Axitinib

别名: AG 013736 中文名称:阿西替尼,阿昔替尼

    Axitinib是一种多靶点抑制剂,作用于 VEGFR1VEGFR2VEGFR3,PDGFRβ和c-Kit,在猪主动脉内皮细胞中IC50分别为0.1 nM,0.2 nM,0.1-0.3 nM,1.6 nM和1.7 nM。

    Axitinib Chemical Structure

    Axitinib Chemical Structure

    CAS: 319460-85-0

    规格 价格 库存 购买数量
    10mM (1mL in DMSO) RMB 647.01 现货
    50mg RMB 570.91 现货
    100mg RMB 975.25 现货
    1g RMB 4013.1 现货
    更大包装 有超大折扣

    400-668-6834

    info@selleck.cn

    免费分装
    免费预溶

    相关VEGFR产品

    客户使用Selleck的Axitinib发表文献174篇:

    产品质控

    批次: 纯度: 99.96%
    99.96

    VEGFR抑制剂选择性比较

    细胞实验数据示例

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    LB2241-RCC M{TNR2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NXWxOlRZRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
    Detroit562 M2j4cWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MnO3QIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
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    A498 NYnBT3FrT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= M4ftWVxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5USU6JRWK8M4E,
    SK-MEL-24 M{HFR2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NWHXd3NDRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
    OVCAR-5 M{\YS2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MX:8ZUB1[XKpZYS9K39jdGGwazegbJJm\j1paIT0dJM7Ny:5d4eu[YJqNmGlLoXrM4Np\W2kbD;jc41xd3WwZG;y[ZBwenShY3Hy[E9EUEWPQlyxNlg6QTJ4Lze+V2FPT0WUPD;hQi=>
    NCI-H1792 Mlu1S5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MkXQQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
    KOSC-2 M1Hqe2dzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NGjWUpA9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;3e5cv\WKrLnHjMpVsN2OqZX3icE9kd22yb4Xu[H9z\XCxcoTfZ4Fz\C:FSFXNRmwyOjh7OUK2M{c,W0GQR1XSQE9iRg>?
    Mo-T M2fp[Gdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NW[wdVl{RGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
    CFPAC-1 NU\mOIRFT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NVjyUlJVRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
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    ML-2 M4PFOWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 NIj3e5E9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;3e5cv\WKrLnHjMpVsN2OqZX3icE9kd22yb4Xu[H9z\XCxcoTfZ4Fz\C:FSFXNRmwyOjh7OUK2M{c,W0GQR1XSQE9iRg>?
    KNS-81-FD MoXMS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? M4[3NlxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5USU6JRWK8M4E,
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    MCF7 NHjONItIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NVru[GlqRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
    P30-OHK NFXlOpVIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MnTqQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
    BPH-1 MljnS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MnzjQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
    U251 M{DhUWdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 MUi8ZUB1[XKpZYS9K39jdGGwazegbJJm\j1paIT0dJM7Ny:5d4eu[YJqNmGlLoXrM4Np\W2kbD;jc41xd3WwZG;y[ZBwenShY3Hy[E9EUEWPQlyxNlg6QTJ4Lze+V2FPT0WUPD;hQi=>
    MKN1 NG[zT2tIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= MWm8ZUB1[XKpZYS9K39jdGGwazegbJJm\j1paIT0dJM7Ny:5d4eu[YJqNmGlLoXrM4Np\W2kbD;jc41xd3WwZG;y[ZBwenShY3Hy[E9EUEWPQlyxNlg6QTJ4Lze+V2FPT0WUPD;hQi=>
    A431 NH7NUmtIem:5dHigTY5pcWKrdHnvckBCe3OjeR?= NIPMW4k9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;3e5cv\WKrLnHjMpVsN2OqZX3icE9kd22yb4Xu[H9z\XCxcoTfZ4Fz\C:FSFXNRmwyOjh7OUK2M{c,W0GQR1XSQE9iRg>?
    C8166 M{jIOGdzd3e2aDDJcohq[mm2aX;uJGF{e2G7 M3XFXVxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5USU6JRWK8M4E,
    HEL MknzS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? NYrQWJR{RGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRlODTlfFVlww[T5?
