.06727 μM	27017265
A2780	Cytotoxicity assay	48 h	IC50 = 0.005 μM	27149641
A549	Cytotoxicity assay	48 h	IC50 = 0.009 μM	27149641
MCF7	Cytotoxicity assay	48 h	IC50 = 0.012 μM	27149641
HCT8	Cytotoxicity assay	48 h	IC50 = 0.019 μM	27149641
A549/CDDP	Cytotoxicity assay	48 h	IC50 = 0.023 μM	27149641
HCT8/VCT	Cytotoxicity assay	48 h	IC50 = 0.125 μM	27149641
MCF7/DX	Cytotoxicity assay	48 h	IC50 = 0.135 μM	27149641
A2780/TAX	Cytotoxicity assay	48 h	IC50 = 5.68 μM	27149641
HeLa	Antiproliferative activity assay	48 h	GI50 = 0.025 μM	27209232
MiaPaCa	Antiproliferative activity assay	48 h	GI50 = 0.056 μM	27209232
IMR32	Antiproliferative activity assay	48 h	GI50 = 0.075 μM	27209232
MDA-MB-231	Antiproliferative activity assay	48 h	GI50 = 0.091 μM	27209232
PC3	Antiproliferative activity assay	72 h	IC50 = 0.002 μM	27214307
NCI-H1993	Antiproliferative activity assay	48 to 96 h	GI50 = 0.004 μM	27218860
MES-SA	Antiproliferative activity assay	48 to 96 h	GI50 = 0.007 μM	27218860
NCI-H2073	Antiproliferative activity assay	48 to 96 h	GI50 = 2.4 μM	27218860
KBVIN	Antiproliferative activity assay	48 h	GI50 = 2.6 μM	27238842
A549	Antiproliferative activity assay	48 h	GI50 = 2.6 μM	27238842
MCF7	Cytotoxicity assay	72 h	IC50 = 0.00125 μM	27311893
HeLa	Cytotoxicity assay	72 h	IC50 = 0.01262 μM	27311893
MDA-MB-231	Anticancer assay	72 h	IC50 = 0.003388 μM	27317645
HeLa	Anticancer assay	72 h	IC50 = 0.01987 μM	27317645
HT-29	Cytotoxicity assay	72 h	IC50 = 0.02 μM	27329938
PC3	Cytotoxicity assay	72 h	IC50 = 0.03 μM	27329938
HL-7702	Cytotoxicity assay	72 h	IC50 = 0.06 μM	27329938
A549	Cytotoxicity assay	72 h	IC50 = 0.08 μM	27329938
HepG2	Cytotoxicity assay	72 h	IC50 = 0.2 μM	27329938
MCF7	Cytotoxicity assay	96 h	IC50 = 0.0002 μM	27434426
HeLa	Cytotoxicity assay	96 h	IC50 = 0.0064 μM	27434426
NCI60	Cytotoxicity assay	48 h	GI50 = 0.0315 μM	27448924
HepG2	Cytotoxicity assay	48 h	IC50 = 0.006 μM	27627130
Hep3B	Cytotoxicity assay	48 h	IC50 = 0.02 μM	27627130
A549	Cytotoxicity assay	48 h	IC50 = 0.03 μM	27627130
MCF7	Cytotoxicity assay	48 h	IC50 = 0.06 μM	27627130
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
HeLa	Cytotoxicity assay	48 h	IC50 = 0.008 μM	27704807
A549	Cytotoxicity assay	48 h	IC50 = 0.02 μM	27704822
MCF7	Cytotoxicity assay	48 h	IC50 = 0.1 μM	27704822
HeLa	Cytotoxicity assay	72 h	IC50 = 1.7 μM	27748595
K562	Cytotoxicity assay	72 h	IC50 = 2.7 μM	27748595
HCT116	Cytotoxicity assay	72 h	IC50 = 3.3 μM	27748595
A549	Cytotoxicity assay	72 h	IC50 = 5.5 μM	27748595
HepG2	Cytotoxicity assay	72 h	IC50 = 6.7 μM	27748595
HELF	Cytotoxicity assay	24 h	IC50 = 7.14 μM	27769031
BGC823	Cytotoxicity assay	24 h	IC50 = 9.26 μM	27769031
KB	Cytotoxicity assay	48 h	IC50 = 0.0008 μM	27797192
A549	Cytotoxicity assay	48 h	IC50 = 0.00099 μM	27797192
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 0.00305 μM	27797192
MCF7	Cytotoxicity assay	48 h	IC50 = 0.02275 μM	27797192
KBVIN	Cytotoxicity assay	48 h	IC50 = 1.896 μM	27797192
HCT116	Cytotoxicity assay	48 h	IC50 = 0.1 μM	27887843
Bel7402	Cytotoxicity assay	48 h	IC50 = 0.1 μM	27887843
OVCAR8	Growth inhibition assay	96 h	IC50 = 5 μM	27894589
HeLa	Growth inhibition assay	96 h	IC50 = 5.3 μM	27894589
HeLa	Growth inhibition assay	48 h	GI50 = 0.0389 μM	27964883
MiaPaCa	Growth inhibition assay	48 h	GI50 = 0.06 μM	27964883
IMR32	Growth inhibition assay	48 h	GI50 = 0.086 μM	27964883
MDA-MB-231	Growth inhibition assay	48 h	GI50 = 0.092 μM	27964883
DU145	Antiproliferative activity assay	48 h	IC50 = 0.011 μM	27979593
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.036 μM	27979593
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.63 μM	27979593
ECA109	Antiproliferative activity assay	48 h	IC50 = 0.94 μM	27979593
MDA-MB-435	Cytotoxicity assay	72 h	IC50 = 0.0002 μM	27983842
HT-29	Cytotoxicity assay	72 h	IC50 = 0.0008 μM	27983842
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0027 μM	27983842
OVCAR3	Cytotoxicity assay	72 h	IC50 = 0.0033 μM	27983842
H1299	Cytotoxicity assay	24 h	IC50 = 1.5 μM	27983842
HEK-Blue	Function assay	3 h	IC50 = 7.94328 μM	28075581
A549	Antiproliferative activity assay	72 h	IC50 = 0.0062 μM	28099003
KB	Antiproliferative activity assay	72 h	IC50 = 0.00627 μM	28099003
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 0.00882 μM	28099003
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.0104 μM	28099003
KBVIN	Antiproliferative activity assay	72 h	IC50 = 1.926 μM	28099003
A549	Cytotoxicity assay	48 h	IC50 = 6.195 μM	28237662
KB	Cytotoxicity assay	48 h	IC50 = 6.587 μM	28237662
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 9.384 μM	28237662
HeLa	Cytotoxicity assay	72 h	IC50 = 0.0014 μM	28240909
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0026 μM	28252962
MDA-MB-435	Cytotoxicity assay	72 h	IC50 = 0.0031 μM	28252962
OVCAR3	Cytotoxicity assay	72 h	IC50 = 0.0075 μM	28252962
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 0.08 μM	28262526
MRC5	Cytotoxicity assay	72 h	IC50 = 0.00052 μM	28282127
A549	Antiproliferative activity assay	72 h	IC50 = 0.0062 μM	28290698
KB	Antiproliferative activity assay	72 h	IC50 = 0.0063 μM	28290698
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 0.0088 μM	28290698
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.0104 μM	28290698
KBVIN	Antiproliferative activity assay	72 h	IC50 = 1.926 μM	28290698
PC3	Antiproliferative activity assay	72 h	IC50 = 0.004 μM	28335606
UACC62	Antiproliferative activity assay	72 h	IC50 = 0.006 μM	28335606
M14	Antiproliferative activity assay	72 h	IC50 = 0.007 μM	28335606
SK-MEL-2	Antiproliferative activity assay	72 h	IC50 = 0.009 μM	28335606
NCI-H460	Antiproliferative activity assay	72 h	IC50 = 0.01 μM	28335606
A375	Antiproliferative activity assay	72 h	IC50 = 0.01 μM	28335606
SF295	Antiproliferative activity assay	72 h	IC50 = 0.056 μM	28335606
ACHN	Antiproliferative activity assay	72 h	IC50 = 0.066 μM	28335606
HeLa	Cytotoxicity assay	48 h	IC50 = 0.00821 μM	28340411
A549	Cytotoxicity assay	48 h	IC50 = 0.00952 μM	28340411
A549/TR	Cytotoxicity assay	48 h	IC50 = 1.51 μM	28340411
HeLa/TR	Cytotoxicity assay	48 h	IC50 = 1.53 μM	28340411
LO2	Cytotoxicity assay	72 h	IC50 = 0.002 μM	28395199
A549	Antiproliferative activity assay	72 h	IC50 = 0.023 μM	28395199
HT-29	Antiproliferative activity assay	72 h	IC50 = 0.025 μM	28395199
NCI-H596	Antiproliferative activity assay	72 h	IC50 = 0.035 μM	28395199
HT-29	Cytotoxicity assay	3 days	IC50 = 0.0014 μM	28409637
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0015 μM	28433513
MDA-MB-435	Antiproliferative activity assay	48 h	IC50 = 0.002 μM	28433513
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	28433513
SKOV3-MDR1-M6/6	Antiproliferative activity assay	48 h	IC50 = 2.33 μM	28433513
A2780	Antiproliferative activity assay	2 days	IC50 = 0.028 μM	28463001
BGC823	Cytotoxicity assay	96 h	IC50 = 0.0008 μM	28530828
NCI-H460	Cytotoxicity assay	96 h	IC50 = 0.001 μM	28530828
HepG2	Cytotoxicity assay	96 h	IC50 = 0.0063 μM	28530828
OVPF008	Antiproliferative activity assay	6 days	IC50 = 1.1 μM	28548825
OVPF038	Antiproliferative activity assay	6 days	IC50 = 1.4 μM	28548825
KB	Cytotoxicity assay	72 h	IC50 = 0.0036 μM	28590124
KBv200	Cytotoxicity assay	72 h	IC50 = 2.117 μM	28590124
MDA-MB-435	Cytotoxicity assay	72 h	IC50 = 0.0005 μM	28594169
OVCAR3	Cytotoxicity assay	72 h	IC50 = 0.002 μM	28594169
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.009 μM	28594169
U937	Cytotoxicity assay	72 h	IC50 = 0.0017 μM	28598633
HL60	Cytotoxicity assay	72 h	IC50 = 0.002 μM	28598633
A549	Cytotoxicity assay	72 h	IC50 = 0.0021 μM	28598633
DU145	Cytotoxicity assay	72 h	IC50 = 0.0023 μM	28598633
HeLa	Cytotoxicity assay	72 h	IC50 = 0.003 μM	28598633
HT-29	Cytotoxicity assay	72 h	IC50 = 0.003 μM	28598633
K562	Cytotoxicity assay	72 h	IC50 = 0.0072 μM	28598633
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0073 μM	28598633
A2780	Cytotoxicity assay	48 h	IC50 = 0.00107 μM	28624703
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0011 μM	28624703
KB	Cytotoxicity assay	48 h	IC50 = 0.0019 μM	28624703
Hela-beta3	Cytotoxicity assay	48 h	IC50 = 0.009 μM	28624703
A2780AD	Cytotoxicity assay	48 h	IC50 = 1.282 μM	28624703
KBV1	Cytotoxicity assay	48 h	IC50 = 9.8 μM	28624703
BGC823	Growth inhibition assay	3 days	IC50 = 0.001 μM	28625363
HepG2	Growth inhibition assay	3 days	IC50 = 0.02 μM	28625363
HCT116	Growth inhibition assay	3 days	IC50 = 0.03 μM	28625363
A2780	Growth inhibition assay	3 days	IC50 = 0.03 μM	28625363
NCI-H1650	Growth inhibition assay	3 days	IC50 = 0.07 μM	28625363
A2780	Antiproliferative activity assay	2 days	IC50 = 0.0137 μM	28648491
KB	Cytotoxicity assay	48 h	GI50 = 0.00512 μM	28653846
A549	Cytotoxicity assay	48 h	GI50 = 0.00703 μM	28653846
MDA-MB-231	Cytotoxicity assay	48 h	GI50 = 0.01 μM	28653846
MCF7	Cytotoxicity assay	48 h	GI50 = 0.0119 μM	28653846
KBVIN	Cytotoxicity assay	48 h	GI50 = 2.716 μM	28653846
MCF7	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	28654256
HL60	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	28654256
SMMC7721	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	28654256
A549	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	28654256
SW480	Antiproliferative activity assay	48 h	IC50 = 0.008 μM	28654256
A375	Antiproliferative activity assay	48 h	IC50 = 0.7 μM	28667872
MIAPaCa2	Antiproliferative activity assay	48 h	IC50 = 2.5 μM	28667872
HEY	Cytotoxicity assay	48 h	IC50 = 0.1041 μM	28719204
A2780	Cytotoxicity assay	48 h	IC50 = 0.1642 μM	28719204
HCT116	Growth inhibition assay	96 h	IC50 = 0.0002 μM	28737396
BGC823	Growth inhibition assay	96 h	IC50 = 0.0006 μM	28737396
HepG2	Growth inhibition assay	96 h	IC50 = 0.0076 μM	28737396
A2780	Growth inhibition assay	96 h	IC50 = 0.0204 μM	28737396
A549	Growth inhibition assay	4 days	GI50 = 0.0037 μM	28740601
PC3	Growth inhibition assay	4 days	GI50 = 0.0058 μM	28740601
NCI-H460	Cytotoxicity assay	72 h	IC50 = 0.006 μM	28740613
HT-29	Cytotoxicity assay	72 h	IC50 = 0.014 μM	28740613
A2780S	Antiproliferative activity assay	48 h	IC50 = 0.0123 μM	28763646
HCT8	Antiproliferative activity assay	48 h	IC50 = 0.0174 μM	28763646
HCT8/T	Antiproliferative activity assay	48 h	IC50 = 9.885 μM	28763646
A549	Cytotoxicity assay	24 h	IC50 = 0.0041 μM	28835794
