MEK1
MEK1/2
MEK2
MEK5

MEK5 选择性抑制剂

目录号	产品名	产品描述	Selective / Pan	IC50 / Ki
S1531	BIX 02189	BIX02189 is a selective inhibitor of MEK5 with IC50 of 1.5 nM, also inhibits ERK5 catalytic activity with IC50 of 59 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.	Selective	MEK5, IC50: 1.5 nM
S1530	BIX 02188	BIX02188 is a selective inhibitor of MEK5 with IC50 of 4.3 nM, also inhibits ERK5 catalytic activity with IC50 of 810 nM, and does not inhibit closely related kinases MEK1, MEK2, ERK2, and JNK2.	Selective	MEK5, IC50: 4.3 nM