    RMG-I MkGwS5Jwf3SqIFnubIljcXSrb36gRZN{[Xl? MnXVQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
    CAL-72 NYDDfnJWT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= MlLzQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xd4f3MoVjcS6jYz71b{9kcGWvYnyvZ49ueG:3bnTfdoVxd3K2X3PhdoQwS0iHTVLMNVI5QTl{Nj:nQnNCVkeHUkyvZV4>
    SW962 NY\qcFlFT3Kxd4ToJGlvcGmkaYTpc44hSXO|YYm= NF3wbpA9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;3e5cv\WKrLnHjMpVsN2OqZX3icE9kd22yb4Xu[H9z\XCxcoTfZ4Fz\C:FSFXNRmwyOjh7OUK2M{c,W0GQR1XSQE9iRg>?
    MCF7 NH20[o1CdnSrcILvcIln\XKjdHn2[UBie3OjeR?= NVPCR4RvPSCmYYnz MkXGQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjN6Mkm1OFkoRjJ|OEK5OVQ6RC:jPh?=
    MDA-MB-468 MYrBcpRqeHKxbHnm[ZJifGm4ZTDhd5NigQ>? NGPiXJY2KGSjeYO= NYPp[WgyRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:vdJVjdWWmLn7jZokvdmyvLn7pbE5od3ZxMkO4Nlk2PDlpPkKzPFI6PTR7PD;hQi=>
    HCC1954 MYnBcpRqeHKxbHnm[ZJifGm4ZTDhd5NigQ>? NXjLXXRTPSCmYYnz NFPvd4s9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{M{iyPVU1QSd-MkO4Nlk2PDl:L3G+
    SKBR3 Ml7hRY51cXC{b3zp[oVz[XSrdnWgZZN{[Xl? MUe1JIRigXN? NFK5ZYU9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{M{iyPVU1QSd-MkO4Nlk2PDl:L3G+
    MDA-MB-231 NFLhWm9CdnSrcILvcIln\XKjdHn2[UBie3OjeR?= M3zxNlUh\GG7cx?= NHSyT489[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{M{iyPVU1QSd-MkO4Nlk2PDl:L3G+
    MCF7 M2jzcmN6fG:2b4jpZ4l1gSCjc4PhfS=> NIewdGk2KGSjeYO= MkK5QIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjR6Nke0NFMoRjJ2OE[3OFA{RC:jPh?=
    MDA-MB-468 NEXTUY1EgXSxdH;4bYNqfHliYYPzZZk> M1XqdVUh\GG7cx?= M2fQblxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4D1Zo1m\C6wY3LpMo5tdS6waXiu[493NzJ2OE[3OFA{Lz5{NEi2O|QxOzxxYU6=
    SKBR3 NGjIZYtEgXSxdH;4bYNqfHliYYPzZZk> NH7HWmU2KGSjeYO= NHzpTok9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{NEi2O|QxOyd-MkS4Olc1ODN:L3G+
    MDA-MB-231 M2X3ZWN6fG:2b4jpZ4l1gSCjc4PhfS=> NFzr[5g2KGSjeYO= NI\tNIo9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{NEi2O|QxOyd-MkS4Olc1ODN:L3G+
    Saos-2 M12wdpFJXFNiYYPzZZk> M3jsb|xiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4D1Zo1m\C6wY3LpMo5tdS6waXiu[493NzJ7NEO1NVM6Lz5{OUSzOVE{QTxxYU6=
    BT-12 NH3icWpyUFSVIHHzd4F6 Mor0QIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjl2M{WxN|koRjJ7NEO1NVM6RC:jPh?=
    OHS-50 Mle3dWhVWyCjc4PhfS=> NVPjZXNpRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:vdJVjdWWmLn7jZokvdmyvLn7pbE5od3ZxMkm0N|UyOzlpPkK5OFM2OTN7PD;hQi=>
    SJ-GBM2 NXrrbIRueUiWUzDhd5NigQ>? MmfxQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjl2M{WxN|koRjJ7NEO1NVM6RC:jPh?=
    SK-N-MC NYLKT5oxeUiWUzDhd5NigQ>? NXSxOVB[RGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:vdJVjdWWmLn7jZokvdmyvLn7pbE5od3ZxMkm0N|UyOzlpPkK5OFM2OTN7PD;hQi=>
    NB-EBc1 NHO4N49yUFSVIHHzd4F6 MmrPQIEhfGG{Z3X0QUdg[myjbnunJIhz\WZ;J3j0eJB{Qi9xcIXicYVlNm6lYnmucoxuNm6raD7nc5YwOjl2M{WxN|koRjJ7NEO1NVM6RC:jPh?=
    Rh18 M3HqU5FJXFNiYYPzZZk> NIi1e5Q9[SC2YYLn[ZQ:L1:kbHHub{chcHKnZk2nbJR1eHN8Lz;weYJu\WRwbnPibU5vdG1wbnnoModwfi9{OUSzOVE{QSd-Mkm0N|UyOzl:L3G+
    HUVEC NXHCdHVySW62aYDyc4xq\mW{YYTpeoUh[XO|YYm= NE\FXIIyKGi{ M1vDS|xiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5EcEWPQly8M4E,
    HUVEC NEfyOXRCdnSrcILvcIln\XKjdHn2[UBie3OjeR?= MoXuNUBpeg>? M2T3dVxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5EcEWPQly8M4E,
    A549 M1rpb2FvfGmycn;sbYZmemG2aY\lJIF{e2G7 NXjycFNCPDhiaILz M2fYclxiKHSjcnfleF0oZ2KuYX7rK{BpemWoPTfoeJRxezpxL4f3e{5m[mlwYXOueYsw[2inbXLsM4NwdXCxdX7kY5JmeG:{dG;jZZJlN0OKRV3CUFEzQDl7Mk[vK|5EcEWPQly8M4E,
    HepG2 MX7BcpRqeHKxbHnm[ZJifGm4ZTDhd5NigQ>? MlLpOFghcHK| NXTsSY1oRGFidHHy[4V1RSehYnzhcosoKGi{ZX[9K4h1fHC|Oj:ve5d4NmWkaT7hZ{52cy:laHXtZoww[2:vcH;1coRgemWyb4L0Y4NiemRxQ1jFUWJNOTJ6OUmyOk8oRkOqRV3CUFww[T5?
    点击查看更多细胞系数据