LNCAP	Antiproliferative activity assay	72 h	IC50 = 0.0019 μM	28857558
PA1	Antiproliferative activity assay	72 h	IC50 = 0.003 μM	28857558
HCT116	Antiproliferative activity assay	72 h	IC50 = 0.0041 μM	28857558
MDA-MB-468	Antiproliferative activity assay	72 h	IC50 = 0.0054 μM	28857558
HCT116/VP35	Antiproliferative activity assay	72 h	IC50 = 0.0063 μM	28857558
NCI-H520	Antiproliferative activity assay	72 h	IC50 = 0.0082 μM	28857558
LS174T	Antiproliferative activity assay	72 h	IC50 = 0.0095 μM	28857558
MCF10A	Cytotoxicity assay	72 h	IC50 = 0.0058 μM	28926237
MDA-MB-468	Cytotoxicity assay	72 h	IC50 = 0.0061 μM	28926237
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0088 μM	28926237
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.059 μM	28926237
HeLa	Cytotoxicity assay	72 h	IC50 = 0.001 μM	29043798
A2780	Cytotoxicity assay	2 days	IC50 = 0.013 μM	29048892
A549	Cytotoxicity assay	72 h	IC50 = 0.0062 μM	29131631
KB	Cytotoxicity assay	72 h	IC50 = 0.0066 μM	29131631
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0094 μM	29131631
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0114 μM	29131631
KBVIN	Cytotoxicity assay	72 h	IC50 = 1.86 μM	29131631
A2780	Function assay	48 h	GI50 = 0.00753 μM	29138028
OVCAR5	Function assay	48 h	GI50 = 0.021 μM	29138028
HCT116	Antiproliferative activity assay	48 h	IC50 = 1.37 μM	29172082
PC3	Antiproliferative activity assay	48 h	IC50 = 4.57 μM	29172082
HeLa	Antiproliferative activity assay	48 h	IC50 = 6.42 μM	29172082
H1299	Antiproliferative activity assay	48 h	IC50 = 7.83 μM	29172082
HCT116	Antiproliferative activity assay	48 h	IC50 = 0.014 μM	29223717
MCF7	Antiproliferative activity assay	48 h	IC50 = 1.428 μM	29223717
143B	Antiproliferative activity assay	48 h	IC50 = 5.56 μM	29223717
MES-SA/Dx5	Growth inhibition assay	72 h	IC50 = 0.21 μM	29251920
MDA435/LCC6	Growth inhibition assay	72 h	IC50 = 0.346 μM	29251920
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29286250
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29286250
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29286250
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29286250
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29286250
A2780	Antiproliferative activity assay	48 h	IC50 = 0.001 μM	29306206
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.002 μM	29306206
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	29306206
MDA-MB-231	Antiproliferative activity assay	48 h	IC50 = 0.003 μM	29306206
KB	Antiproliferative activity assay	72 h	IC50 = 0.0036 μM	29319316
A549	Antiproliferative activity assay	72 h	IC50 = 0.0045 μM	29319316
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 0.007 μM	29319316
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.0088 μM	29319316
KBVIN	Antiproliferative activity assay	72 h	IC50 = 2.36 μM	29319316
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338226
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338226
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338226
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338226
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338226
SMMC7721	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338260
A549	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338260
MCF7	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338260
SW480	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338260
HL60	Cytotoxicity assay	48 h	IC50 = 0.008 μM	29338260
HT-29	Cytotoxicity assay	72 h	IC50 = 0.0008 μM	29350920
HeLa	Cytotoxicity assay	48 h	IC50 = 0.0046 μM	29359935
A2780	Cytotoxicity assay	48 h	IC50 = 0.0134 μM	29359935
Hela-beta3	Cytotoxicity assay	48 h	IC50 = 0.041 μM	29359935
HL60	Cytotoxicity assay	48 h	IC50 = 0.002 μM	29373791
LS180	Cytotoxicity assay	48 h	IC50 = 0.0028 μM	29373791
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 0.003 μM	29373791
A549	Cytotoxicity assay	48 h	IC50 = 0.0068 μM	29373791
HCT116	Cytotoxicity assay	24 h	IC50 = 0.02 μM	29395979
SW480	Cytotoxicity assay	24 h	IC50 = 0.19 μM	29395979
T98G	Cytotoxicity assay	24 h	IC50 = 0.74 μM	29395979
U87	Cytotoxicity assay	24 h	IC50 = 4.67 μM	29395979
DU145	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	29406710
PC3	Cytotoxicity assay	72 h	IC50 = 0.0037 μM	29406710
PC3-TxR	Cytotoxicity assay	72 h	IC50 = 0.1107 μM	29406710
ViBo	Antiproliferative activity assay	24 h	IC50 = 1.59 μM	29407986
CaSki	Antiproliferative activity assay	24 h	IC50 = 2.9 μM	29407986
A549	Growth inhibition assay	48 h	IC50 = 0.008 μM	29412669
HL60	Growth inhibition assay	48 h	IC50 = 0.008 μM	29412669
MCF7	Growth inhibition assay	48 h	IC50 = 0.008 μM	29412669
SMMC7721	Growth inhibition assay	48 h	IC50 = 0.008 μM	29412669
SW480	Growth inhibition assay	48 h	IC50 = 0.008 μM	29412669
HCT116	Growth inhibition assay	72 h	IC50 = 0.0041 μM	29439899
paclitaxel-resistant MCF7	Cytotoxicity assay	72 h	IC50 = 2.29087 μM	29468872
HL60	Antiproliferative activity assay	48 h	IC50 = 0.0026 μM	29475587
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.023 μM	29475587
293T	Cytotoxicity assay	4 days	IC50 = 0.0023 μM	29486949
HAC	Cytotoxicity assay	4 days	IC50 = 0.0121 μM	29486949
KB-3-1	Cytotoxicity assay	72 h	IC50 = 0.0005 μM	29501942
SW620	Cytotoxicity assay	72 h	IC50 = 0.03 μM	29501942
KB-C2	Cytotoxicity assay	72 h	IC50 = 0.25 μM	29501942
SW620/AD300	Cytotoxicity assay	72 h	IC50 = 1.97 μM	29501942
A549	Antiproliferative activity assay	72 h	IC50 = 0.007 μM	29501947
A549/TR	Antiproliferative activity assay	72 h	IC50 = 3.112 μM	29501947
SKOV3	Cytotoxicity assay	72 to 120 h	IC50 = 0.00239 μM	29517223
HEY	Cytotoxicity assay	72 to 120 h	IC50 = 2.7 μM	29517223
SKVLB1	Function assay	72 to 120 h	IC50 = 3.733 μM	29517223
A2780cis	Growth inhibition assay	72 h	IC50 = 0.003 μM	29519737
A2780	Growth inhibition assay	72 h	IC50 = 0.009 μM	29519737
OVCAR8	Growth inhibition assay	72 h	IC50 = 0.01 μM	29519737
ovarian epithelial	Growth inhibition assay	48 h	IC50 = 0.03 μM	29519737
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0024 μM	29648818
PC9	Cytotoxicity assay	72 h	IC50 = 0.0027 μM	29648818
A549	Cytotoxicity assay	72 h	IC50 = 0.0032 μM	29648818
HCC2998	Growth inhibition assay	48 h	GI50 = 0.001 μM	29655610
NCI-H226	Growth inhibition assay	48 h	GI50 = 0.0039 μM	29655610
SW620	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
OVCAR3	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
MCF7	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
HL-60(TB)	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
HCT116	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
MDA-MB-435	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
BT549	Growth inhibition assay	48 h	GI50 = 0.004 μM	29655610
SF539	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
KM12	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
UACC62	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
LOXIMVI	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
M14	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
SF268	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
MOLT4	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
HT-29	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
Hs578T	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
SK-MEL-5	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
CCRF-CEM	Growth inhibition assay	48 h	GI50 = 0.005 μM	29655610
NCI-H23	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
U251	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
SN12C	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
IGROV1	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
A549/ATCC	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
PC3	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
DU145	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
NCI-H460	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
K562	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
SR	Growth inhibition assay	48 h	GI50 = 0.0063 μM	29655610
SNB75	Growth inhibition assay	48 h	GI50 = 0.0079 μM	29655610
A498	Growth inhibition assay	48 h	GI50 = 0.0079 μM	29655610
COLO205	Growth inhibition assay	48 h	GI50 = 0.0079 μM	29655610
OVCAR5	Growth inhibition assay	48 h	GI50 = 0.0079 μM	29655610
OVCAR8	Growth inhibition assay	48 h	GI50 = 0.0079 μM	29655610
SNB19	Growth inhibition assay	48 h	GI50 = 0.01 μM	29655610
NCI-H322M	Growth inhibition assay	48 h	GI50 = 0.0125 μM	29655610
MDA-MB-468	Growth inhibition assay	48 h	GI50 = 0.0125 μM	29655610
MDA-MB-231	Growth inhibition assay	48 h	GI50 = 0.0125 μM	29655610
RXF393	Growth inhibition assay	48 h	GI50 = 0.0158 μM	29655610
NCI-H522	Growth inhibition assay	48 h	GI50 = 0.0158 μM	29655610
HOP62	Growth inhibition assay	48 h	GI50 = 0.019 μM	29655610
TK10	Growth inhibition assay	48 h	GI50 = 0.0199 μM	29655610
RPMI8226	Growth inhibition assay	48 h	GI50 = 0.0199 μM	29655610
HOP92	Growth inhibition assay	48 h	GI50 = 0.025 μM	29655610
SF295	Growth inhibition assay	48 h	GI50 = 0.025 μM	29655610
786-0	Growth inhibition assay	48 h	GI50 = 0.039 μM	29655610
MALME-3M	Growth inhibition assay	48 h	GI50 = 0.05 μM	29655610
EKVX	Growth inhibition assay	48 h	GI50 = 0.079 μM	29655610
UO31	Growth inhibition assay	48 h	GI50 = 0.125 μM	29655610
HCT15	Growth inhibition assay	48 h	GI50 = 0.125 μM	29655610
ACHN	Growth inhibition assay	48 h	GI50 = 0.158 μM	29655610
Caki1	Growth inhibition assay	48 h	GI50 = 0.158 μM	29655610
SK-MEL-28	Growth inhibition assay	48 h	GI50 = 0.4 μM	29655610
SK-MEL-2	Growth inhibition assay	48 h	GI50 = 0.4 μM	29655610
NCI/ADR-RES	Growth inhibition assay	48 h	GI50 = 0.63 μM	29655610
OVCAR4	Growth inhibition assay	48 h	GI50 = 0.63 μM	29655610
SKHEP1	Growth inhibition assay	48 h	GI50 = 0.011 μM	29655982
PC3	Growth inhibition assay	48 h	GI50 = 0.013 μM	29655982
HT-29	Cytotoxicity assay	24 to 72 h	IC50 = 0.011 μM	29656990
OVCAR3	Cytotoxicity assay	24 to 72 h	IC50 = 0.011 μM	29656990
OVCAR8	Growth inhibition assay	96 h	IC50 = 0.004 μM	29730191
MCF7	Growth inhibition assay	96 h	IC50 = 0.0055 μM	29730191
HepG2	Growth inhibition assay	48 h	IC50 = 2.66 μM	29730191
NCI/ADR-RES	Growth inhibition assay	96 h	IC50 = 3.1 μM	29730191
A2780	Cytotoxicity assay	2 days	IC50 = 0.013 μM	29738243
A2780S	Antiproliferative activity assay	48 to 72 h	IC50 = 0.01894 μM	29754076
