| S9805 |
WM-3835 |
WM-3835 is a novel and high-specific small molecule Lysine Acetyltransferase 7 (KAT7, MYST2, HBO1) inhibitor, able to potently suppressed OS cell proliferation and migration, and leads to apoptosis activation. |
Selective |
|
| S8776 |
WM-1119 |
WM-1119 is a highly potent, selective inhibitor of lysine acetyltransferase KAT6A with IC50 of 0.25 μM. It is 1,100-fold and 250-fold more active against KAT6A than against KAT5 or KAT7, respectively. |
Selective |
KAT6A, Kd: 0.002 μM; KAT5, Kd: 2.2 μM; KAT7, Kd: 0.5 μM |
| S6655 |
WM-8014 |
WM-8014 is a highly potent inhibitor of histone acetyltransferase KAT6A with an IC50 of 8 nM. |
Selective |
KAT6A, IC50: 8 nM |
| S7476 |
MG149 |
MG149 (Tip60 HAT inhibitor) is a potent histone acetyltransferase inhibitor with IC50 of 74 μM and 47 μM for Tip60 and MOF,respectively.
|
Selective |
Tip60, IC50: 74 μM; MOF, IC50: 47 μM |
| s7582 |
Anacardic Acid |
Anacardic Acid (6-pentadecylsalicylic Acid) is a potent inhibitor of p300 and p300/CBP-associated factor histone acetyltranferases, which also has antibacterial activity, antimicrobial activity,
prostaglandin synthase inhibition, and tyrosinase and lipoxygenase inhibition.
|
Pan |
|