    生物活性

    产品描述 Axitinib是一种多靶点抑制剂,作用于 VEGFR1VEGFR2VEGFR3,PDGFRβ和c-Kit,在猪主动脉内皮细胞中IC50分别为0.1 nM,0.2 nM,0.1-0.3 nM,1.6 nM和1.7 nM。
    特性 Axitinib与目前使用的sorafenib相比,作为二代治疗法,更有效。
    靶点
    VEGFR1/FLT1 [1]
    (Porcine aorta endothelial cells)
    VEGFR2/Flk1 [1]
    (Porcine aorta endothelial cells)
    VEGFR2/KDR [1]
    (Porcine aorta endothelial cells)
    VEGFR3 [1]
    (Porcine aorta endothelial cells)
    PDGFRβ [1]
    (Porcine aorta endothelial cells)
    点击更多
    0.1 nM 0.18 nM 0.2 nM 0.1 nM-0.3 nM 1.6 nM
    体外研究(In Vitro)
    体外研究活性 Axitinib是受体激酶抑制剂,作用于VEGFR-1, VEGFR-2,VEGFR-3, PDGFR-β和c-KIT时IC50分别为0.1 , 0.2, 0.1-0.3, 1.6 和1.7 nM 。[1]Axitinib可以阻断VEGFR的自磷酸化作用,VEGF调节的内皮细胞活力,微管形成,及下游信号。Axitinib抑制多种细胞系的增殖,如作用于IGR-N91, IGR-NB8, SH-SY5Y ,无VEGF刺激的HUVEC时IC50分别为>1000 nM, 849 nM, 274 nM和573 nM。[2]
    激酶实验 细胞受体激酶磷酸化实验
    生成过量表达全长VEGFR-2, PDGFR-β, 和KIT的PAE 细胞,及过量表达鼠VEGFR-2 (Flk-1) 或 PDGFR-α的NIH-3T3细胞。用2.5 µg/mL VEGFR-2抗体, 0.75 µg/mL anti-PDGFR-β 抗体, 0.25 µg/mL anti-PDGFR-α 抗体, 及0.5 µg/mL anti-KIT 抗体包被96孔板,每孔100ul。或者用1.20 µg/mL Flk-1抗体制成酶联免疫吸附(ELISA)捕获板。通过ELISA测定RTK的磷酸化作用。
    细胞实验 细胞系 HUVEC,SH-SY5Y, IGR-N91,和IGR-NB8细胞
    浓度 1 nM 到10 µM
    孵育时间 72小时
    方法 HUVEC, SH-SY5Y, IGR-N91和IGR-NB8细胞系按5x104密度接种在96孔板上,培养24小时。加入浓度不等(1 nM到10 µM)的Axitinib。72小时后,通过 MTS四唑基底物测定细胞活力,计算IC50值。
    实验图片 检测方法 检测指标 实验图片 PMID
    Western blot p-c-kit / c-kit / p-AKT / AKT / p-ERK / ERK / p-STAT3 / STAT3 / p-STAT5 / STAT5 / p-S6K / S6K / p-S6 / S6 PARP / cleaved PARP / caspase-3 / cleaved caspase-3 31205508
    Immunofluorescence alpha-tubulin 26474283
    Growth inhibition assay Cell viability 26474283
    体内研究(In Vivo)
    体内研究活性 Axitinib抑制常位移植模型,如M24met (黑色素瘤), HCT-116 (结肠直肠癌), 和SN12C (肾细胞癌)。[1]活体研究显示,按动物体重,每千克口服处理30mg Axitinib,与没有Axitinib处理的对照组相比,实验组推迟肿瘤生长达到11.4天;且用于IGR-N91侧腹移植瘤时,与对照组(密度为49)相比实验组(密度降为21)降低血管密度。[2]Axitinib在多种肿瘤包括肾细胞癌,甲状腺癌,非小细胞肺癌,黑色素瘤中显示出单一药效活性。
    动物实验 Animal Models BT474胸腺癌细胞皮下移植到雌性免疫缺陷小鼠内(Nu/nu;8-12周大)
    Dosages 10, 30或100 mg/kg
    Administration 每天口服处理
    NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
    NCT06161558 Not yet recruiting Neoplasms National Cancer Institute (NCI)|National Institutes of Health Clinical Center (CC) January 12 2024 Phase 1
    NCT05969496 Recruiting Renal Cancer|Kidney Cancer|Renal Cell Carcinoma|Inferior Vena Cava Thrombosis University of Colorado Denver|Cancer League of Colorado December 14 2023 Phase 2
    NCT05949632 Not yet recruiting Advanced Solid Tumors Incyte Corporation December 15 2023 Phase 1|Phase 2
    NCT05904730 Enrolling by invitation Breast Cancer|Ovarian Cancer|Breast Neoplasms|Ovarian Neoplasms|BRCA Mutation|HER2-positive Breast Cancer|HER2-negative Breast Cancer|HER-2 Protein Overexpression Lynkcell Europe July 11 2023 Phase 1
    NCT05817903 Recruiting Metastatic Renal Cell Carcinoma Consorzio Oncotech|Pfizer April 18 2023 Phase 2