A549	Antiproliferative activity assay	48 to 72 h	IC50 = 0.02318 μM	29754076
A549/TR	Antiproliferative activity assay	48 to 72 h	IC50 = 0.75939 μM	29754076
MCF7	Cytotoxicity assay	48 h	IC50 = 0.005 μM	29759727
MIAPaCa2	Cytotoxicity assay	48 h	IC50 = 0.006 μM	29759727
PC3	Cytotoxicity assay	48 h	IC50 = 0.007 μM	29759727
HeLaS3	Antiproliferative activity assay	72 h	IC50 = 0.013 μM	29803003
KBVIN	Antiproliferative activity assay	72 h	IC50 = 1.01 μM	29803003
MCF7	Cytotoxicity assay	4 days	IC50 = 0.008 μM	29884535
HL60	Cytotoxicity assay	4 days	IC50 = 0.008 μM	29884535
SMMC7721	Cytotoxicity assay	4 days	IC50 = 0.008 μM	29884535
A549	Cytotoxicity assay	4 days	IC50 = 0.008 μM	29884535
SW480	Cytotoxicity assay	4 days	IC50 = 0.008 μM	29884535
A549	Antiproliferative activity assay	72 h	IC50 = 0.0063 μM	30010341
KB	Antiproliferative activity assay	72 h	IC50 = 0.0068 μM	30010341
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 0.0081 μM	30010341
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.0112 μM	30010341
KBVIN	Antiproliferative activity assay	72 h	IC50 = 2.786 μM	30010341
MCF7	Cytotoxicity assay	72 h	IC50 = 0.0096 μM	30036834
KB	Cytotoxicity assay	72 h	IC50 = 0.0103 μM	30036834
KB/VCR	Cytotoxicity assay	72 h	IC50 = 4 μM	30036834
HT-29	Cytotoxicity assay	72 h	IC50 = 0.009 μM	30057155
MDA-MB-435	Cytotoxicity assay	72 h	IC50 = 0.013 μM	30057155
OVCAR3	Cytotoxicity assay	72 h	IC50 = 0.013 μM	30057155
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.017 μM	30057155
HeLa	Antiproliferative activity assay	72 h	IC50 = 0.0028 μM	30098869
MDA-MB-435	Antiproliferative activity assay	72 h	IC50 = 0.0045 μM	30098869
SKOV3	Antiproliferative activity assay	72 h	IC50 = 0.005 μM	30098869
wild-type Hela-beta3	Antiproliferative activity assay	72 h	IC50 = 0.024 μM	30098869
SKOV3-MDR1-M6/6	Antiproliferative activity assay	72 h	IC50 = 1.2 μM	30098869
A375	Antiproliferative activity assay	72 h	IC50 = 0.0478 μM	30099258
KB	Antiproliferative activity assay	72 h	IC50 = 0.00571 μM	30106296
MCF7	Antiproliferative activity assay	72 h	IC50 = 0.00752 μM	30106296
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 0.00851 μM	30106296
A549	Antiproliferative activity assay	72 h	IC50 = 0.00876 μM	30106296
KBVIN	Antiproliferative activity assay	72 h	IC50 = 2.383 μM	30106296
PC3	Cytotoxicity assay	72 h	IC50 = 0.0011 μM	30122035
DU145	Cytotoxicity assay	72 h	IC50 = 0.0015 μM	30122035
PC3-TxR	Cytotoxicity assay	72 h	IC50 = 0.1139 μM	30122035
KB	Antiproliferative activity assay	72 h	IC50 = 5.9 μM	30189396
A549	Antiproliferative activity assay	72 h	IC50 = 6.8 μM	30189396
MDA-MB-231	Antiproliferative activity assay	72 h	IC50 = 9.6 μM	30189396
MDA-MB-231	Cytotoxicity assay	72 h	IC50 = 0.0026 μM	30192537
MDA-MB-435	Cytotoxicity assay	72 h	IC50 = 0.0031 μM	30192537
OVCAR3	Cytotoxicity assay	72 h	IC50 = 0.0075 μM	30192537
MV411	Antiproliferative activity assay	72 h	IC50 = 0.017 μM	30212198
HGC27	Antiproliferative activity assay	72 h	IC50 = 0.028 μM	30212198
HeLa	Antiproliferative activity assay	72 h	IC50 = 0.046 μM	30212198
A549	Antiproliferative activity assay	72 h	IC50 = 0.051 μM	30212198
HeLa	Antiproliferative activity assay	48 h	IC50 = 0.0028 μM	30297118
SKOV3	Antiproliferative activity assay	48 h	IC50 = 0.005 μM	30297118
SKOV3-MDR1-M6/6	Antiproliferative activity assay	48 h	IC50 = 1.2 μM	30297118
HCC1806	Antiproliferative activity assay	24 h	IC50 = 0.001 μM	30392953
BEAS2B	Antiproliferative activity assay	24 h	IC50 = 0.007 μM	30392953
HT-29	Antiproliferative activity assay	24 h	IC50 = 0.008 μM	30392953
HepG2	Antiproliferative activity assay	24 h	IC50 = 0.009 μM	30392953
PANC1	Antiproliferative activity assay	24 h	IC50 = 0.04 μM	30392953
MDA-MB-231	Cytotoxicity assay	48 h	IC50 = 0.004 μM	30433783
A549	Cytotoxicity assay	48 h	IC50 = 0.004 μM	30433783
PANC1	Cytotoxicity assay	48 h	IC50 = 0.06 μM	30433783
4T1	Cytotoxicity assay	48 h	IC50 = 0.094 μM	30433783
A375	Cytotoxicity assay	48 h	IC50 = 0.1 μM	30433783
LLC	Cytotoxicity assay	48 h	IC50 = 0.189 μM	30433783
B16F10	Cytotoxicity assay	48 h	IC50 = 0.53 μM	30433783
B16F10 spheroid	Cytotoxicity assay	48 h	IC50 = 8.01 μM	30433783
Daudi	Growth Inhibition Assay		IC50 = 0.01708 μM	SANGER
NCI-SNU-5	Growth Inhibition Assay		IC50 = 0.01701 μM	SANGER
LS-123	Growth Inhibition Assay		IC50 = 0.01664 μM	SANGER
MOLT-13	Growth Inhibition Assay		IC50 = 0.01637 μM	SANGER
SNB75	Growth Inhibition Assay		IC50 = 0.0154 μM	SANGER
K-562	Growth Inhibition Assay		IC50 = 0.01516 μM	SANGER
TE-5	Growth Inhibition Assay		IC50 = 0.01496 μM	SANGER
SNU-C2B	Growth Inhibition Assay		IC50 = 0.01496 μM	SANGER
CTV-1	Growth Inhibition Assay		IC50 = 0.01478 μM	SANGER
GI-1	Growth Inhibition Assay		IC50 = 0.01373 μM	SANGER
L-363	Growth Inhibition Assay		IC50 = 0.01351 μM	SANGER
ES1	Growth Inhibition Assay		IC50 = 0.01288 μM	SANGER
HOP-62	Growth Inhibition Assay		IC50 = 0.01276 μM	SANGER
KARPAS-45	Growth Inhibition Assay		IC50 = 0.0127 μM	SANGER
RXF393	Growth Inhibition Assay		IC50 = 0.01257 μM	SANGER
RPMI-8402	Growth Inhibition Assay		IC50 = 0.01256 μM	SANGER
KE-37	Growth Inhibition Assay		IC50 = 0.01234 μM	SANGER
NCI-H1436	Growth Inhibition Assay		IC50 = 0.01231 μM	SANGER
NALM-6	Growth Inhibition Assay		IC50 = 0.01214 μM	SANGER
ST486	Growth Inhibition Assay		IC50 = 0.01204 μM	SANGER
SCC-3	Growth Inhibition Assay		IC50 = 0.01204 μM	SANGER
DOHH-2	Growth Inhibition Assay		IC50 = 0.01203 μM	SANGER
HD-MY-Z	Growth Inhibition Assay		IC50 = 0.01163 μM	SANGER
SF268	Growth Inhibition Assay		IC50 = 0.01151 μM	SANGER
SK-PN-DW	Growth Inhibition Assay		IC50 = 0.01112 μM	SANGER
RPMI-8226	Growth Inhibition Assay		IC50 = 0.01102 μM	SANGER
LB647-SCLC	Growth Inhibition Assay		IC50 = 0.01051 μM	SANGER
QIMR-WIL	Growth Inhibition Assay		IC50 = 0.01033 μM	SANGER
SR	Growth Inhibition Assay		IC50 = 0.01026 μM	SANGER
Calu-6	Growth Inhibition Assay		IC50 = 0.01012 μM	SANGER
NCI-SNU-16	Growth Inhibition Assay		IC50 = 0.01008 μM	SANGER
COR-L279	Growth Inhibition Assay		IC50 = 0.00999 μM	SANGER
HL-60	Growth Inhibition Assay		IC50 = 0.009656 μM	SANGER
A101D	Growth Inhibition Assay		IC50 = 0.009598 μM	SANGER
BL-41	Growth Inhibition Assay		IC50 = 0.009345 μM	SANGER
BL-70	Growth Inhibition Assay		IC50 = 0.009303 μM	SANGER
NCI-H1355	Growth Inhibition Assay		IC50 = 0.009138 μM	SANGER
OVCAR-4	Growth Inhibition Assay		IC50 = 0.009041 μM	SANGER
KNS-42	Growth Inhibition Assay		IC50 = 0.008907 μM	SANGER
A388	Growth Inhibition Assay		IC50 = 0.008738 μM	SANGER
CCRF-CEM	Growth Inhibition Assay		IC50 = 0.008708 μM	SANGER
OCI-AML2	Growth Inhibition Assay		IC50 = 0.008521 μM	SANGER
DEL	Growth Inhibition Assay		IC50 = 0.008449 μM	SANGER
RS4-11	Growth Inhibition Assay		IC50 = 0.008357 μM	SANGER
LXF-289	Growth Inhibition Assay		IC50 = 0.008184 μM	SANGER
HT-144	Growth Inhibition Assay		IC50 = 0.008003 μM	SANGER
8-MG-BA	Growth Inhibition Assay		IC50 = 0.007958 μM	SANGER
LOUCY	Growth Inhibition Assay		IC50 = 0.00775 μM	SANGER
HCE-4	Growth Inhibition Assay		IC50 = 0.007671 μM	SANGER
SW982	Growth Inhibition Assay		IC50 = 0.00766 μM	SANGER
TGBC24TKB	Growth Inhibition Assay		IC50 = 0.007523 μM	SANGER
KURAMOCHI	Growth Inhibition Assay		IC50 = 0.007478 μM	SANGER
CESS	Growth Inhibition Assay		IC50 = 0.007374 μM	SANGER
HC-1	Growth Inhibition Assay		IC50 = 0.007213 μM	SANGER
Becker	Growth Inhibition Assay		IC50 = 0.0072 μM	SANGER
LS-411N	Growth Inhibition Assay		IC50 = 0.007166 μM	SANGER
KGN	Growth Inhibition Assay		IC50 = 0.007124 μM	SANGER
EW-16	Growth Inhibition Assay		IC50 = 0.006937 μM	SANGER
NCI-H510A	Growth Inhibition Assay		IC50 = 0.006652 μM	SANGER
SW962	Growth Inhibition Assay		IC50 = 0.006623 μM	SANGER
OCUB-M	Growth Inhibition Assay		IC50 = 0.006617 μM	SANGER
NOS-1	Growth Inhibition Assay		IC50 = 0.006496 μM	SANGER
KM12	Growth Inhibition Assay		IC50 = 0.006373 μM	SANGER
BE-13	Growth Inhibition Assay		IC50 = 0.006363 μM	SANGER
ALL-PO	Growth Inhibition Assay		IC50 = 0.006298 μM	SANGER
A4-Fuk	Growth Inhibition Assay		IC50 = 0.006109 μM	SANGER
ATN-1	Growth Inhibition Assay		IC50 = 0.00609 μM	SANGER
TE-1	Growth Inhibition Assay		IC50 = 0.006059 μM	SANGER
KS-1	Growth Inhibition Assay		IC50 = 0.005816 μM	SANGER
TE-6	Growth Inhibition Assay		IC50 = 0.005703 μM	SANGER
ES8	Growth Inhibition Assay		IC50 = 0.00538 μM	SANGER
DJM-1	Growth Inhibition Assay		IC50 = 0.005301 μM	SANGER
NB13	Growth Inhibition Assay		IC50 = 0.004912 μM	SANGER
SK-UT-1	Growth Inhibition Assay		IC50 = 0.004803 μM	SANGER
MV-4-11	Growth Inhibition Assay		IC50 = 0.004747 μM	SANGER
NCI-H1648	Growth Inhibition Assay		IC50 = 0.004687 μM	SANGER
IMR-5	Growth Inhibition Assay		IC50 = 0.004496 μM	SANGER
ES4	Growth Inhibition Assay		IC50 = 0.004494 μM	SANGER
GT3TKB	Growth Inhibition Assay		IC50 = 0.004339 μM	SANGER
SK-LMS-1	Growth Inhibition Assay		IC50 = 0.004006 μM	SANGER
EW-1	Growth Inhibition Assay		IC50 = 0.003714 μM	SANGER
no-10	Growth Inhibition Assay		IC50 = 0.003618 μM	SANGER
SIG-M5	Growth Inhibition Assay		IC50 = 0.003272 μM	SANGER
TE-9	Growth Inhibition Assay		IC50 = 0.003255 μM	SANGER
ACN	Growth Inhibition Assay		IC50 = 0.003157 μM	SANGER
BB30-HNC	Growth Inhibition Assay		IC50 = 0.003138 μM	SANGER
KALS-1	Growth Inhibition Assay		IC50 = 0.00308 μM	SANGER
VA-ES-BJ	Growth Inhibition Assay		IC50 = 0.002996 μM	SANGER
MRK-nu-1	Growth Inhibition Assay		IC50 = 0.00299 μM	SANGER
RKO	Growth Inhibition Assay		IC50 = 0.002977 μM	SANGER
MC116	Growth Inhibition Assay		IC50 = 0.002888 μM	SANGER
IA-LM	Growth Inhibition Assay		IC50 = 0.002802 μM	SANGER
MFH-ino	Growth Inhibition Assay		IC50 = 0.00268 μM	SANGER
NTERA-S-cl-D1	Growth Inhibition Assay		IC50 = 0.002088 μM	SANGER
HUTU-80	Growth Inhibition Assay		IC50 = 0.001682 μM	SANGER
TE-10	Growth Inhibition Assay		IC50 = 0.001543 μM	SANGER
ETK-1	Growth Inhibition Assay		IC50 = 0.001521 μM	SANGER
697	Growth Inhibition Assay		IC50 = 0.001495 μM	SANGER
MOLT-4	Growth Inhibition Assay		IC50 = 0.001493 μM	SANGER
PSN1	Growth Inhibition Assay		IC50 = 0.001301 μM	SANGER
TE-11	Growth Inhibition Assay		IC50 = 0.001231 μM	SANGER
SW954	Growth Inhibition Assay		IC50 = 0.001187 μM	SANGER
TE-8	Growth Inhibition Assay		IC50 = 0.001174 μM	SANGER
MZ1-PC	Growth Inhibition Assay		IC50 = 0.0007294 μM	SANGER
RL95-2	Growth Inhibition Assay		IC50 = 0.0006681 μM	SANGER
