- MCT1
- MCT4
- MCT2
MCT4 选择性抑制剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S9929 | VB124 | VB124, a potent and selective MCT4 inhibitor, specifically inhibits lactate efflux/import in MDA-MB-231 cells expressing MCT4, and is used for the research of cardiac hypertrophy, heart failure, and metabolism. | Selective | MCT4, IC50: 8.6 nM; MCT4, IC50: 19 nM |
| S9907 | Syrosingopine | Syrosingopine is a dual MCT1 and MCT4 inhibitor with IC50 values of 2500nM and 40 nM in HAP1 cells, respectively. | Selective | MCT4, IC50: 40 nM |