    化学信息&溶解度

    分子量 386.47 分子式

    C22H18N4OS

    CAS号 319460-85-0 SDF Download Axitinib SDF
    Smiles CNC(=O)C1=CC=CC=C1SC2=CC3=C(C=C2)C(=NN3)C=CC4=CC=CC=N4
    储存条件(自收到货起)

    体外溶解度
    批次:

    DMSO : 26 mg/mL (DMSO吸湿会降低化合物溶解度,请使用新开封DMSO)

    Water : Insoluble

    Ethanol : Insoluble

    摩尔浓度计算器

    体内溶解度
    批次:

    现配现用,请按从左到右的顺序依次添加,澄清后再加入下一溶剂

    动物体内配方计算器

    实验计算

    摩尔浓度计算器

    质量 浓度 体积 分子量

    动物体内配方计算器(澄清溶液)

    第一步:请输入基本实验信息(考虑到实验过程中的损耗,建议多配一只动物的药量)

    mg/kg g μL

    第二步:请输入动物体内配方组成(配方适用于不溶于水的药物;不同批次药物配方比例不同,请联系Selleck为您提供正确的澄清溶液配方)

    % DMSO % % Tween 80 % ddH2O
    %DMSO %

    计算结果:

    工作液浓度: mg/ml;

    DMSO母液配制方法: mg 药物溶于μL DMSO溶液(母液浓度mg/mL,:如该浓度超过该批次药物DMSO溶解度,请先联系Selleck);

    体内配方配制方法:μL DMSO母液,加入μL PEG300,混匀澄清后加入μL Tween 80,混匀澄清后加入μL ddH2O,混匀澄清。

    体内配方配制方法:μL DMSO母液,加入μL Corn oil,混匀澄清。

    注意:1. 首先保证母液是澄清的;
    2.一定要按照顺序依次将溶剂加入,进行下一步操作之前必须保证上一步操作得到的是澄清的溶液,可采用涡旋、超声或水浴加热等物理方法助溶。

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    常见问题及建议解决方法

    问题 1:
    We would like to store at -80℃ after it dissolved in CMC. Do you have any infomation about the suggested concentration in CMC?

    回答:
    Axitinib in 0.5% CMC at up to 30mg/ml is a suspension for oral gavage administration only. We don't suggest customer to freeze down the solution but to make fresh if possible. Customer can store it for 1-2 weeks at 4 degree for continuous use.

    VEGFR相关信号通路图

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