LC-2-ad	Growth Inhibition Assay		IC50 = 0.0003167 μM	SANGER
TE-15	Growth Inhibition Assay		IC50 = 0.0002869 μM	SANGER
A253	Growth Inhibition Assay		IC50 = 0.01738 μM	SANGER
TGBC1TKB	Growth Inhibition Assay		IC50 = 0.01752 μM	SANGER
SJSA-1	Growth Inhibition Assay		IC50 = 0.01767 μM	SANGER
NCCIT	Growth Inhibition Assay		IC50 = 0.01769 μM	SANGER
NCI-H69	Growth Inhibition Assay		IC50 = 0.01778 μM	SANGER
SH-4	Growth Inhibition Assay		IC50 = 0.01895 μM	SANGER
HCC1187	Growth Inhibition Assay		IC50 = 0.01924 μM	SANGER
HCC1599	Growth Inhibition Assay		IC50 = 0.0202 μM	SANGER
ONS-76	Growth Inhibition Assay		IC50 = 0.02036 μM	SANGER
KU812	Growth Inhibition Assay		IC50 = 0.02039 μM	SANGER
ML-2	Growth Inhibition Assay		IC50 = 0.02047 μM	SANGER
HCE-T	Growth Inhibition Assay		IC50 = 0.02092 μM	SANGER
NCI-H446	Growth Inhibition Assay		IC50 = 0.02112 μM	SANGER
RPMI-6666	Growth Inhibition Assay		IC50 = 0.02149 μM	SANGER
MOLT-16	Growth Inhibition Assay		IC50 = 0.02153 μM	SANGER
JiyoyeP-2003	Growth Inhibition Assay		IC50 = 0.02176 μM	SANGER
MHH-PREB-1	Growth Inhibition Assay		IC50 = 0.02191 μM	SANGER
MC-CAR	Growth Inhibition Assay		IC50 = 0.02326 μM	SANGER
BC-3	Growth Inhibition Assay		IC50 = 0.02344 μM	SANGER
KINGS-1	Growth Inhibition Assay		IC50 = 0.02355 μM	SANGER
PF-382	Growth Inhibition Assay		IC50 = 0.02378 μM	SANGER
J-RT3-T3-5	Growth Inhibition Assay		IC50 = 0.02383 μM	SANGER
SF539	Growth Inhibition Assay		IC50 = 0.02401 μM	SANGER
LB831-BLC	Growth Inhibition Assay		IC50 = 0.02485 μM	SANGER
DMS-114	Growth Inhibition Assay		IC50 = 0.02502 μM	SANGER
LB1047-RCC	Growth Inhibition Assay		IC50 = 0.0251 μM	SANGER
BB65-RCC	Growth Inhibition Assay		IC50 = 0.02534 μM	SANGER
LB771-HNC	Growth Inhibition Assay		IC50 = 0.02534 μM	SANGER
BV-173	Growth Inhibition Assay		IC50 = 0.02554 μM	SANGER
ARH-77	Growth Inhibition Assay		IC50 = 0.02601 μM	SANGER
IST-MEL1	Growth Inhibition Assay		IC50 = 0.02623 μM	SANGER
NB1	Growth Inhibition Assay		IC50 = 0.02687 μM	SANGER
EoL-1-cell	Growth Inhibition Assay		IC50 = 0.02688 μM	SANGER
KY821	Growth Inhibition Assay		IC50 = 0.02697 μM	SANGER
CMK	Growth Inhibition Assay		IC50 = 0.02734 μM	SANGER
NCI-H2126	Growth Inhibition Assay		IC50 = 0.02768 μM	SANGER
NCI-H526	Growth Inhibition Assay		IC50 = 0.02891 μM	SANGER
COLO-684	Growth Inhibition Assay		IC50 = 0.02908 μM	SANGER
NCI-H747	Growth Inhibition Assay		IC50 = 0.02933 μM	SANGER
JAR	Growth Inhibition Assay		IC50 = 0.02946 μM	SANGER
MEG-01	Growth Inhibition Assay		IC50 = 0.02978 μM	SANGER
MONO-MAC-6	Growth Inhibition Assay		IC50 = 0.03023 μM	SANGER
IST-SL1	Growth Inhibition Assay		IC50 = 0.03042 μM	SANGER
CPC-N	Growth Inhibition Assay		IC50 = 0.03079 μM	SANGER
NCI-H1963	Growth Inhibition Assay		IC50 = 0.03131 μM	SANGER
K052	Growth Inhibition Assay		IC50 = 0.03247 μM	SANGER
KM-H2	Growth Inhibition Assay		IC50 = 0.03307 μM	SANGER
TE-12	Growth Inhibition Assay		IC50 = 0.03309 μM	SANGER
TK10	Growth Inhibition Assay		IC50 = 0.03356 μM	SANGER
NMC-G1	Growth Inhibition Assay		IC50 = 0.03452 μM	SANGER
no-11	Growth Inhibition Assay		IC50 = 0.03478 μM	SANGER
NCI-H524	Growth Inhibition Assay		IC50 = 0.03529 μM	SANGER
MHH-CALL-2	Growth Inhibition Assay		IC50 = 0.03562 μM	SANGER
GB-1	Growth Inhibition Assay		IC50 = 0.036 μM	SANGER
OPM-2	Growth Inhibition Assay		IC50 = 0.03673 μM	SANGER
RH-1	Growth Inhibition Assay		IC50 = 0.03819 μM	SANGER
NCI-H64	Growth Inhibition Assay		IC50 = 0.03857 μM	SANGER
EVSA-T	Growth Inhibition Assay		IC50 = 0.03923 μM	SANGER
KARPAS-299	Growth Inhibition Assay		IC50 = 0.0398 μM	SANGER
MZ7-mel	Growth Inhibition Assay		IC50 = 0.0404 μM	SANGER
LB373-MEL-D	Growth Inhibition Assay		IC50 = 0.04105 μM	SANGER
HEL	Growth Inhibition Assay		IC50 = 0.0414 μM	SANGER
SW872	Growth Inhibition Assay		IC50 = 0.0421 μM	SANGER
DU-4475	Growth Inhibition Assay		IC50 = 0.04244 μM	SANGER
IST-SL2	Growth Inhibition Assay		IC50 = 0.04275 μM	SANGER
NCI-H82	Growth Inhibition Assay		IC50 = 0.04307 μM	SANGER
LC4-1	Growth Inhibition Assay		IC50 = 0.04351 μM	SANGER
HDLM-2	Growth Inhibition Assay		IC50 = 0.04392 μM	SANGER
MMAC-SF	Growth Inhibition Assay		IC50 = 0.04534 μM	SANGER
L-540	Growth Inhibition Assay		IC50 = 0.04639 μM	SANGER
MZ2-MEL	Growth Inhibition Assay		IC50 = 0.04742 μM	SANGER
LU-134-A	Growth Inhibition Assay		IC50 = 0.04773 μM	SANGER
UACC-257	Growth Inhibition Assay		IC50 = 0.04849 μM	SANGER
NCI-H1581	Growth Inhibition Assay		IC50 = 0.04953 μM	SANGER
NB17	Growth Inhibition Assay		IC50 = 0.04979 μM	SANGER
SBC-1	Growth Inhibition Assay		IC50 = 0.05042 μM	SANGER
TALL-1	Growth Inhibition Assay		IC50 = 0.05045 μM	SANGER
NCI-H1304	Growth Inhibition Assay		IC50 = 0.05208 μM	SANGER
NEC8	Growth Inhibition Assay		IC50 = 0.05286 μM	SANGER
CAL-148	Growth Inhibition Assay		IC50 = 0.05439 μM	SANGER
CGTH-W-1	Growth Inhibition Assay		IC50 = 0.05449 μM	SANGER
NCI-H889	Growth Inhibition Assay		IC50 = 0.05592 μM	SANGER
GR-ST	Growth Inhibition Assay		IC50 = 0.05621 μM	SANGER
KARPAS-422	Growth Inhibition Assay		IC50 = 0.0565 μM	SANGER
RPMI-8866	Growth Inhibition Assay		IC50 = 0.05712 μM	SANGER
SCLC-21H	Growth Inhibition Assay		IC50 = 0.05884 μM	SANGER
COR-L88	Growth Inhibition Assay		IC50 = 0.05927 μM	SANGER
LU-139	Growth Inhibition Assay		IC50 = 0.05986 μM	SANGER
SF126	Growth Inhibition Assay		IC50 = 0.06133 μM	SANGER
NCI-H1882	Growth Inhibition Assay		IC50 = 0.06424 μM	SANGER
EW-24	Growth Inhibition Assay		IC50 = 0.06483 μM	SANGER
CP67-MEL	Growth Inhibition Assay		IC50 = 0.0681 μM	SANGER
DG-75	Growth Inhibition Assay		IC50 = 0.06899 μM	SANGER
LOXIMVI	Growth Inhibition Assay		IC50 = 0.07028 μM	SANGER
HH	Growth Inhibition Assay		IC50 = 0.07157 μM	SANGER
K5	Growth Inhibition Assay		IC50 = 0.07226 μM	SANGER
EC-GI-10	Growth Inhibition Assay		IC50 = 0.07257 μM	SANGER
SK-N-DZ	Growth Inhibition Assay		IC50 = 0.07307 μM	SANGER
A3-KAW	Growth Inhibition Assay		IC50 = 0.07351 μM	SANGER
MLMA	Growth Inhibition Assay		IC50 = 0.07465 μM	SANGER
LB996-RCC	Growth Inhibition Assay		IC50 = 0.07707 μM	SANGER
OS-RC-2	Growth Inhibition Assay		IC50 = 0.07748 μM	SANGER
CTB-1	Growth Inhibition Assay		IC50 = 0.0781 μM	SANGER
IST-MES1	Growth Inhibition Assay		IC50 = 0.07912 μM	SANGER
LS-1034	Growth Inhibition Assay		IC50 = 0.08035 μM	SANGER
HT	Growth Inhibition Assay		IC50 = 0.08086 μM	SANGER
NCI-H2141	Growth Inhibition Assay		IC50 = 0.081 μM	SANGER
LB2518-MEL	Growth Inhibition Assay		IC50 = 0.08141 μM	SANGER
GI-ME-N	Growth Inhibition Assay		IC50 = 0.08452 μM	SANGER
TGW	Growth Inhibition Assay		IC50 = 0.08607 μM	SANGER
SK-NEP-1	Growth Inhibition Assay		IC50 = 0.08641 μM	SANGER
NOMO-1	Growth Inhibition Assay		IC50 = 0.09275 μM	SANGER
ES6	Growth Inhibition Assay		IC50 = 0.09589 μM	SANGER
NCI-H209	Growth Inhibition Assay		IC50 = 0.09786 μM	SANGER
GAK	Growth Inhibition Assay		IC50 = 0.1016 μM	SANGER
BC-1	Growth Inhibition Assay		IC50 = 0.10361 μM	SANGER
KLE	Growth Inhibition Assay		IC50 = 0.10443 μM	SANGER
EW-3	Growth Inhibition Assay		IC50 = 0.1098 μM	SANGER
NKM-1	Growth Inhibition Assay		IC50 = 0.111 μM	SANGER
D-336MG	Growth Inhibition Assay		IC50 = 0.11244 μM	SANGER
NB69	Growth Inhibition Assay		IC50 = 0.11301 μM	SANGER
D-263MG	Growth Inhibition Assay		IC50 = 0.11712 μM	SANGER
KP-N-YS	Growth Inhibition Assay		IC50 = 0.12291 μM	SANGER
NCI-H1155	Growth Inhibition Assay		IC50 = 0.12558 μM	SANGER
BOKU	Growth Inhibition Assay		IC50 = 0.12579 μM	SANGER
LAMA-84	Growth Inhibition Assay		IC50 = 0.1299 μM	SANGER
Raji	Growth Inhibition Assay		IC50 = 0.13117 μM	SANGER
LU-65	Growth Inhibition Assay		IC50 = 0.13307 μM	SANGER
NCI-H187	Growth Inhibition Assay		IC50 = 0.13924 μM	SANGER
GCIY	Growth Inhibition Assay		IC50 = 0.14901 μM	SANGER
NCI-H2107	Growth Inhibition Assay		IC50 = 0.1508 μM	SANGER
NCI-H1522	Growth Inhibition Assay		IC50 = 0.15266 μM	SANGER
NB6	Growth Inhibition Assay		IC50 = 0.15623 μM	SANGER
EM-2	Growth Inhibition Assay		IC50 = 0.15706 μM	SANGER
HCC2218	Growth Inhibition Assay		IC50 = 0.1598 μM	SANGER
NCI-H748	Growth Inhibition Assay		IC50 = 0.16376 μM	SANGER
MS-1	Growth Inhibition Assay		IC50 = 0.16537 μM	SANGER
NB5	Growth Inhibition Assay		IC50 = 0.16597 μM	SANGER
OMC-1	Growth Inhibition Assay		IC50 = 0.16688 μM	SANGER
NCI-H345	Growth Inhibition Assay		IC50 = 0.16928 μM	SANGER
L-428	Growth Inhibition Assay		IC50 = 0.16945 μM	SANGER
SCH	Growth Inhibition Assay		IC50 = 0.18685 μM	SANGER
NCI-H1417	Growth Inhibition Assay		IC50 = 0.19227 μM	SANGER
COLO-320-HSR	Growth Inhibition Assay		IC50 = 0.19532 μM	SANGER
BT-474	Growth Inhibition Assay		IC50 = 0.20892 μM	SANGER
GDM-1	Growth Inhibition Assay		IC50 = 0.21971 μM	SANGER
NCI-H2196	Growth Inhibition Assay		IC50 = 0.22235 μM	SANGER
KP-N-RT-BM-1	Growth Inhibition Assay		IC50 = 0.22349 μM	SANGER
KNS-81-FD	Growth Inhibition Assay		IC50 = 0.22958 μM	SANGER
COLO-668	Growth Inhibition Assay		IC50 = 0.23675 μM	SANGER
C2BBe1	Growth Inhibition Assay		IC50 = 0.26747 μM	SANGER
Ramos-2G6-4C10	Growth Inhibition Assay		IC50 = 0.26954 μM	SANGER
CAS-1	Growth Inhibition Assay		IC50 = 0.27096 μM	SANGER
GOTO	Growth Inhibition Assay		IC50 = 0.27894 μM	SANGER
LP-1	Growth Inhibition Assay		IC50 = 0.28057 μM	SANGER
NCI-SNU-1	Growth Inhibition Assay		IC50 = 0.29422 μM	SANGER
EB-3	Growth Inhibition Assay		IC50 = 0.29979 μM	SANGER
MHH-NB-11	Growth Inhibition Assay		IC50 = 0.30402 μM	SANGER
SK-N-FI	Growth Inhibition Assay		IC50 = 0.31692 μM	SANGER
HCC2157	Growth Inhibition Assay		IC50 = 0.33913 μM	SANGER
SIMA	Growth Inhibition Assay		IC50 = 0.34581 μM	SANGER
MDA-MB-134-VI	Growth Inhibition Assay		IC50 = 0.36928 μM	SANGER
NCI-H1694	Growth Inhibition Assay		IC50 = 0.37 μM	SANGER
EHEB	Growth Inhibition Assay		IC50 = 0.39085 μM	SANGER
U-266	Growth Inhibition Assay		IC50 = 0.39846 μM	SANGER
LC-1F	Growth Inhibition Assay		IC50 = 0.43765 μM	SANGER
SHP-77	Growth Inhibition Assay		IC50 = 0.47855 μM	SANGER
LS-513	Growth Inhibition Assay		IC50 = 0.49307 μM	SANGER
TE-441-T	Growth Inhibition Assay		IC50 = 0.52479 μM	SANGER
D-247MG	Growth Inhibition Assay		IC50 = 0.59924 μM	SANGER
SNU-C1	Growth Inhibition Assay		IC50 = 0.61887 μM	SANGER
SU-DHL-1	Growth Inhibition Assay		IC50 = 0.6289 μM	SANGER
DB	Growth Inhibition Assay		IC50 = 0.82872 μM	SANGER
CP66-MEL	Growth Inhibition Assay		IC50 = 0.95198 μM	SANGER
NCI-H1650	Growth Inhibition Assay		IC50 = 1.04651 μM	SANGER
