- PGD1
- PGD2
- PGE2
- PGE4
- PGF2α
- PGI2
- TXA2
- TXB2
PGD1 选择性激动剂 | 拮抗剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S0099 | Asapiprant | Asapiprant(S-555739) is a potent and selective DP1 receptor antagonist with a Ki of 0.44 nM, which has potential as a novel therapy for allergic airway diseases. | Selective | DP1, Ki: 0.44 nM |
| S0325 | Treprostinil sodium | Treprostinil sodium (UT-15, Remodulin, Orenitram, Tyvaso, Trevyent) is a potent agonist of DP1, EP2 and IP receptors with Ki 4.4 nM, 3.6 nM and 32 nM, respectively. | Pan | DP1, Ki: 4.4 nM |
