- NMDA receptor
- AMPA receptor
- mGluR2
- mGluR3
- mGluR4
- mGluR5
mGluR3 激动剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S6001 | pomaglumetad (LY404039) | LY404039 is a potent agonist of recombinant human mGlu2/mGlu3 receptors with Ki of 149 nM/92 nM, shows >100-fold selectivity over ionotropic glutamate receptors, glutamate transporters, and other receptors. Phase 3. | Pan | Recombinant human mGlu3, Ki: 92 nM; Rat neurons expressing native mGlu2/3, Ki: 88 nM |