DMS-153	Growth Inhibition Assay		IC50 = 1.10124 μM	SANGER
A498	Growth Inhibition Assay		IC50 = 1.21534 μM	SANGER
U-698-M	Growth Inhibition Assay		IC50 = 1.22557 μM	SANGER
NCI-H1092	Growth Inhibition Assay		IC50 = 1.30719 μM	SANGER
NCI-H23	Growth Inhibition Assay		IC50 = 1.3319 μM	SANGER
JVM-2	Growth Inhibition Assay		IC50 = 1.42177 μM	SANGER
MSTO-211H	Growth Inhibition Assay		IC50 = 1.43905 μM	SANGER
A704	Growth Inhibition Assay		IC50 = 1.51191 μM	SANGER
ECC4	Growth Inhibition Assay		IC50 = 1.54949 μM	SANGER
NCI-H226	Growth Inhibition Assay		IC50 = 1.71489 μM	SANGER
CA46	Growth Inhibition Assay		IC50 = 1.73216 μM	SANGER
NCI-H719	Growth Inhibition Assay		IC50 = 1.73651 μM	SANGER
KMS-12-PE	Growth Inhibition Assay		IC50 = 1.90481 μM	SANGER
MPP-89	Growth Inhibition Assay		IC50 = 1.94182 μM	SANGER
NCI-H2171	Growth Inhibition Assay		IC50 = 2.20593 μM	SANGER
CHP-126	Growth Inhibition Assay		IC50 = 2.24737 μM	SANGER
DMS-79	Growth Inhibition Assay		IC50 = 2.27644 μM	SANGER
SCC-15	Growth Inhibition Assay		IC50 = 2.30678 μM	SANGER
REH	Growth Inhibition Assay		IC50 = 2.31165 μM	SANGER
NCI-H2081	Growth Inhibition Assay		IC50 = 2.32315 μM	SANGER
NCI-H720	Growth Inhibition Assay		IC50 = 2.55972 μM	SANGER
KMOE-2	Growth Inhibition Assay		IC50 = 2.75712 μM	SANGER
D-502MG	Growth Inhibition Assay		IC50 = 2.86805 μM	SANGER
MN-60	Growth Inhibition Assay		IC50 = 2.95245 μM	SANGER
LU-165	Growth Inhibition Assay		IC50 = 3.01956 μM	SANGER
DSH1	Growth Inhibition Assay		IC50 = 3.23442 μM	SANGER
SK-MM-2	Growth Inhibition Assay		IC50 = 3.54385 μM	SANGER
LAN-6	Growth Inhibition Assay		IC50 = 3.54788 μM	SANGER
NCI-H1838	Growth Inhibition Assay		IC50 = 4.18573 μM	SANGER
U-87-MG	Growth Inhibition Assay		IC50 = 4.18673 μM	SANGER
NB7	Growth Inhibition Assay		IC50 = 4.40376 μM	SANGER
BB49-HNC	Growth Inhibition Assay		IC50 = 4.94617 μM	SANGER
NCI-H1395	Growth Inhibition Assay		IC50 = 5.00345 μM	SANGER
RCC10RGB	Growth Inhibition Assay		IC50 = 5.06271 μM	SANGER
COLO-824	Growth Inhibition Assay		IC50 = 5.08313 μM	SANGER
NCI-H322M	Growth Inhibition Assay		IC50 = 5.186 μM	SANGER
SW684	Growth Inhibition Assay		IC50 = 5.23288 μM	SANGER
P30-OHK	Growth Inhibition Assay		IC50 = 5.35052 μM	SANGER
COLO-829	Growth Inhibition Assay		IC50 = 5.49884 μM	SANGER
HAL-01	Growth Inhibition Assay		IC50 = 5.73185 μM	SANGER
LNCaP-Clone-FGC	Growth Inhibition Assay		IC50 = 6.34489 μM	SANGER
SK-MEL-1	Growth Inhibition Assay		IC50 = 6.70896 μM	SANGER
THP-1	Growth Inhibition Assay		IC50 = 6.72583 μM	SANGER
EW-18	Growth Inhibition Assay		IC50 = 7.03675 μM	SANGER
EKVX	Growth Inhibition Assay		IC50 = 7.16865 μM	SANGER
NB14	Growth Inhibition Assay		IC50 = 7.8139 μM	SANGER
ES5	Growth Inhibition Assay		IC50 = 7.86662 μM	SANGER
SK-MEL-2	Growth Inhibition Assay		IC50 = 8.45976 μM	SANGER
COLO-800	Growth Inhibition Assay		IC50 = 8.4787 μM	SANGER
EB2	Growth Inhibition Assay		IC50 = 9.19835 μM	SANGER
ES3	Growth Inhibition Assay		IC50 = 9.30665 μM	SANGER
SKM-1	Growth Inhibition Assay		IC50 = 9.39459 μM	SANGER
MFM-223	Growth Inhibition Assay		IC50 = 9.50127 μM	SANGER
LB2241-RCC	Growth Inhibition Assay		IC50 = 10.0386 μM	SANGER
EW-13	Growth Inhibition Assay		IC50 = 10.3333 μM	SANGER
D-283MED	Growth Inhibition Assay		IC50 = 10.4959 μM	SANGER
EW-11	Growth Inhibition Assay		IC50 = 11.6694 μM	SANGER
NCI-H128	Growth Inhibition Assay		IC50 = 12.1334 μM	SANGER
ES7	Growth Inhibition Assay		IC50 = 15.2494 μM	SANGER
AM-38	Growth Inhibition Assay		IC50 = 15.4166 μM	SANGER
NCI-H716	Growth Inhibition Assay		IC50 = 17.9299 μM	SANGER
NCI-H1770	Growth Inhibition Assay		IC50 = 18.3851 μM	SANGER
JVM-3	Growth Inhibition Assay		IC50 = 20.8985 μM	SANGER
CW-2	Growth Inhibition Assay		IC50 = 21.1349 μM	SANGER
YT	Growth Inhibition Assay		IC50 = 21.4691 μM	SANGER
C8166	Growth Inhibition Assay		IC50 = 22.2746 μM	SANGER
SUP-T1	Growth Inhibition Assay		IC50 = 23.2512 μM	SANGER
KASUMI-1	Growth Inhibition Assay		IC50 = 23.5119 μM	SANGER
IM-9	Growth Inhibition Assay		IC50 = 23.6979 μM	SANGER
NH-12	Growth Inhibition Assay		IC50 = 24.1654 μM	SANGER
WSU-NHL	Growth Inhibition Assay		IC50 = 25.7261 μM	SANGER
TUR	Growth Inhibition Assay		IC50 = 26.6533 μM	SANGER
RL	Growth Inhibition Assay		IC50 = 27.2242 μM	SANGER
EW-12	Growth Inhibition Assay		IC50 = 28.0702 μM	SANGER
KG-1	Growth Inhibition Assay		IC50 = 28.2865 μM	SANGER
P31-FUJ	Growth Inhibition Assay		IC50 = 29.0489 μM	SANGER
NB10	Growth Inhibition Assay		IC50 = 31.509 μM	SANGER
COLO205	Cytotoxicity assay		GI50 = 0.00176 μM	7908950
SF539	Cytotoxicity assay		GI50 = 0.00366 μM	7908950
SNB75	Cytotoxicity assay		GI50 = 0.00808 μM	7908950
DMS114	Cytotoxicity assay		GI50 = 0.0123 μM	7908950
OVCAR-3	Cytotoxicity assay		GI50 = 0.0197 μM	7908950
NCI-H460	Cytotoxicity assay		GI50 = 0.0219 μM	7908950
HOP62	Cytotoxicity assay		GI50 = 0.0671 μM	7908950
mammary carcinoma	Cytotoxicity assay		IC50 = 0.299 μM	8182698
NCI60	Cytotoxicity assay		GI50 = 0.00065 μM	9461653
MCF-7	Growth inhibition assay		GI50 = 0.0011 μM	9873597
murine leukemic P388	Growth inhibition assay		GI50 = 0.016 μM	9873597
KB	Cytotoxicity assay		IC50 = 0.006 μM	10978200
MCF-7	Cytotoxicity assay		ED50 = 0.004 μM	11334567
uterine sarcoma (MES-SA)	Cytotoxicity assay		IC50 = 0.00004 μM	11728191
nonsmall cell lung carcinoma (NCI-H460)	Cytotoxicity assay		IC50 = 0.00014 μM	11728191
colon adenocarcinoma (HT-29)	Cytotoxicity assay		IC50 = 0.00016 μM	11728191
prostate carcinoma (DU-145)	Cytotoxicity assay		IC50 = 0.00489 μM	11728191
L2987	Cytotoxicity assay		IC50 = 0.2 μM	12443783
colon adenocarcinoma RKO	Cytotoxicity assay		IC50 = 0.01 μM	12852768
KB	Cytotoxicity assay		ED50 = 0.0004 μM	15043407
Lu1	Cytotoxicity assay		ED50 = 0.002 μM	15043407
LNCAP	Cytotoxicity assay		ED50 = 0.005 μM	15043407
RPE1	Cytotoxicity assay		ED50 = 0.023 μM	15043407
Col2	Cytotoxicity assay		ED50 = 0.046 μM	15043407
A431	Cell cycle arrest assay		EC50 = 0.009 μM	16377187
Aro	Cytotoxicity assay		IC50 = 0.0002 μM	16539377
PT45	Cytotoxicity assay		IC50 = 0.005 μM	16539377
A549	Cytotoxicity assay		IC50 = 0.006 μM	16539377
MCF7	Cytotoxicity assay		IC50 = 0.007 μM	16539377
HeLa	Cytotoxicity assay		IC50 = 0.008 μM	16539377
Ovcar3	Cytotoxicity assay		IC50 = 0.01 μM	16539377
HT29	Cytotoxicity assay		IC50 = 0.05 μM	16539377
H295R	Cytotoxicity assay		IC50 = 0.08 μM	16539377
BNL	Cytotoxicity assay		IC50 = 0.2 μM	16539377
4T1	Cytotoxicity assay		IC50 = 0.2 μM	16539377
HepG2	Cytotoxicity assay		IC50 = 0.3 μM	16539377
VA13	Cytotoxicity assay		IC50 = 0.0059 μM	16724842
WI38	Cytotoxicity assay		IC50 = 0.0468 μM	16724842
HepG2	Cytotoxicity assay		IC50 = 9.49 μM	16724842
HT29	Cytotoxicity assay		EC50 = 0.006 μM	16870428
K562	Cytotoxicity assay		EC50 = 0.014 μM	16870428
MCF7	Cytotoxicity assay		EC50 = 0.036 μM	16870428
VA-13	Cytotoxicity assay		IC50 = 0.005 μM	16933868
WI38	Cytotoxicity assay		IC50 = 0.04 μM	16933868
VA13	Cytotoxicity assay		IC50 = 0.005 μM	17067155
WI38	Cytotoxicity assay		IC50 = 0.04 μM	17067155
Hep G2	Cytotoxicity assay		IC50 = 8.1 μM	17067155
TW01	Cytotoxicity assay		IC50 = 0.0003 μM	17113288
MCF7	Cytotoxicity assay		IC50 = 0.0005 μM	17113288
MKN45	Cytotoxicity assay		IC50 = 0.0005 μM	17113288
MES-SA	Cytotoxicity assay		IC50 = 0.0005 μM	17113288
HCT116	Cytotoxicity assay		IC50 = 0.0006 μM	17113288
RPTEC	Cytotoxicity assay		IC50 = 0.0009 μM	17113288
Hep3B	Cytotoxicity assay		IC50 = 0.0054 μM	17113288
NCI-H226	Cytotoxicity assay		IC50 = 0.0068 μM	17113288
A498	Cytotoxicity assay		IC50 = 0.061 μM	17113288
MDA435/LCC6	Antiproliferative activity assay		IC50 = 0.0029 μM	17154505
multidrug resistant MDA435/LCC6	Antiproliferative activity assay		IC50 = 0.0048 μM	17154505
P388	Antiproliferative activity assay		IC50 = 0.022 μM	17154505
adriamycin resistant P388	Antiproliferative activity assay		IC50 = 0.03 μM	17154505
A2780	Cytotoxicity assay		IC50 = 0.001 μM	17206139
A2780-1A9	Cytotoxicity assay		IC50 = 0.0011 μM	17206139
A549	Cytotoxicity assay		IC50 = 0.0036 μM	17206139
1A9PTX22	Cytotoxicity assay		IC50 = 0.019 μM	17206139
1A9PTX10	Cytotoxicity assay		IC50 = 0.03 μM	17206139
A2780AD	Cytotoxicity assay		IC50 = 0.9 μM	17206139
KB	Antiproliferative activity assay		IC50 = 0.00245 μM	17228873
COLO205	Cytotoxicity assay		IC50 = 0.0033 μM	17228873
KB8.5	Antiproliferative activity assay		IC50 = 0.026 μM	17228873
KBV1	Antiproliferative activity assay		IC50 = 2.013 μM	17228873
A2780	Cytotoxicity assay		IC50 = 0.0007 μM	17239597
2780AD	Cytotoxicity assay		IC50 = 0.535 μM	17239597
1A9	Cytotoxicity assay		ED50 = 0.001 μM	17350834
MCF7	Cytotoxicity assay		ED50 = 0.0011 μM	17350834
DU145	Cytotoxicity assay		ED50 = 0.0013 μM	17350834
KB	Cytotoxicity assay		ED50 = 0.0018 μM	17350834
A549	Cytotoxicity assay		ED50 = 0.0023 μM	17350834
LNCAP	Cytotoxicity assay		ED50 = 0.0026 μM	17350834
PC3	Cytotoxicity assay		ED50 = 0.0555 μM	17350834
KBVIN	Cytotoxicity assay		ED50 = 0.311 μM	17350834
A2780	Cytotoxicity assay		IC50 = 0.0016 μM	17395465
A2780/AD	Cytotoxicity assay		IC50 = 0.92 μM	17395465
KB	Antiproliferative activity assay		IC50 = 0.00245 μM	17416524
COLO205	Cytotoxicity assay		IC50 = 0.0033 μM	17416524
KB8.5	Antiproliferative activity assay		IC50 = 0.026 μM	17416524
KBV1	Antiproliferative activity assay		IC50 = 2.013 μM	17416524
neural precursor	Antiproliferative activity assay		EC50 = 0.01 μM	17417631
OVCAR-3	Cytotoxicity assay		IC50 = 0.0002 μM	17419065
MDA-MB-231	Cytotoxicity assay		IC50 = 0.0045 μM	17419065
MCF7	Cytotoxicity assay		IC50 = 0.0049 μM	17419065
A2780	Cytotoxicity assay		IC50 = 0.025 μM	17419065
PC3	Cytotoxicity assay		IC50 = 0.077 μM	17419065
LoVo	Cytotoxicity assay		IC50 = 0.09 μM	17419065
L2987	Cytotoxicity assay		IC50 = 0.2 μM	17419065
cells	Cytotoxicity assay		IC50 = 0.0059 μM	17442577
cells	Cytotoxicity assay		IC50 = 0.01 μM	17485207
A2780	Growth inhibition assay		IC50 = 0.0028 μM	17490878
VA13	Growth inhibition assay		IC50 = 0.005 μM	17490878
WI38	Growth inhibition assay		IC50 = 0.04 μM	17490878
2780AD	Growth inhibition assay		IC50 = 0.183 μM	17490878
HepG2	Growth inhibition assay		IC50 = 8.1 μM	17490878
cells expressing MRP1	Growth inhibition assay		IC50 = 0.0025 μM	17567121
cells expressing Pgp/MRP1	Growth inhibition assay		IC50 = 2.7 μM	17567121
VA13	Growth inhibition assay		IC50 = 5 μM	17595134
MCF7	Function assay		IC50 = 0.0018 μM	17601739
