MCT1
MCT4
MCT2

MCT1 选择性抑制剂

目录号	产品名	产品描述	Selective / Pan	IC50 / Ki
S6732	7ACC2	7ACC2 is a potent inhibitor of mitochondrial pyruvate transport 1 (MCT1) with an IC50 value of 10 nM for lactate uptake in SiHa human cervix carcinoma cells.	Selective
S7339	AZD3965	AZD3965 is a potent, selective and orally available monocarboxylate transporter 1 (MCT1) inhibitor with a binding affinity of 1.6 nM, 6-fold selective over MCT2. Phase 1.	Selective
S7919	AR-C155858	AR-C155858 is a selective monocarboxylate transporter MCT1 and MCT2 inhibitor with Ki value of 2.3 nM and 10 nM, respectively.	Pan	MCT1, Ki: 2.3 nM
S9907	Syrosingopine	Syrosingopine is a dual MCT1 and MCT4 inhibitor with IC50 values of 2500nM and 40 nM in HAP1 cells, respectively.	Pan	MCT1, IC50: 2500 nM