adriamycin-resistant MCF7	Function assay		IC50 = 8.2 μM	17601739
RPMI8226	Cytotoxicity assay		GI50 = 0.002 μM	17696332
HT29	Cytotoxicity assay		GI50 = 0.002 μM	17696332
COLO205	Cytotoxicity assay		GI50 = 0.003 μM	17696332
HCC2998	Cytotoxicity assay		GI50 = 0.003 μM	17696332
HS578T	Cytotoxicity assay		GI50 = 0.003 μM	17696332
PC3	Cytotoxicity assay		GI50 = 0.004 μM	17696332
SNB75	Cytotoxicity assay		GI50 = 0.004 μM	17696332
A549	Cytotoxicity assay		GI50 = 0.004 μM	17696332
KM12	Cytotoxicity assay		GI50 = 0.004 μM	17696332
DU145	Cytotoxicity assay		GI50 = 0.005 μM	17696332
SK-OV3	Cytotoxicity assay		GI50 = 0.008 μM	17696332
NCI-H322M	Cytotoxicity assay		GI50 = 0.013 μM	17696332
UACC257	Cytotoxicity assay		GI50 = 0.04 μM	17696332
HCT15	Cytotoxicity assay		GI50 = 0.158 μM	17696332
ACHN	Cytotoxicity assay		GI50 = 0.398 μM	17696332
HeLa	Cytotoxicity assay		IC50 = 0.0056 μM	17764148
MCF7	Cytotoxicity assay		IC50 = 0.0124 μM	17764148
A549	Cytotoxicity assay		IC50 = 0.0126 μM	17764148
HGC27	Cytotoxicity assay		IC50 = 0.7778 μM	17764148
HeLa	Cytotoxicity assay		IC50 = 0.02 μM	17911017
HepG2	Cytotoxicity assay		IC50 = 0.82 μM	17911017
BGC823	Cytotoxicity assay		IC50 = 1.15 μM	17911017
cells assessed as accumulation at G2/M phase after 24 hrs by flow cytometric analysis	Cell cycle arrest assay		EC50 = 0.049 μM	17973361
cells after 48 hrs by XTT assay	Antiproliferative activity assay		IC50 = 0.4 μM	17973361
A2780	Cytotoxicity assay		IC50 = 0.0063 μM	18001087
BGC823	Cytotoxicity assay		IC50 = 0.007 μM	18001087
A549	Cytotoxicity assay		IC50 = 0.019 μM	18001087
HCT8	Cytotoxicity assay		IC50 = 0.037 μM	18001087
Bel7402	Cytotoxicity assay		IC50 = 0.1 μM	18001087
cells by alamar blue assay	Function assay		IC50 = 0.04 μM	18070965
HT29	Antiproliferative activity assay		GI50 = 0.015 μM	18502639
M21	Antiproliferative activity assay		GI50 = 0.037 μM	18502639
MCF7	Antiproliferative activity assay		GI50 = 0.054 μM	18502639
HCT116	Cytotoxicity assay		IC50 = 0.0136 μM	18606540
SF268	Cytotoxicity assay		IC50 = 0.0153 μM	18606540
A549	Cytotoxicity assay		IC50 = 0.0231 μM	18606540
MDA-MB-231	Cytotoxicity assay		IC50 = 0.0405 μM	18606540
SF295	Cytotoxicity assay		IC50 = 0.29 μM	18606540
SKOV3	Cytotoxicity assay		IC50 = 2.43 μM	18701281
KB	Cytotoxicity assay		IC50 = 2.54 μM	18701281
Eca109	Cytotoxicity assay		IC50 = 2.73 μM	18701281
PC3	Cytotoxicity assay		IC50 = 2.85 μM	18701281
SMMC7721	Cytotoxicity assay		IC50 = 2.86 μM	18701281
MCF7	Cytotoxicity assay		IC50 = 2.98 μM	18701281
HeLa	Cytotoxicity assay		IC50 = 3.11 μM	18701281
HCT8	Cytotoxicity assay		IC50 = 3.29 μM	18701281
K562	Cytotoxicity assay		IC50 = 3.65 μM	18701281
A549	Cytotoxicity assay		IC50 = 0.002 μM	18715782
MCF7	Cytotoxicity assay		ED50 = 0.0032 μM	18926701
NCI/ADR-RES	Cytotoxicity assay		ED50 = 1.5 μM	18926701
MCF7	Cytotoxicity assay		ED50 = 0.0021 μM	18977659
NCI/ADR-RES	Cytotoxicity assay		ED50 = 2 μM	18977659
cells after 72 hrs by MTT assay	Cytotoxicity assay		IC50 = 5.14 μM	19053781
KB	Growth inhibition assay		ED50 = 0.023 μM	19161316
HepG2	Cytotoxicity assay		GI50 = 0.001 μM	19195901
WI38	Cytotoxicity assay		GI50 = 0.0137 μM	19195901
RKO	Antiproliferative activity assay		IC50 = 0.02 μM	19220018
KB/HeLa	Antiproliferative activity assay		IC50 = 0.03 μM	19220018
SKOV3	Antiproliferative activity assay		IC50 = 0.05 μM	19220018
SF268	Antiproliferative activity assay		IC50 = 0.05 μM	19220018
NCI-H460	Antiproliferative activity assay		IC50 = 0.07 μM	19220018
A2780	Function assay		IC50 = 0.386 μM	19239240
A2780	Cytotoxicity assay		IC50 = 0.014 μM	19282186
A431	Antiproliferative activity assay		GI50 = 0.00001 μM	19394218
MESSA	Antiproliferative activity assay		GI50 = 0.00001 μM	19394218
HCT15	Antiproliferative activity assay		GI50 = 0.011 μM	19394218
MES-SA/Dx5	Antiproliferative activity assay		GI50 = 0.16 μM	19394218
HCT15/CLO2	Antiproliferative activity assay		GI50 = 0.83 μM	19394218
paclitaxel-resistant A2780TC1	Function assay		IC50 = 5.898 μM	19423340
HepG2	Cytotoxicity assay		GI50 = 0.059 μM	19476336
PtK2	Growth inhibition assay		IC50 = 0.021 μM	19601594
rat A10	Growth inhibition assay		IC50 = 0.038 μM	19601594
MES-SA/Dx5	Cytotoxicity assay		IC50 = 7.538 μM	19679475
A549	Cytotoxicity assay		IC50 = 0.0023 μM	19708679
BGC823	Cytotoxicity assay		IC50 = 0.0033 μM	19708679
HCT8	Cytotoxicity assay		IC50 = 0.0036 μM	19708679
A2780	Cytotoxicity assay		IC50 = 0.0079 μM	19708679
Bel7404	Cytotoxicity assay		IC50 = 0.0123 μM	19708679
A2780	Cytotoxicity assay		IC50 = 0.0028 μM	19877653
A2780AD	Cytotoxicity assay		IC50 = 0.415 μM	19877653
KBVIN	Cytotoxicity assay		IC50 = 0.00109 μM	20036537
KB	Cytotoxicity assay		IC50 = 0.00155 μM	20036537
A549	Cytotoxicity assay		IC50 = 0.00193 μM	20036537
DU145	Cytotoxicity assay		IC50 = 0.00235 μM	20036537
KB	Cytotoxicity assay		IC50 = 0.08 μM	20122764
786-0	Cytotoxicity assay		IC50 = 0.08 μM	20122764
A375	Cytotoxicity assay		IC50 = 0.81 μM	20122764
BGC	Cytotoxicity assay		IC50 = 1.5 μM	20122764
769-P	Cytotoxicity assay		IC50 = 7.1 μM	20122764
HT-29	Cytotoxicity assay		IC50 = 0.0014 μM	20553003
HCT116	Cytotoxicity assay		IC50 = 0.00321 μM	20553003
KB	Cytotoxicity assay		IC50 = 0.08 μM	20627721
786-0	Cytotoxicity assay		IC50 = 0.08 μM	20627721
HepG2	Cytotoxicity assay		IC50 = 0.08 μM	20627721
OS-RC2	Cytotoxicity assay		IC50 = 0.08 μM	20627721
22Rv1	Cytotoxicity assay		IC50 = 0.08 μM	20627721
HT-29	Cytotoxicity assay		IC50 = 0.38 μM	20627721
A375	Cytotoxicity assay		IC50 = 0.81 μM	20627721
MCF7	Cytotoxicity assay		IC50 = 1.3 μM	20627721
BCG823	Cytotoxicity assay		IC50 = 1.5 μM	20627721
769-P	Cytotoxicity assay		IC50 = 7.1 μM	20627721
KB	Cytotoxicity assay		IC50 = 0.08 μM	20716468
786-0	Cytotoxicity assay		IC50 = 0.08 μM	20716468
OS-RC2	Cytotoxicity assay		IC50 = 0.08 μM	20716468
22Rv1	Cytotoxicity assay		IC50 = 0.08 μM	20716468
HepG2	Cytotoxicity assay		IC50 = 0.08 μM	20716468
HT-29	Cytotoxicity assay		IC50 = 0.38 μM	20716468
A375	Cytotoxicity assay		IC50 = 0.81 μM	20716468
MCF7	Cytotoxicity assay		IC50 = 1.3 μM	20716468
BGC823	Cytotoxicity assay		IC50 = 1.5 μM	20716468
769-P	Cytotoxicity assay		IC50 = 7.1 μM	20716468
DU145	Cytotoxicity assay		ED50 = 0.003 μM	20738103
KB	Cytotoxicity assay		ED50 = 0.007 μM	20738103
A549	Cytotoxicity assay		ED50 = 0.008 μM	20738103
multidrug-resistant MDA-MB-435/LCCMDR1	Function assay		IC50 = 0.0693 μM	20919720
LNCAP	Cytotoxicity assay		IC50 = 0.0223 μM	20936874
HeLa	Antiproliferative activity assay		IC50 = 0.0016 μM	20973488
SKOV3	Antiproliferative activity assay		IC50 = 0.003 μM	20973488
HT-29	Anticancer assay		ED50 = 0.0001 μM	21067206
MES-SA	Antiproliferative activity assay		IC50 = 0.00296 μM	21324686
MES-SA	Antiproliferative activity assay		IC50 = 0.00296 μM	21324687
SF295	Antiproliferative activity assay		IC50 = 0.02455 μM	21324687
MES-SA	Cytotoxicity assay		IC50 = 0.00296 μM	21324692
KB	Cell cycle arrest assay		EC50 = 0.002 μM	21480626
786-0	Antiproliferative activity assay		IC50 = 0.004 μM	21774499
PC3	Antiproliferative activity assay		IC50 = 0.00043 μM	21775150
DU145	Antiproliferative activity assay		IC50 = 0.0023 μM	21775150
MDA-MB-435	Antiproliferative activity assay		IC50 = 0.016 μM	21775150
KB	Cytotoxicity assay		IC50 = 6.684 μM	21784631
DU145	Cytotoxicity assay		IC50 = 8.626 μM	21784631
A549	Cytotoxicity assay		IC50 = 9.265 μM	21784631
HeLa	Antiproliferative activity assay		IC50 = 0.00138 μM	21786793
SKOV3	Antiproliferative activity assay		IC50 = 0.00295 μM	21786793
HT-29	Cytotoxicity assay		GI50 = 0.002 μM	21839640
RPMI8226	Cytotoxicity assay		GI50 = 0.002 μM	21839640
HCC2998	Cytotoxicity assay		GI50 = 0.003 μM	21839640
Hs578T	Cytotoxicity assay		GI50 = 0.003 μM	21839640
COLO205	Cytotoxicity assay		GI50 = 0.003 μM	21839640
PC3	Cytotoxicity assay		GI50 = 0.004 μM	21839640
A549	Cytotoxicity assay		GI50 = 0.004 μM	21839640
SNB75	Cytotoxicity assay		GI50 = 0.004 μM	21839640
KM12	Cytotoxicity assay		GI50 = 0.004 μM	21839640
DU145	Cytotoxicity assay		GI50 = 0.005 μM	21839640
SKOV3	Cytotoxicity assay		GI50 = 0.008 μM	21839640
NCI-H322M	Cytotoxicity assay		GI50 = 0.013 μM	21839640
UACC257	Cytotoxicity assay		GI50 = 0.04 μM	21839640
HCT15	Cytotoxicity assay		GI50 = 0.158 μM	21839640
ACHN	Cytotoxicity assay		GI50 = 0.398 μM	21839640
KB	Cytotoxicity assay		IC50 = 0.08 μM	21875764
786-0	Cytotoxicity assay		IC50 = 0.08 μM	21875764
OS-RC2	Cytotoxicity assay		IC50 = 0.08 μM	21875764
22Rv1	Cytotoxicity assay		IC50 = 0.08 μM	21875764
HepG2	Cytotoxicity assay		IC50 = 0.08 μM	21875764
HT-29	Cytotoxicity assay		IC50 = 0.38 μM	21875764
A375	Cytotoxicity assay		IC50 = 0.81 μM	21875764
MCF7	Cytotoxicity assay		IC50 = 1.3 μM	21875764
BGC823	Cytotoxicity assay		IC50 = 1.5 μM	21875764
769-P	Cytotoxicity assay		IC50 = 7.1 μM	21875764
BGC823	Cytotoxicity assay		IC50 = 0.00329 μM	21928797
HT-29	Cytotoxicity assay		IC50 = 0.00394 μM	21928797
HepG2	Cytotoxicity assay		IC50 = 0.0044 μM	21928797
A375	Cytotoxicity assay		IC50 = 0.0049 μM	21928797
A549	Cytotoxicity assay		IC50 = 0.0449 μM	21928797
NCI-H460	Cytotoxicity assay		IC50 = 8 μM	21942765
HBL100	Growth inhibition assay		GI50 = 0.000017 μM	21986585
HeLa	Growth inhibition assay		GI50 = 0.000033 μM	21986585
T47D	Growth inhibition assay		GI50 = 0.00015 μM	21986585
WiDr	Growth inhibition assay		GI50 = 0.00022 μM	21986585
A2780	Growth inhibition assay		GI50 = 0.00027 μM	21986585
SW1573	Growth inhibition assay		GI50 = 0.005 μM	21986585
A2780	Antiproliferative activity assay		IC50 = 0.017 μM	21995542
DU145	Cytotoxicity assay		EC50 = 0.0059 μM	22142543
KB	Cytotoxicity assay		EC50 = 0.006 μM	22142543
A549	Cytotoxicity assay		EC50 = 0.0064 μM	22142543
SKOV3	Cytotoxicity assay		IC50 = 0.0001 μM	22506620
BGC823	Cytotoxicity assay		IC50 = 0.0033 μM	22506620
HepG2	Cytotoxicity assay		IC50 = 0.0044 μM	22506620
A549	Cytotoxicity assay		IC50 = 0.016 μM	22506620
HCT8	Cytotoxicity assay		IC50 = 0.051 μM	22506620
HCT116	Cytotoxicity assay		IC50 = 0.05 μM	22691179
SKBR3	Cytotoxicity assay		IC50 = 0.11 μM	22691179
SK-MEL-5	Cytotoxicity assay		IC50 = 0.15 μM	22691179
SKOV3	Cytotoxicity assay		IC50 = 0.4 μM	22691179
MCF7	Cytotoxicity assay		IC50 = 0.9 μM	22691179
HeLa	Cytotoxicity assay		IC50 = 1 μM	23103097
A2780	Cytotoxicity assay		IC50 = 1.1 μM	23103097
MES-SA	Cytotoxicity assay		IC50 = 0.003 μM	23141916
NUGC3	Growth inhibition assay		GI50 = 0.02 μM	23167614
HONE1	Growth inhibition assay		GI50 = 0.02 μM	23167614
NCI-H460	Growth inhibition assay		GI50 = 0.03 μM	23167614
MCF7	Growth inhibition assay		GI50 = 0.03 μM	23167614
A549	Growth inhibition assay		GI50 = 0.06 μM	23167614
HepG2	Growth inhibition assay		GI50 = 0.18 μM	23167614
OVCAR8	Cytotoxicity assay		IC50 = 0.005 μM	23214452
NCI/ADR-RES	Cytotoxicity assay		IC50 = 3.3 μM	23214452
DU145	Growth inhibition assay		GI50 = 0.0065 μM	23274123
KB	Growth inhibition assay		GI50 = 0.00777 μM	23274123
A549	Growth inhibition assay		GI50 = 0.00818 μM	23274123
KBVIN	Growth inhibition assay		GI50 = 1.803 μM	23274123
K562	Antiproliferative activity assay		IC50 = 0.41 μM	23274570
CaEs17	Antiproliferative activity assay		IC50 = 0.43 μM	23274570
MGC803	Antiproliferative activity assay		IC50 = 0.85 μM	23274570
Bel7402	Antiproliferative activity assay		IC50 = 1.89 μM	23274570
HT-29	Cytotoxicity assay		ED50 = 0.001 μM	23301897
NCI-H358	Cytotoxicity assay		IC50 = 0.01 μM	23425970
A2780S	Cytotoxicity assay		IC50 = 0.02 μM	23425970
DU145	Cytotoxicity assay		IC50 = 0.03 μM	23425970
SKOV3	Cytotoxicity assay		IC50 = 0.1 μM	23425970
ES2	Cytotoxicity assay		IC50 = 0.1 μM	23425970
HCT15	Cytotoxicity assay		IC50 = 0.12 μM	23425970
PC3	Cytotoxicity assay		IC50 = 0.14 μM	23425970
SKHEP1	Cytotoxicity assay		IC50 = 0.24 μM	23425970
HT-29	Cytotoxicity assay		IC50 = 0.45 μM	23425970
MCF7	Cytotoxicity assay		IC50 = 0.66 μM	23425970
C26	Cytotoxicity assay		IC50 = 1.05 μM	23425970
SPC-A1	Cytotoxicity assay		IC50 = 5.3 μM	23425970
A2780	Cytotoxicity assay		IC50 = 8.25 μM	23425970
A2780	Cytotoxicity assay		IC50 = 0.001 μM	23547884
BGC823	Cytotoxicity assay		IC50 = 0.001 μM	23547884
Bel7402	Cytotoxicity assay		IC50 = 0.006 μM	23547884
A549	Cytotoxicity assay		IC50 = 0.016 μM	23547884
HCT8	Cytotoxicity assay		IC50 = 0.051 μM	23547884
A2780	Cytotoxicity assay		IC50 = 0.028 μM	23659371
HCT116	Cytotoxicity assay		GI50 = 0.01 μM	23725535
T47D	Cytotoxicity assay		GI50 = 0.01 μM	23725535
LOXIMVI	Cytotoxicity assay		GI50 = 0.016 μM	23725535
OVCAR3	Cytotoxicity assay		GI50 = 0.02 μM	23725535
DU145	Cytotoxicity assay		GI50 = 0.032 μM	23725535
MOLT4	Cytotoxicity assay		GI50 = 0.032 μM	23725535
SNB19	Cytotoxicity assay		GI50 = 0.04 μM	23725535
NCI-H322M	Cytotoxicity assay		GI50 = 0.05 μM	23725535
RXF393	Cytotoxicity assay		GI50 = 0.05 μM	23725535
2008	Growth inhibition assay		GI50 = 0.003 μM	23750455
MES-SA	Growth inhibition assay		GI50 = 0.004 μM	23750455
MES-SA/Dx5	Growth inhibition assay		GI50 = 0.75 μM	23750455
2008/17/4	Growth inhibition assay		GI50 = 2 μM	23750455
MOLT4	Cytotoxicity assay		IC50 = 0.0018 μM	23806112
U937	Cytotoxicity assay		IC50 = 0.0019 μM	23806112
BGC823	Cytotoxicity assay		IC50 = 0.0035 μM	23806112
A549	Cytotoxicity assay		IC50 = 0.0036 μM	23806112
K562	Cytotoxicity assay		IC50 = 0.0049 μM	23806112
MCF7	Cytotoxicity assay		IC50 = 0.005 μM	23806112
DU145	Cytotoxicity assay		GI50 = 0.006 μM	23867604
KB	Cytotoxicity assay		GI50 = 0.0064 μM	23867604
A549	Cytotoxicity assay		GI50 = 0.0076 μM	23867604
KBVIN	Cytotoxicity assay		GI50 = 1.21 μM	23867604
HL60	Cytotoxicity assay		IC50 = 0.002 μM	23937981
DU145	Cytotoxicity assay		IC50 = 0.005 μM	23937981
MES-SA	Cytotoxicity assay		IC50 = 0.005 μM	23937981
MDA435	Cytotoxicity assay		IC50 = 0.005 μM	23937981
Bowes	Cytotoxicity assay		IC50 = 0.005 μM	23937981
A549	Cytotoxicity assay		IC50 = 0.01 μM	23937981
Clone A	Cytotoxicity assay		IC50 = 0.5 μM	23937981
MIP101	Cytotoxicity assay		IC50 = 1.1 μM	23937981
PBMC	Cytotoxicity assay		IC50 = 5 μM	23937981
39SK	Cytotoxicity assay		IC50 = 5 μM	23937981
MCF7	Cytotoxicity assay		IC50 = 3.1 μM	24195466
DU145	Cytotoxicity assay		GI50 = 0.006 μM	24315191
A549	Cytotoxicity assay		GI50 = 0.0076 μM	24315191
KB	Cytotoxicity assay		GI50 = 0.008 μM	24315191
KBVIN	Cytotoxicity assay		GI50 = 1.8 μM	24315191
MCF7	Growth inhibition assay		GI50 = 0.00129 μM	24405702
Bel7402	Growth inhibition assay		GI50 = 0.001792 μM	24405702
MOLT4	Growth inhibition assay		GI50 = 0.002232 μM	24405702
A431	Growth inhibition assay		GI50 = 0.002355 μM	24405702
U937	Growth inhibition assay		GI50 = 0.002392 μM	24405702
PANC1	Growth inhibition assay		GI50 = 0.002409 μM	24405702
SGC7901	Growth inhibition assay		GI50 = 0.003088 μM	24405702
HeLa	Growth inhibition assay		GI50 = 0.003206 μM	24405702
BGC823	Growth inhibition assay		GI50 = 0.003605 μM	24405702
HT1080	Growth inhibition assay		GI50 = 0.003889 μM	24405702
DU145	Growth inhibition assay		GI50 = 0.005568 μM	24405702
K562	Growth inhibition assay		GI50 = 0.007014 μM	24405702
A549	Growth inhibition assay		GI50 = 0.01873 μM	24405702
HuH7	Growth inhibition assay		GI50 = 0.2067 μM	24405702
HeLa	Cytotoxicity assay		IC50 = 0.0025 μM	24422592
DU145	Cytotoxicity assay		GI50 = 0.006 μM	24502232
KB	Cytotoxicity assay		GI50 = 0.0064 μM	24502232
A549	Cytotoxicity assay		GI50 = 0.0076 μM	24502232
KBVIN	Cytotoxicity assay		GI50 = 1.21 μM	24502232
A2780	Cytotoxicity assay		IC50 = 0.00138 μM	24680057
1A9PTX22	Cytotoxicity assay		IC50 = 0.1607 μM	24680057
1A9PTX10	Cytotoxicity assay		IC50 = 0.53295 μM	24680057
BCG823	Cytotoxicity assay		IC50 = 0.0028 μM	24684840
HepG2	Cytotoxicity assay		IC50 = 0.0064 μM	24684840
HL-7702	Cytotoxicity assay		IC50 = 0.0518 μM	24684840
NCI-ADR-RES	Cytotoxicity assay		EC50 = 0.013 μM	24801610
OVCAR8	Cytotoxicity assay		EC50 = 0.018 μM	24801610
HeLa	Antiproliferative activity assay		IC50 = 0.00121 μM	24890652
MDA-MB-435	Antiproliferative activity assay		IC50 = 0.00193 μM	24890652
SKOV3	Antiproliferative activity assay		IC50 = 0.003 μM	24890652
SKOV3	Cytotoxicity assay		GI50 = 0.0047 μM	24893224
P-gp expressing SKOV3-M6/6	Cytotoxicity assay		GI50 = 0.6 μM	24893224
HT-29	Cytotoxicity assay		IC50 = 0.001 μM	24937209
MCF7	Cytotoxicity assay		IC50 = 0.0015 μM	24960143
HepG2	Cytotoxicity assay		IC50 = 0.0046 μM	24960143
MDA-MB-231	Cytotoxicity assay		IC50 = 0.0082 μM	24960143
HL7702	Cytotoxicity assay		IC50 = 1.1 μM	24960143
A2780	Cytotoxicity assay		IC50 = 0.0004 μM	25047938
HeLa	Cytotoxicity assay		IC50 = 0.0007 μM	25047938
MCF7	Cytotoxicity assay		IC50 = 0.0017 μM	25047938
1A9	Cytotoxicity assay		IC50 = 0.0039 μM	25047938
1A9/A8	Cytotoxicity assay		IC50 = 0.0042 μM	25047938
1A9PTX22	Cytotoxicity assay		IC50 = 0.0328 μM	25047938
1A9PTX10	Cytotoxicity assay		IC50 = 0.0814 μM	25047938
MCF7/R	Cytotoxicity assay		IC50 = 0.299 μM	25047938
A2780AD	Cytotoxicity assay		IC50 = 1.244 μM	25047938
KB	Antiproliferative activity assay		IC50 = 0.0033 μM	25059503
KB-7d	Antiproliferative activity assay		IC50 = 0.0079 μM	25059503
KB-S15	Antiproliferative activity assay		IC50 = 0.273 μM	25059503
COLO205	Cytotoxicity assay		IC50 = 0.003 μM	25091926
NCI-H460	Cytotoxicity assay		IC50 = 0.01 μM	25091926
DU145	Cytotoxicity assay		IC50 = 1.5 μM	25105722
MCF7	Cytotoxicity assay		IC50 = 1.8 μM	25105722
HeLa	Cytotoxicity assay		IC50 = 5 μM	25105722
PANC1	Cytotoxicity assay		IC50 = 1.18 μM	25466201
HeLa	Cytotoxicity assay		IC50 = 1.3 μM	25466201
Calu1	Cytotoxicity assay		IC50 = 1.33 μM	25466201
H460	Cytotoxicity assay		IC50 = 1.43 μM	25466201
HCT116	Cytotoxicity assay		IC50 = 1.55 μM	25466201
ACHN	Cytotoxicity assay		IC50 = 2.33 μM	25466201
HeLa	Growth inhibition assay		IC50 = 0.0035 μM	25685941
DU145	Growth inhibition assay		IC50 = 0.004 μM	25685941
PC3	Growth inhibition assay		IC50 = 0.04 μM	25685941
SKOV3	Growth inhibition assay		IC50 = 6.2 μM	25685941
Hep3B2	Cytotoxicity assay		IC50 = 0.000016 μM	25760674
PANC1	Cytotoxicity assay		IC50 = 0.0011 μM	25760674
CNE1-LMP1	Cytotoxicity assay		IC50 = 0.0042 μM	25760674
MGC	Cytotoxicity assay		IC50 = 0.0064 μM	25760674
A375	Cytotoxicity assay		IC50 = 0.0089 μM	25760674
MCF7	Cytotoxicity assay		IC50 = 0.014 μM	25760674
HaCaT	Cytotoxicity assay		IC50 = 0.024 μM	25760674
A549	Cytotoxicity assay		IC50 = 0.03 μM	25760674
EC109	Cytotoxicity assay		IC50 = 0.14 μM	25760674
NIH/3T3	Cytotoxicity assay		IC50 = 4.2 μM	25760674
DU145	Antiproliferative activity assay		GI50 = 0.0057 μM	25770782
KB	Antiproliferative activity assay		GI50 = 0.0064 μM	25770782
A549	Antiproliferative activity assay		GI50 = 0.0071 μM	25770782
KBVIN	Antiproliferative activity assay		GI50 = 0.95 μM	25770782
DU145	Antiproliferative activity assay		GI50 = 0.006 μM	26242242
KB	Antiproliferative activity assay		GI50 = 0.0064 μM	26242242
A549	Antiproliferative activity assay		GI50 = 0.0076 μM	26242242
vincristine-resistant KBVIN	Antiproliferative activity assay		GI50 = 1.21 μM	26242242
K562	Cytotoxicity assay		IC50 = 0.9 μM	26287401
A549	Cytotoxicity assay		IC50 = 0.0063 μM	26448037
cells after 48 hrs by SRB assay	Cytotoxicity assay		GI50 = 0.00148 μM	26462052
cells assessed as cell growth inhibition after 48 hrs by MTT assay	Cytotoxicity assay		IC50 = 0.65 μM	26638041
MCF7	Cytotoxicity assay		IC50 = 0.0006 μM	27441892
HCT116	Cytotoxicity assay		IC50 = 0.0009 μM	27441892
BGC823	Cytotoxicity assay		IC50 = 0.0033 μM	27441892
HepG2	Cytotoxicity assay		IC50 = 0.012 μM	27441892
Capan2	Cytotoxicity assay		IC50 = 0.017 μM	27441892
A375	Cytotoxicity assay		IC50 = 0.022 μM	27441892
A549	Cytotoxicity assay		IC50 = 0.023 μM	27441892
A2780	Cytotoxicity assay		IC50 = 0.038 μM	27441892
NCI-H1650	Cytotoxicity assay		IC50 = 0.068 μM	27441892
MDA-MB-435	Antiproliferative activity assay		GI50 = 0.001 μM	28112516
HepG2	Cytotoxicity assay		IC50 = 0.3 μM	28262527
Hep3B	Cytotoxicity assay		IC50 = 0.73 μM	28262527
KB	Antiproliferative activity assay		IC50 = 0.0059 μM	28457756
A549	Antiproliferative activity assay		IC50 = 0.00685 μM	28457756
MDA-MB-231	Antiproliferative activity assay		IC50 = 0.00963 μM	28457756
MCF7	Antiproliferative activity assay		IC50 = 0.01146 μM	28457756
KBVIN	Antiproliferative activity assay		IC50 = 2.035 μM	28457756
1A9	Cytotoxicity assay		IC50 = 0.00371 μM	28850227
A549	Growth inhibition assay		IC50 = 0.0071 μM	29439899
A549-T24	Growth inhibition assay		IC50 = 0.07 μM	29439899
HCT116	Cytotoxicity assay		IC50 = 0.0338 μM	29468872
HeLa	Antiproliferative activity assay		IC50 = 0.0016 μM	29655610
SKOV3	Antiproliferative activity assay		IC50 = 0.003 μM	29655610
SKOV3-MDR1-M6/6	Antiproliferative activity assay		IC50 = 2.6 μM	29655610
点击查看更多细胞系数据

生物活性

产品描述

Paclitaxel是一种microtubule聚合物稳定剂，在人内皮细胞中IC50为0.1 pM。Paclitaxel可引起有丝分裂停滞和细胞凋亡。 Paclitaxel还会诱导自噬。

特性

Paclitaxel 是有丝分裂抑制剂。

靶点

Microtubule (human endothelial cells) ^[1]

0.1 pM

体外研究(In Vitro)
体外研究活性	Paclitaxel在10⁴到 10⁵倍更高浓度时，抑制非内皮性人类细胞，IC50 为1 nM -10 nM。Paclitaxel选择性抑制细胞增殖，具有种属特异性，在Paclitaxel极低浓度时，小鼠内皮细胞对 Paclitaxel不敏感。极低浓度Paclitaxel抑制人类内皮细胞，但是不影响细胞微管结构，且处理的细胞在 G2/M 期没有出现细胞周期停滞和凋亡，说明这是一种新型尚未查明的作用机制。在体外血管生成实验中，在三维纤维蛋白基质中，极低浓度Paclitaxel阻断人类内皮细胞形成芽管。^[1] 在SMF存在时, Paclitaxel 作用于 K562 细胞的有效浓度从50 ng/ml降低到 10 ng/ml。在有或无SMF时，Paclitaxel 使K562 细胞周期停滞与DNA损伤相关。^[2] Paclitaxel单独处理四种细胞系，包括A549 细胞,H358, H1395 细胞和H1666 细胞，抑制CDK1，这种作用存在时间依赖性。^[3]
细胞实验	细胞系	细胞，包括人类新生儿皮肤微血管内皮细胞(HMVECs), 人脐静脉内皮细胞(HUVECs), 人脐动脉内皮细胞 (HUAVECs), 正常人类星形胶质细胞(NHAs), 正常人体皮肤成纤维细胞(NHDFs), 正常人表皮角质形成细胞(NHEKs), 人类乳腺上皮细胞(HMEpCs), 人前列腺上皮细胞(PrEpCs) 和人脐动脉平滑肌细胞(UASMCs)
	浓度	0.1 pM-100 pM
	孵育时间	72 小时
	方法	培养细胞，包括人类新生儿皮肤微血管内皮细胞(HMVECs), 人脐静脉内皮细胞(HUVECs), 人脐动脉内皮细胞 (HUAVECs), 正常人类星形胶质细胞(NHAs), 正常人体皮肤成纤维细胞(NHDFs), 正常人表皮角质形成细胞(NHEKs), 人类乳腺上皮细胞(HMEpCs), 人前列腺上皮细胞(PrEpCs) 和人脐动脉平滑肌细胞(UASMCs)。在96孔板中使用6和12通道的细胞进行增殖。细胞按每孔3000–5000个细胞接种，然后粘附4小时。Paclitaxel在培养基中稀释，然后按一式四份加到孔中，细胞温育3天，然后加入MTS 试剂，然后定量测量每孔中的活细胞。
实验图片	检测方法	检测指标	实验图片	PMID
	Western blot	p-ERK / ERK MARCKS (pSer159/163) Src (pTyr416) p-JAK2 / p-STAT3 / p-AKT / p-MAPK / Bcl-xl / MCL-1 Id1 MARCKS		20068074
	Growth inhibition assay	Cell viability		28823711
	Immunofluorescence	α-tubulin Rab11a/BV9		22904633

体内研究(In Vivo)
体内研究活性	Paclitaxel单独处理 BC-V 和 BC-ER肿瘤的抑制定额分别为49.78 和 51.23%。20 mg/kg Paclitaxel处理6个周期，显著降低Ki-67阳性细胞百分比,BC-V肿瘤中降到20.4%，BC-ER 肿瘤中降到25.1%。^[4]

NCT Number	Recruitment	Conditions	Sponsor/Collaborators	Start Date	Phases
临床试验信息 (data from https://clinicaltrials.gov, updated on 2024-05-22)
NCT05312372	Withdrawn	Esophageal Squamous Cell Carcinoma	Institut de Recherches Internationales Servier\|ADIR a Servier Group company\|Servier	May 2025	Phase 1\|Phase 2
NCT04715542	Not yet recruiting	Chemotherapy Induced Peripheral Neuropathy (CIPN)	University of Bern\|Insel Gruppe AG University Hospital Bern\|Hospital of Thun\|Tumor- und Brustzentrum ZeTuP St.Gallen\|Gesundheitszentrum Fricktal AG\|Kantonsspital Winterthur KSW\|Kantonsspital Graubünden\|Kantonsspital Aarau	August 2024	Phase 3
NCT06387901	Not yet recruiting	Breast Cancer\|Paclitaxel Adverse Reaction\|Chemotherapeutic Toxicity\|Chemotherapeutic Agent Toxicity\|Body Weight\|Physical Inactivity	Universitair Ziekenhuis Brussel\|Vrije Universiteit Brussel\|University Ghent	May 6 2024	--
NCT05826015	Not yet recruiting	Recurrent High Grade Uterine Cancer	Washington University School of Medicine\|National Cancer Institute (NCI)\|Aravive Inc.	May 31 2024	Phase 1
NCT05695313	Recruiting	Breast Cancer	Centre Georges Francois Leclerc	April 12 2024	Phase 2

参考文献
[1] Wang J, et al. Anticancer Drugs. 2003, 14(1), 13-19. [2] Sun RG, et al. Gen Physiol Biophys. 2012, 31(1), 1-10. [3] Zhang XH, et al. Cancer Lett. 2012, 322(2), 213-222. [4] Chang J, et al. Breast Cancer Res Treat. 2012. [5] Dziadyk JM, et al. Anticancer Res. 2004 Jan-Feb;24(1):27-36. + 展开

参考文献

+ 展开

化学信息&溶解度

分子量	853.91	分子式	C₄₇H₅₁NO₁₄
CAS号	33069-62-4	SDF	Download Paclitaxel SDF
Smiles	CC1=C2C(C(=O)C3(C(CC4C(C3C(C(C2(C)C)(CC1OC(=O)C(C(C5=CC=CC=C5)NC(=O)C6=CC=CC=C6)O)O)OC(=O)C7=CC=CC=C7)(CO4)OC(=O)C)O)C)OC(=O)C
储存条件(自收到货起)	3年-20°C粉状	储备液保存和期限建议分装储备液，避免反复冻融！	1年-80°C溶于溶剂
储存条件(自收到货起)	3年-20°C粉状	储备液保存和期限建议分装储备液，避免反复冻融！	1个月-20°C溶于溶剂

体外溶解度
批次：

DMSO : 100 mg/mL ( (117.1 mM) ；DMSO吸湿会降低化合物溶解度，请使用新开封DMSO)

Ethanol : 23 mg/mL (26.93 mM)

Water : Insoluble

DMSO : 100 mg/mL ( (117.1 mM) ；DMSO吸湿会降低化合物溶解度，请使用新开封DMSO)

Ethanol : 20 mg/mL (23.42 mM)

Water : Insoluble

DMSO : 100 mg/mL ( (117.1 mM) ；DMSO吸湿会降低化合物溶解度，请使用新开封DMSO)

Ethanol : 90 mg/mL (105.39 mM)

Water : Insoluble

DMSO : 100 mg/mL ( (117.1 mM) ；DMSO吸湿会降低化合物溶解度，请使用新开封DMSO)

Ethanol : 100 mg/mL (117.1 mM)

Water : Insoluble

摩尔浓度计算器

体内溶解度
批次：

现配现用，请按从左到右的顺序依次添加，澄清后再加入下一溶剂

动物体内配方计算器

实验计算

摩尔浓度计算器

质量	浓度	体积	分子量
=	×	×

稀释计算器分子量计算器

动物体内配方计算器（澄清溶液）

第一步：请输入基本实验信息（考虑到实验过程中的损耗，建议多配一只动物的药量）

给药剂量 mg/kg 动物平均体重 g 每只动物给药体积 μL 动物数量只

第二步：请输入动物体内配方组成（配方适用于不溶于水的药物；不同批次药物配方比例不同，请联系Selleck为您提供正确的澄清溶液配方）

% DMSO + % + % Tween 80 + % ddH2O

%DMSO+ %

计算结果：

工作液浓度： mg/ml；

DMSO母液配制方法： mg 药物溶于μL DMSO溶液（母液浓度mg/mL，注：如该浓度超过该批次药物DMSO溶解度，请先联系Selleck）；

体内配方配制方法：取μL DMSO母液，加入μL PEG300，混匀澄清后加入μL Tween 80，混匀澄清后加入μL ddH₂O，混匀澄清。

体内配方配制方法：取μL DMSO母液，加入μL Corn oil，混匀澄清。

注意：1. 首先保证母液是澄清的；
2.一定要按照顺序依次将溶剂加入，进行下一步操作之前必须保证上一步操作得到的是澄清的溶液，可采用涡旋、超声或水浴加热等物理方法助溶。

技术支持

在订购、运输、储存和使用我们的产品的任何阶段，您遇到的任何问题，均可以通过拨打我们的热线电话400-668-6834，或者技术支持邮箱tech@selleck.cn，直接联系到我们。我们会在24小时内尽快联系您。

操作手册

如果有其他问题，请给我们留言。

* 必填项

常见问题及建议解决方法

问题 1:
I am interested in the product S1150 for in vivo studies, could you please give some suggestions for the formulation?

回答：
S1150 in 1% DMSO+30% polyethylene glycol+1% Tween 80 at 30mg/ml is a suspension. If the you want to inject it, there is another vehicle, 5% DMSO+5% Tween 80+ddH2O. S1150 can dissolve in it at 2.5mg/ml as a clear solution. It is a common formulation we used, but is not cited from reference.

问题 2:
the compound was dissolved into 1ml DMSO and diluted with 1x PBS or water (500ul + 9.5 ml PBS or water). I found the white precipitation goes out. How to figure it out?

回答：
Paclitaxel has very low solubility in water based solution and that's why it precipitated out once you dilute the stock with water. The vehicle we suggest is: 1% DMSO+30% polyethylene glycol+1% Tween 80.

C1=C0/X	C1:	LOG(C1):
C2=C1/X	C2:	LOG(C2):
C3=C2/X	C3:	LOG(C3):
C4=C3/X	C4:	LOG(C4):
C5=C4/X	C5:	LOG(C5):
C6=C5/X	C6:	LOG(C6):
C7=C6/X	C7:	LOG(C7):
C8=C7/X	C8:	LOG(C8):